Skip to main content
Current Pharmaceutical Design publishes timely in-depth reviews covering all aspects of current research in rational drug design. Each issue is devoted to a single major therapeutic area. A Guest Editor who is an acknowledged authority in a therapeutic field has solicits for each issue comprehensive and timely reviews from leading researchers in the pharmaceutical industry and academia.

Each thematic issue of Current Pharmaceutical Design covers all subject areas of major importance to modern drug design, including: medicinal chemistry, pharmacology, drug targets and disease mechanism.

Publisher: Bentham Science Publishers

More about this publication?
Volume 18, Number 20, 2012

Articles

Conformationally Constrained Peptides as Protein Tyrosine Kinase Inhibitors
pp. 2852-2866(15)
Authors: K. Tiwari, Rakesh; Parang, Keykavous

Favourites:
ADD
Favourites:
ADD

Recent Advances in Designing Substrate-Competitive Protein Kinase Inhibitors
pp. 2875-2882(8)
Authors: Han, Ki-Cheol; Yeon Kim, So; Gyeong Yang, Eun

Favourites:
ADD

Free Content Perspective of Cyclin-dependent kinase 9 (CDK9) as a Drug Target
pp. 2883-2890(8)
Authors: Krystof, Vladimir; Baumli, Sonja; Furst, Robert

Favourites:
ADD

Kinase Inhibitor Conjugates
pp. 2891-2900(10)
Authors: Harmsen, Stefan; Jan Kok, Robbert

Favourites:
ADD

Insulin-like Growth Factor-1 Receptor (IGF-1R) Kinase Inhibitors in Cancer Therapy: Advances and Perspectives
pp. 2901-2913(13)
Authors: Xue, Mengzhu; Cao, Xianwen; Zhong, Ye; Kuang, Dong; Liu, Xiaofeng; Zhao, Zhenjiang; Li, Honglin

Favourites:
ADD

Exploiting Substrate Recognition for Selective Inhibition of Protein Kinases
pp. 2914-2920(7)
Authors: Licht-Murava, Avital; Eldar-Finkelman, Hagit

Favourites:
ADD

Selective VEGFR Inhibitors for Anticancer Therapeutics in Clinical Use and Clinical Trials
pp. 2921-2935(15)
Authors: Zhang, Cunlong; Tan, Chunyan; Ding, Huaiwei; Xin, Tian; Jiang, Yuyang

Favourites:
ADD
Favourites:
ADD

Molecular Dynamics of Protein Kinase-Inhibitor Complexes: A Valid Structural Information
pp. 2946-2963(18)
Authors: Caballero, Julio; H. Alzate-Morales, Jans

Favourites:
ADD
Favourites:
ADD

Cyclin-dependent kinase Inhibitors Inspired by Roscovitine: Purine Bioisosteres
pp. 2974-2980(7)
Authors: Jorda, Radek; Paruch, Kamil; Krystof, Vladimir

Favourites:
ADD

Recent Advances in Thymidine Kinase 2 (TK2) Inhibitors and New Perspectives for Potential Applications
pp. 2981-2994(14)
Authors: Priego, Eva-Maria; Karlsson, Anna; Gago, Federico; Camarasa, Maria-Jose; Balzarini, Jan; Perez-Perez, Maria-Jesus

Favourites:
ADD

  • Access Key
  • Free content
  • Partial Free content
  • New content
  • Open access content
  • Partial Open access content
  • Subscribed content
  • Partial Subscribed content
  • Free trial content