Letters in Drug Design & Discovery

Graphical Abstracts
pp. i-viii(8)

Synthesis of Oxygenated Chalcones with Anti-Staphylococcal Activity
pp. 525-530(6)
Authors: Dalla-Vechia, Luciana; Janine Kiekow, Cintia; Correa Ramos Leal, Ivana; Regina Netto Dos Santos, Katia; Cristina Baggio Gnoatto, Simone; Verli, Hugo; Octavio Mendonca Alves de Souza, Rodrigo; Gosmann, Grace

Designing New 5-Nitroimidazoles: Towards Safer Anti-infectious Agents
pp. 531-559(29)
Authors: D. Crozet, Maxime; Terme, Thierry; Vanelle, Patrice

Novel Urea/Thiourea Derivatives of Quinazolin-4(3H)-one: Design, Synthesis, Antimicrobial and Anti-TB Study
pp. 560-571(12)
Authors: R. Shah, Dhruvin; P. Modh, Rahul; V. Desai, Dhara; H. Chikhalia, Kishor

Novel 4-bromo-2-(3-methyl-1-(substituted-phenylsulfonyl)-4,5-dihydro-1- H-pyrazol-5-yl)phenol Derivatives: Synthesis and Antibacterial Activity
pp. 572-577(6)
Authors: Chenga, Qing; Jia, Ying-Ming; Cheng, Fei-Hu; Liu, Xin-Hua

Synthesis and Anticancer Activity of Some 2-[3/4-(2-Substituted Phenyl-2- oxoethoxy)benzylidene]-6-substituted-2,3-dihydro-1H-inden-1-one Derivatives
pp. 578-585(8)
Authors: Gundogdu-Karaburun, Nalan; Cagri Karaburun, Ahmet; Demirayak, Seref; Kayagil, Ismail; Yurttas, Leyla

Synthesis and Antitumor Activities of α-,γ-mangostin Derivatives
pp. 586-593(8)
Authors: Cheng, Kai; Zhang, Gui-lin; Qiu, Sheng-xiang; Liu, Yan-qing; Wang, Yan-fei; Liu, Song; Shan, Yan; Yu, Bo; Lu, Yu

A Facile Synthesis and Anticancer Activity Evaluation of Spiro Analogues of Benzothiazolylchromeno/pyrano Derivatives
pp. 594-600(7)
Authors: Kumar Arya, Anand; Rana, Kulbhushan; Kumar, Mahendra

Design, Synthesis and In-Vitro Evaluation of Polymer-linked Prodrug of Methotrexate for the Targeted Delivery to the Colon
pp. 601-610(10)
Authors: Singla, Nishu; Sharma, Rajiv; Bhardwaj, T.R.

Potent Neuroprotective Activity of Monoterpene Derived 4-[(3aR,7aS)- 1,3,3a,4,5,7a-Hexahydro-3,3,6-trimethylisobenzofuran-1-yl]-2-methoxyphenol in MPTP Mice Model
pp. 611-617(7)
Authors: V. Pavlova, Alla; V. Il'ina, Irina; A. Morozova, Ekaterina; V. Korchagina, Dina; Yu. Kurbakova, Svetlana; V. Sorokina, Irina; G. Tolstikova, Tatyana; P. Volcho, Konstantin; F. Salakhutdinov, Nariman

QSAR Study on Diketo Acid and Carboxamide Derivatives as Potent HIV- 1 Integrase Inhibitor
pp. 618-627(10)
Authors: Olayide Adebimpe, Arodola; Charan Dash, Radha; E. S. Soliman, Mahmoud

Synthesis and Anticonvulsant Activity Evaluation of 4-butyl-5-(4- alkoxyphenyl)-2H-1,2,4-triazole-3(4H)-ones
pp. 628-635(8)
Authors: Zhu, Zi-Shi; Wang, Shi-Ben; Deng, Xian-Qing; Liu, Da-Chuan; Quan, Zhe-Shan

Artificial Neural Networks Modeling of Release of Olanzapine From Glycerol Monooleate Matrices
pp. 636-648(13)
Authors: Bagheri, G.; Vasheghani-Farahani, E.; Ardjmand, M.; Attar, H.; A. Dorkoosh, F.

4D-QSAR Model for Compounds with Binding Affinity Towards Dopamine D2 Receptors
pp. 649-664(16)
Authors: Rodrigues Silva, Daniela; C. Ramalho, Teodorico; F. F. da Cunha, Elaine

A Combined DFT and QSAR Calculations to Study Substituted Biphenyl imidazoles as Bombesin Receptor Subtype-3 Agonists
pp. 665-676(12)
Authors: Shahlaei, Mohsen; Nowroozi, Amin; Khodarahmi, Reza

Synthesis and In Vivo Hepatoprotective Activity of Some Novel Andrographolide Derivatives
pp. 677-685(9)
Authors: Tang, Chunlei; Gu, Guolong; Yang, Baowei; Wang, Xuekun; Qian, Hai; Huang, Wenlong; Zhu, Xiaoyun; Li, Jing

Development of Pyrazole Compounds as Antidiabetic Agent: A Review
pp. 686-703(18)
Authors: A. Datar, Prasanna; R. Jadhav, Sonali