Current Topics in Medicinal Chemistry

Graphical Abstracts
pp. i-iv(4)

Targeting the DCN1-UBC12 Protein-Protein Interaction for Selective Modulation of Cullin Substrates
pp. 1423-1425(3)
Authors: Fang, Yuan; Yu, Lei; Liao, Guochao; Yu, Bin

Synthesis and Biological Profiles of 1,2,3-Triazole Scaffold
pp. 1426-1427(2)
Authors: de Carvalho da Silva, Fernando; Ferreira, Vitor F.; da Silva Magalhães Forezi, Luana

Alternative Routes to the Click Method for the Synthesis of 1,2,3-Triazoles, an Important Heterocycle in Medicinal Chemistry
pp. 1428-1453(26)
Authors: da S.M. Forezi, Luana; Cardoso, Mariana F.C.; Gonzaga, Daniel T.G.; de C. da Silva, Fernando; Ferreira, Vitor F.

Design, Synthesis and Antileishmanial Activity of Naphthotriazolyl-4-Oxoquinolines
pp. 1454-1464(11)
Authors: Oliveira, Vanessa G.; dos Santos Faiões, Viviane; Gonçalves, Gabrieli B.R.; Lima, Miriam F.O.; Boechat, Fernanda C.S.; Cunha, Anna C.; de Andrade-Neto, Valter V.; de C. da Silva, Fernando; Torres-Santos, Eduardo C.; de Souza, Maria Cecília B.V.

A Novel Naphthotriazolyl-4-oxoquinoline Derivative that Selectively Controls Breast Cancer Cells Survival Through the Induction of Apoptosis
pp. 1465-1474(10)
Authors: Branco, Jessica R.; Oliveira, Vanessa G.; Esteves, Amanda M.; Chipoline, Ingrid C.; Lima, Miriam F.O.; Boechat, Fernanda C.S.; da Silva, Fernando C.; Ferreira, V F.; Sola-Penna, Mauro; de Souza, Maria C.B.V.; Zancan, Patricia

Novel Symmetrical 1,4-Disubstituted-bis-1,2,3-Triazoles: Synthesis by Double CuAAC and Cytotoxicity Evaluation
pp. 1475-1482(8)
Authors: Reis, Wallace J.; Moreira, Paulo O.L.; Alves, Rosemeire B.; Oliveira, Helo H.M.; Silva, Luciana M.; Varotti, Fernando P.; Freitas, Rossimiriam P.

A Novel Triazole Derivative Drug Presenting In Vitro and In Vivo Anticancer Properties
pp. 1483-1493(11)
Authors: Filho, Ricardo I.; Gonzaga, Daniel T.G.; Demaria, Thainá M.; Leandro, João G.B.; Costa, Dora C.S.; Ferreira, Vitor F.; Sola-Penna, Mauro; de C. da Silva, Fernando; Zancan, Patricia

New Efavirenz Derivatives and 1,2,3-Triazolyl-phosphonates as Inhibitors of Reverse Transcriptase of HIV-1
pp. 1494-1505(12)
Authors: Costa, Carolina C.P.; Boechat, Nubia; Bastos, Monica M.; da Silva, Fernando de C.; Marttorelli, Andressa; Souza, Thiago M.L.; Baptista, Mayara S.; Hoelz, Lucas V.B.; Cafffarena, Ernesto R.

Oxazolone–1,2,3-Triazole Hybrids: Design, Synthesis and Antimicrobial Evaluation
pp. 1506-1513(8)
Authors: Lal, Kashmiri; Kumar, Lokesh; Kumar, Ashwani; Kumar, Anil