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Current Medicinal Chemistry covers all the latest and outstanding developments in medicinal chemistry and rational drug design. Each issue contains a series of timely in-depth reviews written by leaders in the field covering a range of the current topics in medicinal chemistry. Current Medicinal Chemistry is an essential journal for every medicinal chemist who wishes to be kept informed and up-to-date with the latest and most important developments.

Publisher: Bentham Science Publishers

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Volume 25, Number 42, 2018

Editorial

Free Content Current Medicinal Chemistry: Striving for Excellence
pp. 5799-5799(1)
Author: Atta-ur-Rahman

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Review article

Structural Insights into Azole-based Inhibitors of Heme Oxygenase-1: Development of Selective Compounds for Therapeutic Applications
pp. 5803-5821(19)
Authors: Rahman, Mona N.; Vukomanovic, Dragic; Vlahakis, Jason Z.; Szarek, Walter A.; Nakatsu, Kanji; Jia, Zongchao

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A Focus on the Synthesis and Pharmacokinetics of Tocainide and its Analogues
pp. 5822-5834(13)
Authors: Carocci, Alessia; Corbo, Filomena; Lentini, Giovanni; Cavalluzzi, Maria M.; Franchini, Carlo; Catalano, Alessia

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Liver and Statins: A Critical Appraisal of the Evidence
pp. 5835-5846(12)
Authors: Licata, Anna; Giammanco, Antonina; Minissale, Maria G.; Pagano, Salvatore; Petta, Salvatore; Averna, Maurizio

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Development of Bruton's Tyrosine Kinase Inhibitors for Rheumatoid Arthritis
pp. 5847-5859(13)
Authors: Lv, Jiahui; Wu, Jingde; He, Feng; Qu, Ying; Zhang, Qiuqiong; Yu, Chenggong

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Biologics for the Treatment of Juvenile Idiopathic Arthritis
pp. 5860-5893(34)
Authors: Poddighe, Dimitri; Romano, Micol; Gattinara, Maurizio; Gerloni, Valeria

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Essentials and Perspectives of Computational Modelling Assistance for CNS-oriented Nanoparticle-based Drug Delivery Systems
pp. 5894-5913(20)
Authors: Kisała, Joanna; Hęclik, Kinga I.; Pogocki, Krzysztof; Pogocki, Dariusz

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Gold-Based Nanoparticles Systems in Phototherapy - Current Strategies
pp. 5914-5929(16)
Authors: Błaszkiewicz, Paulina; Kotkowiak, Michał

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Current Understanding of Interactions between Nanoparticles and ABC Transporters in Cancer Cells
pp. 5930-5944(15)
Authors: Yin, Jian; Deng, Xudong; Zhang, Jie; Lin, Jun

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Ischemic Stroke and Kynurenines: Medicinal Chemistry Aspects
pp. 5945-5957(13)
Authors: Hertelendy, Péter; Toldi, József; Fülöp, Ferenc; Vécsei, László

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Herbal Compounds with Special Reference to Gastrodin as Potential Therapeutic Agents for Microglia Mediated Neuroinflammation
pp. 5958-5974(17)
Authors: Li, Juan-Juan; Liu, Shun-Jin; Liu, Xiao-Yu; Ling, Eng-Ang

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Virtual Screening for the Development of New Effective Compounds Against Staphylococcus aureus
pp. 5975-5985(11)
Authors: Diniz, Roseane C.; Soares, Lucas Weba; Nascimento da Silva, Luís Cláudio

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Tuber Lectins with Potentially Exploitable Bioactivities
pp. 5986-6001(16)
Authors: Cheung, Randy C. F.; Wong, Jack H.; Ng, Tzi Bun; Naude, Ryno; Rolka, Krzysztof; Tse, Ryan; Tse, Tak Fu; Chan, Helen; Sze, Stephen Cho Wing

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Selected Applications for Current Polymers in Prosthetic Dentistry - State of the Art
pp. 6002-6012(11)
Authors: Kawala, Maciej; Smardz, Joanna; Adamczyk, Lukasz; Grychowska, Natalia; Wieckiewicz, Mieszko

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Bacterial Transferase MraY, a Source of Inspiration towards New Antibiotics
pp. 6013-6029(17)
Authors: Fer, Mickaël J.; Corre, Laurent L.; Pietrancosta, Nicolas; Evrard-Todeschi, Nathalie; Olatunji, Samir; Bouhss, Ahmed; Calvet-Vitale, Sandrine; Gravier-Pelletier, Christine

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Medicinal Chemistry Updates on Bacterial Efflux Pump Modulators
pp. 6030-6069(40)
Authors: Durães, Fernando; Pinto, Madalena; Sousa, Emília

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The Importance of Complying with Vaccination Protocols in Developed Countries: “Anti-Vax” Hysteria and the Spread of Severe Preventable Diseases
pp. 6070-6081(12)
Authors: Pandolfi, F.; Franza, L.; Todi, L.; Carusi, V.; Centrone, M.; Buonomo, A.; Chini, R.; Newton, E.E.; Schiavino, D.; Nucera, E.

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Articles

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