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Current Drug Metabolism aims to cover all the latest and outstanding developments in drug metabolism and disposition. The journal serves as an international forum for the publication of timely reviews in drug metabolism. Current Drug Metabolism is an essential journal for academic, clinical, government and pharmaceutical scientists who wish to be kept informed and up-to-date with the latest and most important developments. The journal covers the following areas:

In vitro systems including CYP-450; enzyme induction and inhibition; drug-drug interactions and enzyme kinetics; pharmacokinetics, toxicokinetics, species scaling and extrapolations; P-glycoprotein and transport carriers; target organ toxicity and interindividual variability; drug metabolism and disposition studies; extrahepatic metabolism; phase I and phase II metabolism; recent developments for the identification of drug metabolites and adducts.

Publisher: Bentham Science Publishers

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Volume 21, Number 13, 2020

Abstract

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pp. i-iv(4)

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pp. 995-995(1)
Author: Xing, Jie

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Review article

Metabolism and Distribution of Novel Tumor Targeting Drugs In Vivo
pp. 996-1008(13)
Authors: Wang, Mengli; Du, Qiuzheng; Zuo, Lihua; Xue, Peng; Lan, Chao; Sun, Zhi

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Concomitant Drug Treatment and Elimination in the RCC-affected Kidneys: Can We Kill Two Birds with One Stone?
pp. 1009-1021(13)
Authors: Ahmed, Muhammad B.; Salman Ul Islam; Lee, Young Sup

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Research article

Differential Impacts of Azole Antifungal Drugs on the Pharmacokinetic Profiles of Dasatinib in Rats by LC-MS-MS
pp. 1022-1030(9)
Authors: Luo, Xingxian; Xue, Xuecai; Li, Taifeng; Zhang, Ying; Huang, Lin; Cheng, Gang

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A Randomized Study on the Bioequivalence of Desloratadine in Healthy Chinese Subjects and the Association of Different Metabolic Phenotypes With UGT2B10 and CYP2C8 Genotypes
pp. 1031-1039(9)
Authors: Niu, Suping; Li, Yan; Dong, Wenliang; Xia, Lin; Shen, Tiantian; Wang, Jiaxue; Wang, Qian; Zhang, Tan; Zhang, Minjie; Liu, Gang; Guo, Danjie; Fang, Yi

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CYP2C and CYP2B Mediated Metabolic Activation of Retrorsine in Cyp3a Knockout Mice
pp. 1040-1051(12)
Authors: Pang, Xiaoyan; Tang, Chongzhuang; Kong, Fandi; Chen, Meixia; Chen, Xiaoyan

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The Genetic Polymorphism of CYP3A4 rs2242480 is Associated with Sirolimus Trough Concentrations among Adult Renal Transplant Recipients
pp. 1052-1059(8)
Authors: Lolita, Lolita; Zheng, Ming; Zhang, Xiang; Han, Zhijian; Tao, Jun; Fei, Shuang; Wang, Zijie; Guo, Miao; Yang, Haiwei; Ju, Xiaobing; Tan, Ruoyun; Wei, Ji-Fu; Gu, Min

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Breast Cancer Resistance Protein and Multidrug Resistance Protein 2 Mediate the Disposition of Leonurine-10-O-β-glucuronide
pp. 1060-1067(8)
Authors: Li, Xiaocui; Xie, Yushan; Qu, Wei; Ou, Xiaojun; Ou, Xiaowen; Wang, Chuang; Qi, Xiaoxiao; Wang, Ying; Liu, Zhongqiu; Zhu, Lijun

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