Letters in Drug Design & Discovery

Letters in Drug Design & Discovery publishes original letters on all areas of rational drug design and discovery including medicinal chemistry, in-silico drug design, combinatorial chemistry, high-throughput screening, drug targets, and structure-activity relationships. The emphasis will be on publishing quality papers very rapidly. Letters will be processed rapidly by taking full advantage of Internet technology for both the submission and review of manuscripts. The journal is essential reading to all pharmaceutical scientists involved in research in drug design and discovery.

Publisher: Bentham Science Publishers

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Analysis of Proteasome Inhibition Prediction Using Atom-Based Quadratic Indices Enhanced by Machine Learning Classification Techniques
pp. 705-711(7)
Authors: M. Casanola-Martin, Gerardo; Le-Thi-Thu, Huong; Marrero-Ponce, Yovani; A Castillo-Garit, Juan; Torrens, Francisco; Perez-Gimenez, Facundo; Abad, Concepcion

Design, Synthesis and Biological Evaluation of Some Oxadiazole Derivatives as Novel Amide-Based Inhibitors of Soluble Epoxide Hydrolase
pp. 721-730(10)
Authors: Rezaee Zavareh, Elham; Hedayati, Mahdi; Hoghooghi Rad, Laleh; Kiani, Azin; Shahhosseini, Soraya; Faizi, Mehrdad; Abbas Tabatabai, Sayyed

A Potential Anticancer Agent 1,2-di(quinazolin-4-yl)diselane
pp. 731-735(5)
Authors: Huang, Yinjiu; Liu, Gang; Hu, Xiaomei; Liu, Hao; Hu, Jianguo; Feng, Zhenzhong; Tang, Bi; Qian, Jun; Wang, Qiyi; Long, Xuehui

Synthesis and Anti-Cancer Activities of Aryl Benzyl Ethers with Fluoro Substituents
pp. 736-741(6)
Authors: Jiang, Yi; Xu, Hong; Liu, Li; He, Rui; Song, Xiaomei; Li, Na

Anticancer Activity and DNA Binding of 4-Alkylenediamines Modified Naphthalimide Derivatives
pp. 742-748(7)
Authors: Wang, Ke-Rang; Qian, Feng; Yang, Zi-Bo; An, Hong-Wei; Han, Dan; Chen, Hua; Zhang, Ping-Zhu; Li, Xiao-Liu

Design, Synthesis and Biological Evaluation of 5-Amino-1H-pyrazole-4- carboxamide Derivatives as Potential Antitumor Agents
pp. 749-755(7)
Authors: Yang, Baowei; Liu, Wukun; Mei, Yicheng; Huang, Dandan; Qian, Hai; Huang, Wenlong; Gust, Ronald

Synthesis of Novel Macrocyclic Tetraamides
pp. 756-761(6)
Authors: Kumar Mehta, Barun; Rambabu, Dandela; Raja, Guttikonda; Prasad, ASG.; Fang, Jim-Min; Venkata Basaveswara Rao, Mandava

Design, Synthesis and Biological Evaluation of 2, 4, 5-Triphenylimidazole Derivatives with Preliminary SAR
pp. 762-769(8)
Authors: Hu, Chunqi; Shen, Jianfeng; Bian, Kejun; Zhang, Ruoyu; Deng, Liping

Pharmacokinetic Analysis of Tetramethylpyrazine Bis-Nitrone TN-2 in Rats and its Protein Binding In Vitro
pp. 770-777(8)
Authors: Sun, Yewei; Liao, Kaiyi; Li, Sai; Zhang, Zaijun; Yu, Pei; Wang, Yuqiang

Novel 4-Oxothienopyrimidinyl Propanoic Acid Derivatives as AMPActivated Protein Kinase (AMPK) Activators
pp. 778-785(8)
Authors: K. Sasmal, Pradip; Jaleel, Mahaboobi; Tirumala Rao, P.; Munikumar, M.; Bhattacharya, Megha; Ravi Kumar, Nutakki; Neelima, Poondla.; Abdul Rawoof, Khaji; Narasimha Rao, P.; Abbineni, Chandrasekhar; Roshaiah, M.; Sridhar, S.; Ranjith Kumar, Thammera; C. A. Vinu, Menon; Potluri, Vijay; Misra, Parimal; Talwar, Rashmi; Kumar Das, Saibal

Influence of the Preparation Method on the Dissolution Properties of Piroxicam - Cyclodextrins Systems
pp. 786-808(23)
Authors: Bouchal, F.; Skiba, M.; Fatmi, S.; Chaffai, N.; Lahiani-Skiba, M.

Synthesis and Biological Activity of Thiazole Dithiocarbamate Derivatives
pp. 814-823(10)
Author: Gundogdu-Karaburun, Nalan

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