Medicinal Chemistry

Synthesis and Pharmacological Evaluation of 4-Phenoxy-1,2,3,4- Tetrahydroisoquinolines and 4,5,6,6a-Tetrahydrochromeno [2,3,4-de]isoquinolines
pp. 1-10(10)
Authors: Giorgioni, G.; Ruggieri, S.; Claudi, F.; Stefano, A. D.; Ljung, E.; Carlsson, T.

Insight into the Bioreductive Mode of Action of Antitrypanosomal 5- Nitrofuryl Containing Thiosemicarbazones
pp. 11-17(7)
Authors: Gambino, D.; Otero, L.; Maya, J. D.; Morello, A.; Rigol, C.; Barriga, G.; Rodriguez, J.; Folch, C.; Norambuena, E.; Gonzalez, M.; Azar, C. O.; Cerecetto, H.

Synthesis, Molecular Docking and PTP1B Inhibitory Activity of Functionalized 4,5-Dihydronaphthofurans and Dibenzofurans
pp. 18-24(7)
Authors: Goel, Atul; Dixit, Manish; Saeed, Uzma; Kumar, Amit; Siddiqi, Mohammad I.; Tamrakar, Akhilesh K.; Srivastava, Arvind K.

Synthesis and Theoretical Calculations of 5-Aminosalicylic Acid Derivatives as Potential Analgesic Agents
pp. 25-29(5)
Authors: Jose, Trujillo-Ferrara; Jose, Correa-Basurto; Rosales-Hernandez, M. C.; Eduardo, Ramirez-San J.; Abigail, Badillo; Carlos, Z. Gomez-Castro; Fabila-Castillo, L. H.

Estimation of Human Carbonic Anhydrase II Inhibition Using Topological Indices and their Combination with Quantum-Theoretical Descriptors
pp. 30-66(37)
Authors: Khadikar, Padmakar V.; Singh, Jyoti; Singh, Shalini; Mishra, Rajika; Supuran, Claudiu T.; Clare, Brian W.; Lakhwani, Meenakshi

Studies on the Structure-Activity Relationship of the Basic Amine of Phenylpiperazines as Melanocortin-4 Receptor Antagonists
pp. 67-74(8)
Authors: Chen, Chen; Tran, Joe A.; Arellano, Melissa; Fleck, Beth A.; Pontillo, Joseph; Marinkovic, Dragan; Tucci, Fabio C.; Wen, Jenny; Saunders, John

HIV Protease Inhibitors Impact on Apoptosis
pp. 75-79(5)
Authors: Rizza, Stacey A.; Badley, Andrew D.

Simulation of Sequential Screening Experiments Using Emerging Chemical Patterns
pp. 80-90(11)
Authors: Bajorath, Jurgen; Auer, Jens