Medicinal Chemistry

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pp. i-vi(6)

Meet Our Editorial Board Member
pp. 427-427(1)
Author: Alves, Diego

Emerging Roles of Purinergic Signaling in Diabetes
pp. 428-438(11)
Authors: Fotino, Carmen; Dal Ben, Diego; Adinolfi, Elena

Towards the In-silico Design of New HSP90 Inhibitors: Molecular Docking and 3D-QSAR CoMFA Studies of Tetrahydropyrido [4, 3-d] Pyrimidine Derivatives as HSP90 Inhibitors
pp. 439-450(12)
Authors: Sepehri, Bakhtyar; Ghavami, Raouf

Facile Synthesis, Crystal Structure, DFT Calculation and Biological Activities of 4-(2-fluorophenyl)-3-(3-methoxybenzyl)-1H-1,2,4-triazol-5 (4H)-one (5)
pp. 451-459(9)
Authors: Saleem, Muhammad; Rafiq, Muhammad; Jeong, Yeon K.; Cho, Dae Won; Kim, Chong-Hyeak; Seo, Sung-Yum; Choi, Chang-Shik; Hong, Seong-Karp; Lee, Ki Hwan

Activity of Diosgenyl 2-amino-2-deoxy-β-D-glucopyranoside, its Hydrochloride, and N,N-dialkyl Derivatives Against Non-albicans Candida Isolates
pp. 460-467(8)
Authors: Dawgul, Malgorzata A.; Grzywacz, Daria; Liberek, Beata; Kamysz, Wojciech; Myszka, Henryk

Synthesis and Structure-Activity Relationship; Exploration of some Potent Anti-Cancer Phenyl Amidrazone Derivatives
pp. 468-477(10)
Authors: Habashneh, Almeqdad Y.; El-Abadelah, Mustafa M.; Bardaweel, Sanaa K.; Taha, Mutasem O.

Scaffold Hopping Strategy for the Design, Synthesis and Biological Activity Evaluation of Novel Hexacyclic Scutellarein Derivatives with a 1,3-Oxazine Ring Fused at A-ring
pp. 478-484(7)
Authors: Zhong, Yue; Lu, Yu-Ting; Sun, Ying; Li, Nian-Guang; Gu, Ting; Wu, Wen-Yu; Yu, Shao-Peng; Shi, Zhi-Hao

Design and Synthesis of 3,4-diarylpyrrole Analogues as Potent Topoisomerase Inhibitors
pp. 485-494(10)
Authors: Chen, Wang; Feng, Zili; He, Xu; Zhao, Qiang; Liang, Qi

Prodrugs for Nitroreductase Based Cancer Therapy- 1: Metabolite Profile, Cell Cytotoxicity and Molecular Modeling Interactions of Nitro Benzamides with Ssap-NtrB
pp. 495-507(13)
Authors: Gungor, Tugba; Yetis, Gulden; Onder, Ferah C.; Tokay, Esra; Tok, Tugba T.; Celik, Ayhan; Ay, Mehmet; Kockar, Feray

Inhibition of Adipogenesis by Thiourea Derivatives
pp. 508-515(8)
Authors: Hina Siddiqui; Sarah Shafi; Farah Mukhtar; Asma Ejaz; Atta-ur-Rahman; M. Iqbal Choudhary

Anthranilic Acid Derivatives: Novel Inhibitors of Protein Glycation and the Associated Oxidative Stress in the Hepatocytes
pp. 516-523(8)
Authors: Humera Jahan; Muhammad I. Choudhary; Amber Atta; Khalid M. Khan; Atta-ur-Rahman

Xanthine Oxidase Inhibitory and Molecular Docking Studies on Pyrimidones
pp. 524-535(12)
Authors: Humaira Zafar; Sarosh Iqbal; Sumaira Javaid; Khalid M. Khan, M.; Muhammad I. Choudhary, I.

New Bis-Pyrazolones as Potential Leads for ROS Inhibition; Environment Friendly Green Synthesis, Structural Characterization, and In Vitro Studies
pp. 536-548(13)
Authors: Sahar Yousuf; Khalid M.Khan; Uzma Salar; Almas Jabeen; Shakil Ahmed; Munira T. Muhammad; Aisha Faheem; Shahnaz Perveen