Medicinal Chemistry

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pp. i-iv(4)

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pp. 601-601(1)
Author: Pal Singh, Inder

Synthesis, Cytotoxic Activity on Leukemia Cell Lines and Quantitative Structure-Activity Relationships (QSAR) Studies of Morita-Baylis-Hillman Adducts
pp. 602-612(11)
Authors: G. Lima128;“Junior, Claudio; V. Faheina128;“Martins, Gláucia; C. B. Bomfim, Caio; B. Dantas, Bruna; P. Silva, Everton; A. M. de Araújo, Demetrius; B. A. Filho, Edilson; L. A. A. Vasconcellos, Mário

Integrated In Silico-In Vitro Discovery of Lung Cancer-related Tumor Pyruvate Kinase M2 (PKM2) Inhibitors
pp. 613-620(8)
Authors: Ye, Xiangyun; Sun, Yinjia; Xu, Yunhua; Chen, Zhiwei; Lu, Shun

Design, Synthesis, and Cytotoxicity of Novel 2,4,6-Trisubstituted 1,3,5- triazines Bearing Aryl Hydrazone Moiety as Potent Antitumor Agent
pp. 621-630(10)
Authors: Wang, Limei; Zhao, Sijia; Bao, Guanglong; Zhang, Yu; Xi, Shuancheng; Zhou, Guolin; Zhai, Xin; Gong, Ping

Synthesis and Biological Evaluation of Novel 1,3,4-thiadiazole Derivatives Incorporating Benzisoselenazolone Scaffold as Potential Antitumor Agents
pp. 631-639(9)
Authors: Fu, Xiaoyun; Li, Sha; Jing, Fen; Wang, Xuefeng; Li, Baolin; Zhao, Jijun; Liu, Yuming; Chen, Baoquan

Synthesis and Antifungal Activity of Some 4,6-Dimethylisoxazolo[3,4- b]pyridin-3(1H)-one Derivatives
pp. 640-646(7)
Authors: Saczewski, Jaroslaw; Fedorowicz, Joanna; Kedzia, Anna; Ziolkowska-Klinkosz, Marta; Jalinska, Aleksandra

Synthesis of Cyclic Imides (Methylphtalimides, Carboxylic Acid Phtalimides and Itaconimides) and Evaluation of their Antifungal Potential
pp. 647-654(8)
Authors: Stiz, Dorimar; Corrêa, Rogério; D. D`Auria, Felicia; Simonetti, Giovanna; Cechinel-Filho, Valdir

Antiplasmodial Limonoids from Trichilia rubescens (Meliaceae)
pp. 655-661(7)
Authors: T. Armelle, Tsamo; K. Pamela, Nangmo; Pierre, Mkounga; B. Müller, Ingrid; Marat, Kirk; Sass, Gabriele; A. Ephrem, Nkengfack

Three Arachidonoylamide Derivatives Inhibit Pro-Inflammatory Genes Expression by Modulating NF-ΚB and AP1 Activities
pp. 662-673(12)
Authors: Gregorelli, Alex; Sgarbossa, Anna; Khan, Shahbaz; Soriente, Annunziata; De Rosa, Margherita; Saturnino, Carmela; Menegazzi, Marta

Synthesis, in vivo Anticoagulant Evaluation and Molecular Docking Studies of Bicoumarins Obtained from Furocoumarin Peucedanin
pp. 674-683(10)
Authors: V. Lipeeva, Alla; V. Khvostov, Mikhail; S. Baev, Dmitry; M. Shakirov, Makhmut; G. Tolstikova, Tatijana; E. Shults, Elvira

Biologically Active New N, N', N''-Tri-Substituted Ferrocenyl Phenylguanidines and their Characterization
pp. 684-698(15)
Authors: Gul, Rukhsana; A. Altaf, Ataf; Badshah, Amin; Shah, Afzal; ur Rehman, Zia; Naz, Rabia; N. Tahir, Muhammad; Junaid, Asif