Letters in Drug Design & Discovery

Graphical Abstracts
pp. i-v(5)
Author: Bentham Science Publishers

Editorial
pp. 1-1(1)
Author: Atta-ur-Rahman

Design and Synthesis of 3-Arylisoxazoline-5-Carboxamide and 3-Arylisoxazoline-5-Acetamide Libraries as Potential Factor Xa Inhibitors
pp. 2-7(6)
Authors: F. Quinn, John; T. Gregg, Brian; B. Kitchen, Douglas; M. Lewis, Robert; A. Razzano, Dana; E. Kayser, Lauren; J. Schilling, Levon; C. Golden, Kathryn

Antioxidant Activity of Resveratrol Analogs
pp. 8-11(4)
Authors: Oliveira Calil, Natalia; Senra Goncalves de Carvalho, Gustavo; Cristina Zimmermann Franco, Danielle; David da Silva, Adilson; Rezende Barbosa Raposo, Nadia

Semi-Automatic Synthesis of Distamycin Analogues and their DNA Binding Properties
pp. 12-16(5)
Authors: Drozdowska, Danuta; Szerszenowicz, Jakub

Ligand and Structure-Based Pharmacophore Modeling for the Discovery of Potential Human HNMT Inhibitors
pp. 17-29(13)
Authors: Elumalai, Pavadai; Liu, Hsuan-Liang; Zhou, Zheng-Li; Zhao, Jian-Hua; Chen, Wilson; Chuang, Chih-Kuang; Tsai, Wei-Bor; Ho, Yih

Synthesis and Anti-Paracoccidioides Activity of Calix[n]arenes
pp. 30-36(7)
Authors: Coimbra de Oliveira, Marcilene; Souza Reis, Fabiano; de Fatima, Angelo; Furtado Ferreira Magalhaes, Thais; Leticia da Silva, Danielle; Rodrigues Porto, Raphael; Almeida Watanabe, Giselle; Viviane Buzanello Martins, Cleide; Leite da Silva, Daniel; Lucia Tasca Gois Ruiz, Ana; Antonio Fernandes, Sergio; Ernesto de Carvalho, Joao; Aparecida de Resende-Stoianoff, Maria

Preliminary Evaluation of Anticonvulsant Activity of Some Aminoalkanol and Amino Acid Cinnamic Acid Derivatives
pp. 37-43(7)
Authors: Gunia, Agnieszka; M. Waszkielewicz, Anna; Cegla, Marek; Marona, Henryk

Discovery of 5,6-Dihydro-indolo[1,2-a]quinoxaline Derivatives as New HIV-1 Inhibitors In Vitro
pp. 44-47(4)
Authors: Fan, Ling-Ling; Huang, Ning; Yang, Rui-Ge; He, Shu-Zhen; Yang, Liu-Meng; Xu, Hui; Zheng, Yong-Tang

Evaluation of the Radioprotective Potential of the Polyphenol Norbadione A
pp. 48-53(6)
Authors: Le Roux, Antoine; Josset, Elodie; Benzina, Sami; Nadal, Brice; Desage-El Murr, Marine; Heurtaux, Benoit; Taran, Frederic; Denis, Jean-Marc; Le Gall, Thierry; Meunier, Stephane; Bischoff, Pierre

Lobeline Docking on AChBP and Nicotinic Receptors: Discriminating Importance of the Pocket Geometry and of the Ligand Configuration
pp. 54-62(9)
Authors: Colas, Claire; Brotel, Xavier; Duclert-Savatier, Nathalie; Nilges, Michael; Joseph, Delphine; E. Malliavin, Therese

Synthesis and Biological Evaluation of Some Novel Thiazolylhydrazinomethylideneferrocenes as Antimicrobial Agents
pp. 63-68(6)
Authors: Chandak, Navneet; Kumar, Pawan; Sharma, Chetan; R. Aneja, Kamal; K. Sharma, Pawan

Synthesis, Biochemical Evaluation and Rationalisation of a Series of (3-O-Sulfonate) Derivatives of Estrone (E1) as Probes of the Active Site of Type 3 of the 17β-Hydroxysteroid Dehydrogenase (17β-HSD) Family of Enzymes
pp. 69-76(8)
Authors: Akbarzadeh, Mohsen; S. Olusanjo, Moniola; Ahmed, Sabbir

Pramipexole Tachyphylaxis and its Management in Bipolar Depression
pp. 77-77(1)
Author: Sharma, Verinder

Design, Synthesis and Biological Evaluation of Scutellarein Derivatives as Potential Anti-Alzheimer's Disease Candidates Based on Metabolic Mechanism
pp. 78-83(6)
Authors: Song, Shu-Lin; Li, Nian-Guang; Tang, Yu-Ping; Wang, Zhen-Jiang; Qian, Li-Hua; Tang, Hao; Duan, Jin-Ao

Small Molecule Tyrosine Kinase Inhibitors: The New Dawn for Cancer Therapy
pp. 84-125(42)
Authors: N. Noolvi, Malleshappa; M. Patel, Harun