Letters in Drug Design & Discovery

Structure-Based Drug Design of Peptide Mimetics Containing Large P3 Moieties as Inhibitors of Factor VIIa
pp. 86-92(7)
Authors: Shiraishi, Takuya; Kadono, Shojiro; Haramura, Masayuki; Kodama, Hirofumi; Ono, Yoshiyuki; Iikura, Hitoshi; Esaki, Tohru; Koga, Takaki; Hattori, Kunihiro; Watanabe, Yoshiaki; Sakamoto, Akihisa; Yoshihashi, Kazutaka; Kitazawa, Takehisa; Esaki, Keiko; Ohta, Masateru; Sato, Haruhiko; Kozono, Toshiro

Prediction of Binding Affinities for Hydroxamic Acid Derivatives as Urease Inhibitors by Molecular Docking and 3D-QSAR Studies
pp. 93-100(8)
Authors: Zaheer-ul-Haq; Wadood, Abdul

Novel N-Substituted Thiazolidinones as Proton Pump Inhibitors and Potent Anti-Ulcer Agents: SAR Study
pp. 101-106(6)
Authors: Chandrappa, S.; Vinaya, K.; Srikanta, B. M.; Kumar, C.S. A.; Thimmegowda, N. R.; Ranganatha, S. R.; Dharmesh, Shylaja M.; Rangappa, K. S.

Synthesis of Substituted 1H-Pyrrol-2(5H)-ones and 2(5H)-Furanones as Inhibitors of P. aeruginosa Biofilm
pp. 107-113(7)
Authors: Guo, Jia-Liang; Li, Bing-Zhou; Chen, Wei-Min; Sun, Ping-Hua; Wang, Yuqiang

Investigation of the Structural Requirement for Blocking the Human CCR5 Chemokine Receptor. An Insight from Quantitative Structure Activity Relationships Study
pp. 114-124(11)
Author: Dessalew, Nigus

Physical Stability of PLGA Microparticles for DNA Encapsulation
pp. 125-128(4)
Authors: Migueliz, Itziar; Diez, Sonsoles; Navarro, Gemma; de ILarduya, Conchita T.

A Novel Synthesis Method of Apogossypolone and its Antitumor Activity
pp. 129-132(4)
Authors: Zhan, Yonghua; Jia, Guangfeng

Synthesis and Antiproliferative Activity of Coumarin-Estrogen Conjugates against Breast Cancer Cell Lines
pp. 133-138(6)
Authors: Musa, Musiliyu A.; F. Khan, M. O.; Cooperwood, John S.

Presentation of the β -Carboxamidophosphonate Arrangement in Substrate Structures Targeting HIV-1 PR
pp. 139-145(7)
Authors: Wardle, N. J.; Hudson, H. R.; Matthews, R. W.; Nunn, C.; Vella, C.; Bligh, S.W. A.

Synthesis and In Vitro Antimicrobial Activity of Medicinally Important Novel N-alkyl, N-aryl and Urea Derivatives of 1-benzhydryl Piperizine: A Structure-Activity Relationship Study
pp. 146-154(9)
Authors: Ananda Kumar, Channapillekoppal S.; Murthy, Karunakara; Sadashiva, Marlinganadoddi Panchegowda; Vinaya, Mallappanahally Kambappa; Thimmegowda, Naraganahalli Ramegowda; Benaka Prasad, Salekoppal Boregowda; Chandrappa, Siddappa; Rangappa, Kanchugarakoppal Subbegowda

Complex of Nifedipine with Glycyrrhizic Acid as a Novel Water-Soluble Antihypertensive and Antiarrhythmic Agent
pp. 155-158(4)
Authors: Tolstikova, T. G.; Khvostov, M. V.; Bryzgalov, A. O.; Dushkin, A. V.; Meteleva, E. S.

α 2-Adrenoceptor Antagonist SL84.0418 Involvement in the Development of Opioid Withdrawal
pp. 159-162(4)
Authors: Capasso, Anna; Gallo, Chiara

3-Aminosterol Compounds as a New Class of Anti-Malarial Agents against Chloroquine-Susceptible and -Resistant Plasmodium falciparum
pp. 163-166(4)
Authors: Salmi, Chanaz; Loncle, Celine; Vidal, Nicolas; Rogier, Christophe; Letourneux, Yves; Pradines, Bruno; Brunel, Jean M.