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Current Pharmaceutical Design publishes timely in-depth reviews covering all aspects of current research in rational drug design. Each issue is devoted to a single major therapeutic area. A Guest Editor who is an acknowledged authority in a therapeutic field has solicits for each issue comprehensive and timely reviews from leading researchers in the pharmaceutical industry and academia.

Each thematic issue of Current Pharmaceutical Design covers all subject areas of major importance to modern drug design, including: medicinal chemistry, pharmacology, drug targets and disease mechanism.

Publisher: Bentham Science Publishers

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Volume 16, Number 29, 2010

Articles

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Recent Advances in Structural Studies of the Carbonic Anhydrase Family: The Crystal Structure of Human CA IX and CA XIII
pp. 3246-3254(9)
Authors: T. Supuran, Claudiu; Di Fiore, Anna; Alterio, Vincenzo; Maria Montib, Simona; De Simone, Giuseppina

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Carbonic Anhydrase IX as an Anticancer Therapy Target: Preclinical Evaluation of Internalizing Monoclonal Antibody Directed to Catalytic Domain
pp. 3255-3263(9)
Authors: Zatovicova, M.; Jelenska, L.; Hulikova, A.; Csaderova, L.; Ditte, Z.; Ditte, P.; Goliasova, T.; Pastorek, J.; Pastorekova, S.

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Carbonic Anhydrase Related Protein VIII and its Role in Neurodegeneration and Cancer
pp. 3264-3276(13)
Authors: Aspatwar, Ashok; E.E. Tolvanen, Martti; Ortutay, Csaba; Parkkila, Seppo

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Carbonic Anhydrase Inhibitors Developed Through ‘Click Tailing’
pp. 3277-3287(11)
Authors: Lopez, Marie; J. Salmon, Adam; T. Supuran, Claudiu; Poulsen, Sally-Ann

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Modulation of Carbonic Anhydrase 9 (CA9) in Human Brain Cancer
pp. 3288-3299(12)
Authors: M. Said, Harun; T. Supuran, Claudiu; Hageman, Carsten; Staab, Adrian; Polat, Buelent; Katzer, Astrid; Scozzafava, Andrea; Anacker, Jelena; Flentje, Michael; Vordermark, Dirk

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The β-Carbonic Anhydrases from Mycobacterium tuberculosis as Drug Targets
pp. 3300-3309(10)
Authors: Nishimoria, Isao; Minakuchia, Tomoko; Marescab, Alfonso; Cartab, Fabrizio; Scozzafava, Andrea; T. Supuran, Claudiu

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Brucella Carbonic Anhydrases: New Targets for Designing Anti-Infective Agents
pp. 3310-3316(7)
Authors: Winum, Jean-Yves; Kohler, Stephan; T. Supuran, Claudiu

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3-Phenyl-1H-Indole-5-Sulfonamides: Structure-Based Drug Design of a Promising Class of Carbonic Anhydrase Inhibitors
pp. 3317-3326(10)
Authors: Guzela, Ozlen; Innocenti, Alessio; Vullo, Daniela; Scozzafava, Andrea; T. Supuran, Claudiu

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Saccharomyces cerevisiae β-Carbonic Anhydrase: Inhibition and Activation Studies
pp. 3327-3336(10)
Authors: Isika, Semra; Ozensoy Guler, Ozen; Kockar, Feray; Aydin, Meltem; Arslan, Oktay; T. Supuran, Claudiu

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