Medicinal Chemistry

Novel Gastrin Receptor-Directed Contrast Agents - Potential in Brain Tumor Magnetic Resonance Imaging
pp. 133-137(5)
Authors: Sturzu, Alexander; Sheikh, Sumbla; Klose, Uwe; Deeg, Martin; Echner, Hartmut; Nagele, Thomas; Ernemann, Ulrike; Heckl, Stefan

Anticancer Agents for Treatment of Tumors in the Central Nervous System by Correspondent Substituent Substitution and Elucidation by Pattern Recognition Methods
pp. 138-144(7)
Author: Bartzatt, Ronald

Facile Synthesis and Biological Evaluation of Novel Symmetrical Biphenyls as Antitumor Agents
pp. 145-150(6)
Authors: Zhang, Jie; Zhang, Yanmin; Pan, Xiaoyan; Wang, Chen; Hu, Zhigang; Wang, Sicen; He, Langchong

Synthesis and Anticancer Activity of Novel Benzimidazole and Benzothiazole Derivatives against HepG2 Liver Cancer Cells
pp. 151-162(12)
Authors: M. Youssef, Amal; Malki, Ahmed; H. Badr, Mona; Y. Elbayaa, Rasha; S. Sultan, Ahmed

Synthesis and Cytotoxic Evaluation of Quinazolin-4(3H)-one Derivatives Bearing Thiocarbamate, Thiourea or N-Methyldithiocarbamate Side Chains
pp. 163-173(11)
Authors: Cao, Sheng-Li; Xu, Hong; Wang, Yao; Liao, Ji; Zhang, Jing-Jing; Li, Zhong-Feng; Guo, Yan-Wen; Li, Xiao-Rong; Cui, Xue-Mei; Xu, Xingzhi

Optimization of Important Early ADME(T) Parameters of NADPH Oxidase-4 Inhibitor Molecules
pp. 174-181(8)
Authors: Borbely, Gabor; Huszar, Monika; Varga, Attila; Futosi, Krisztina; Mocsai, Attila; Orfi, Laszlo; Idei, Miklos; Mandl, Jozsef; Keri, Gyorgy; Vantus, Tibor

Design, Synthesis & Biological Evaluation of Some Novel Quinazolinone Scaffolds
pp. 182-192(11)
Authors: P. Modh, Rahul; C. Patel, Amit; H. Chikhalia, Kishor

Synthesis and Anti-HIV Activities of Suramin Conjugates of 3'-Fluoro- 2',3'-dideoxythymidine and 3'-Azido-2',3'-dideoxythymidine
pp. 193-197(5)
Authors: K. Agarwal, Hitesh; F. Doncel, Gustavo; Parang, Keykavous

A Pharmacophore Model Specific to Active Site of CYP1A2 with a Novel Molecular Modeling Explorer and CoMFA
pp. 198-207(10)
Authors: Zhang, Tao; Wei, Dong-Qing; Chou, Kuo-Chen

Molecular Dynamics Simulations of CYP2E1
pp. 208-221(14)
Authors: Li, Jue; Wei, Dong-Qing; Wang, Jing-Fang; Yu, Zheng-Tian; Chou, Kuo-Chen

Synthesis of a Fluorescently Labeled Compound for the Detection of Arsenic-induced Apoptotic HL60 Cells
pp. 222-229(8)
Authors: Lis Femia, A.; Facundo Temprana, C.; Silvia Amor, M.; Grasselli, Mariano; del V. Alonso, Silvia

An In Silico Stereo-electronic Comparison of Conventional Pyridinium Oximes and K-oximes for Organophosphate (OP) Poisoning
pp. 230-245(16)
Authors: K. Bhattacharjee, Apurba; Kuca, Kamil; Musilek, Kamil; K. Gordon, Richard

Synthesis and Study the Analgesic Effects of New Analogues of Ketamine on Female Wistar Rats
pp. 246-251(6)
Authors: Ahmadi, Abbas; Khalili, Mohsen; Hajikhani, Ramin; Hosseini, Horiesadat; Afshin, Nasrin; Nahri-Niknafs, Babak

2D Chemometrics Analyses of Tetrahydroquinoline and Ethylenediamine Derivatives with Antimalarial Activity
pp. 252-265(14)
Authors: Fonseca de Freitas, Humberto; Santos Castilho, Marcelo

Synthesis and In Vivo Antimalarial Evaluation of Novel Hydroxyethylamine Derivatives
pp. 266-272(7)
Authors: Conceicao de Souza, Mariana; Goncalves-Silva, Triciana; Moreth, Marcele; R.B. Gomes, Claudia; Roland Kaiser, Carlos; das Gracas Muller de Oliveira Henriques, Maria; V.N. de Souza, Marcus

Small Molecule Hydrazide Agents to Inhibit Growth and Proliferation of Mycobacterium Tuberculosis
pp. 273-280(8)
Authors: Bartzatt, Ronald; L.G. Cirillo, Suat; D. Cirillo, Jeffrey

Structure-Activity Relationships of 2-Benzylsulfanylbenzothiazoles: Synthesis and Selective Antimycobacterial Properties
pp. 281-292(12)
Authors: Klimesova, Vera; Koci, Jan; Palat, Karel; Stolarikova, Jirina; Dahse, Hans-Martin; Mollmann, Ute

Synthesis and Preliminary Antihyperlipidaemic Activities Evaluation of Andrographolide Derivatives
pp. 293-298(6)
Authors: Wang, Bin; Tang, Chunlei; Han, Yaodan; Guo, Ruzhou; Qian, Hai; Huang, Wenlong

Identification of Structural Features for 4-Methyl-3-(6-[Phenyl Methylene] Amino} Pyridine-3-yl)-2h Chromen-2-One Derivatives as Clotting Factor XA Inhibitors
pp. 299-307(9)
Authors: B. Ingale, Kundan; S. Bhatia, Manish