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Current Drug Metabolism aims to cover all the latest and outstanding developments in drug metabolism and disposition. The journal serves as an international forum for the publication of timely reviews in drug metabolism. Current Drug Metabolism is an essential journal for academic, clinical, government and pharmaceutical scientists who wish to be kept informed and up-to-date with the latest and most important developments. The journal covers the following areas:

In vitro systems including CYP-450; enzyme induction and inhibition; drug-drug interactions and enzyme kinetics; pharmacokinetics, toxicokinetics, species scaling and extrapolations; P-glycoprotein and transport carriers; target organ toxicity and interindividual variability; drug metabolism and disposition studies; extrahepatic metabolism; phase I and phase II metabolism; recent developments for the identification of drug metabolites and adducts.

Publisher: Bentham Science Publishers

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Volume 5, Number 5, 2004

Review article

Cigarette Smoking, Metabolic Activation and Carcinogenesis
pp. 363-373(11)
Authors: Nishikawa, Akiyoshi; Mori, Yukio; Lee, In-Seon; Tanaka, Takuji; Hirose, Masao

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Biopharmaceutic Classification System: A Scientific Framework for Pharmacokinetic Optimization in Drug Research
pp. 375-388(14)
Authors: Varma, Manthena V.S.; Khandavilli, Sateesh; Ashokraj, Yasvanth; Jain, Amit; Dhanikula, Anandbabu; Sood, Anurag; Thomas, Narisetty S.; Pillai, Omathanu; Sharma, Pradeep; Gandhi, Rajesh; Agrawal, Shrutidevi; Nair, Vinod; Panchagnula, Ramesh

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Therapeutic Drugs that Behave as Mechanism-Based Inhibitors of Cytochrome P450 3A4
pp. 415-442(28)
Authors: Zhou, Shufeng; Chan, Eli; Lim, Lee Y.; Boelsterli, Urs A.; Li, Shu Chuen; Wang, Jiancheng; Zhang, Qiang; Huang, Min; Xu, Anlong

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Human Hepatocytes in Primary Culture: The Choice to Investigate Drug Metabolism in Man
pp. 443-462(20)
Authors: Gomez-Lechon, M. J.; Donato, M. T.; Castell, J. V.; Jover, R.

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