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Current Pharmaceutical Design publishes timely in-depth reviews covering all aspects of current research in rational drug design. Each issue is devoted to a single major therapeutic area. A Guest Editor who is an acknowledged authority in a therapeutic field has solicits for each issue comprehensive and timely reviews from leading researchers in the pharmaceutical industry and academia.

Each thematic issue of Current Pharmaceutical Design covers all subject areas of major importance to modern drug design, including: medicinal chemistry, pharmacology, drug targets and disease mechanism.

Publisher: Bentham Science Publishers

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Volume 22, Number 38, 2016

Articles

In Vitro and Ex Vivo Model Systems to Measure ABC Transporter Activity at the Blood-Brain Barrier
pp. 5768-5773(6)
Authors: M. de Wit, Nienke; Kooij, Gijs; E. de Vries, Helga

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Design and Synthesis of New Selective P-gp Substrates and Inhibitors
pp. 5774-5778(5)
Authors: Cantore, Mariangela; Leopoldo, Marcello; Berardi, Francesco; Perrone, Roberto; Colabufo, Nicola Antonio

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PET Tracers for Imaging of ABC Transporters at the Blood-Brain Barrier: Principles and Strategies
pp. 5779-5785(7)
Authors: Luurtsema, Gert; Elsinga, Philip; Dierckx, Rudi; Boellaard, Ronald; Waarde, Aren van

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ABC Transporters and Drug Resistance in Patients with Epilepsy
pp. 5793-5807(15)
Authors: Feldmann, Maria; Koepp, Matthias

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Blood-Brain Barrier ABC-transporter P-glycoprotein in Alzheimer's Disease: Still a Suspect?
pp. 5808-5816(9)
Authors: M.E. van Assema, Danielle; N.M. van Berckel, Bart

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Importance of ABC Transporters in Drug Development
pp. 5817-5829(13)
Authors: Benadiba, Marcel; Maor, Yehoshua

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Importance of P-gp PET Imaging in Pharmacology
pp. 5830-5836(7)
Author: Toyohara, Jun

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Neuronutrient Amino-Acid Therapy Protects Against Reward Deficiency Syndrome: Dopaminergic Key to Homeostasis and Neuroplasticity
pp. 5837-5854(18)
Authors: Blum, Kenneth; Febo, Marcelo; D. Badgaiyan, Rajendra; R. Braverman, Eric; Dushaj, Kristina; Li, Mona; Demetrovics, Zsolt

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Shear Stress-sensitive Carriers for Localized Drug Delivery
pp. 5855-5867(13)
Authors: Xia, Yu; Shi, Chun-Yang; Xiong, Wei; Hou, Xiao-Long; Fang, Jian-Guo; Wang, Wen-Qing

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Site-Specific Thiol-mediated PEGylation of Streptokinase Leads to Improved Properties with Clinical Potential
pp. 5868-5878(11)
Authors: Sawhney, Pooja; Kumar, Shekhar; Maheshwari, Neeraj; Singh Guleria, Sumeet; Dhar, Neelam; Kashyap, Radhika; Sahni, Girish

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