Letters in Drug Design & Discovery

Graphical Abstract:
pp. i-v(5)

Meet the Editorial Board Member:
pp. 343-343(1)
Author: Lucian Pascu, Mihail

Discovery of Novel HDAC Inhibitors by Structure-based Optimization of Cinnamic Hydroxamic Scaffold
pp. 344-350(7)
Authors: Ning, Chengqing; Huang, Wenyuan; Wu, Wen; Lu, Cheng; He, Yujun; Yao, Lei; Liu, Lifei; Zhen, Xiaohe; Liu, Xiaoyu; Yu, Niefang

Development of Structure Activity Correlation Model on Azetidin-2-ones as Tubulin Polymerization Inhibitors
pp. 351-365(15)
Authors: Kumar Patel, Vijay; Singh Chouhan, Kavibhushan; Singh, Avineesh; Kumar Jain, Deepak; Veerasamy, Ravichandran; Kumar. Singour, Pradeep; Singh Pawar, Rajesh; Rajak, Harish

Synthesis and Anticancer Activity of 7,8-dihydroxy-4-arylcoumarins
pp. 366-373(8)
Authors: Wu, Jianrui; Peng, Ting; Chen, Fang; Leng, Yixin; Tong, Linjiang; Li, Mengyuan; Qu, Rong; Xie, Hua; Ding, Jian; Duan, Wenhu

Hybrid Pharmacophore Design and Synthesis of Naphthalimide– Benzimidazole Conjugates as Potential Anticancer Agents
pp. 374-384(11)
Authors: Kamal, Ahmed; Praveen Kumar, Pogula; Naseer Ahmed Khan, Mohammed; Naga Sheshadri, Bobburi; Srinivas, Olepu

Promising Anticancer Drug Candidates Based on the 7-methoxychromone Scaffold: Synthesis and Evaluation of Antiproliferative Activity
pp. 385-392(8)
Authors: Le Tuan Anh, Hoang; Thi Cuc, Nguyen; Hai Yen, Pham; Xuan Nhiem, Nguyen; Huu Tai, Bui; Thi Thao, Do; Hoai Nam, Nguyen; Van Minh, Chau; Van Kiem, Phan; Ho Kim, Young

Design, Synthesis and Biological Evaluation of Novel Fluorinated Heterocyclic Hybrid Molecules Based on Triazole & Quinoxaline Scaffolds Lead to Highly Potent Antimalarials and Antibacterials
pp. 393-407(15)
Authors: Chandra Shekhar, Adimulam; Pedda Venkat Lingaiah, Boddupally; Shanthan Rao, Pamulaparthy; Narsaiah, Banda; Devi Allanki, Aparna; Singh Sijwali, Puran

Synthesis of Derivatives of Artesunate α-Aminophosphonate and Their Antimicrobial Activities
pp. 408-416(9)
Authors: He, Sheng; Ouyang, Xilin; Huang, Xiaochao; Hu, Weisong; Dai, Weilong; Tian, Xiaoyan; Pan, Yingming; Huang, Shiwen; Wang, Hengshan

Synthesis and Preliminary Biological Evaluation of New Heterocyclic Carboxamide Models
pp. 417-429(13)
Authors: Sweidan, Kamal; Engelmann, Jorn; Abu Rayyan, Walid; Sabbah, Dima; Abu Zarga, Musa; Al-Qirim, Tariq; Al-Hiari, Yusuf; Abu Sheikha, Ghassan; Shattat, Ghassan

Synthesis and Analysis of Anticonvulsant Activities of New 4-[2-(4- alkoxybenzylamino)ethyl]-2H-1,2,4-triazol-3(4H)-one Derivatives
pp. 430-438(9)
Authors: Shen, Qing-Kun; Wang, Shi-Ben; Gong, Guo-Hua; Yin, Xiu-Mei; Quan, Zhe-Shan

Nematicidal Activity of Sprio and Bridged Heterocyclic Neonicotinoid Analogues against Meloidogyne incognita
pp. 439-445(7)
Authors: Zou, Minming; Tian, Xue; Chen, Nanyang; Shao, Xusheng