Search Results

Phase I study of TLR9 agonist PF-3512676 in combination with carboplatin and paclitaxel in patients with advanced non-small-cell lung cancer

Authors: Yamada, Kazuhiko; Nakao, Masao; Fukuyama, Chikara; Nokihara, Hiroshi; Yamamoto, Noboru; Sekine, Ikuo; Kunitoh, Hideo; Ohe, Yuichiro; Ohki, Emiko; Hashimoto, Junichi; Tamura, Tomohide

Source: Cancer Science, Volume 101, Number 1, January 2010 , pp. 188-195(8)

Publisher: Blackwell Publishing

Cognitive enhancement as a pharmacotherapy target for stimulant addiction

Author: Sofuoglu, Mehmet

Source: Addiction, Volume 105, Number 1, January 2010 , pp. 38-48(11)

Publisher: Blackwell Publishing

Dual effect of the novel peptide antagonist K-14585 on proteinase-activated receptor-2-mediated signalling

Authors: Goh, Fui Goon; Ng, Pei Yuen; Nilsson, Mary; Kanke, Toru; Plevin, Robin

Source: British Journal of Pharmacology, Volume 158, Number 7, December 2009 , pp. 1695-1704(10)

Publisher: Blackwell Publishing

Agonist and blocking actions of choline and tetramethylammonium on human muscle acetylcholine receptors

Authors: Lape, Remigijus; Krashia, Paraskevi; Colquhoun, David; Sivilotti, Lucia G.

Source: The Journal of Physiology, Volume 587, Number 21, November 2009 , pp. 5045-5072(28)

Publisher: Blackwell Publishing

Novel selective ligands for free fatty acid receptors GPR120 and GPR40

Authors: Hara, Takafumi; Hirasawa, Akira; Sun, Qi; Sadakane, Keiko; Itsubo, Chisato; Iga, Tomoyo; Adachi, Tetsuya; Koshimizu, Taka-aki; Hashimoto, Toshihiro; Asakawa, Yoshinori; Tsujimoto, Gozoh

Source: Naunyn-Schmiedeberg's Archives of Pharmacology, Volume 380, Number 3, September 2009 , pp. 247-255(9)

Publisher: Springer

Effects of inactivation-resistant agonists on the signalling, desensitization and down-regulation of bradykinin B₂ receptors

Authors: Bawolak, Marie-Thérèse; Fortin, Sébastien; Bouthillier, Johanne; Adam, Albert; Gera, Lajos; C.-Gaudreault, René; Marceau, François

Source: British Journal of Pharmacology, Volume 158, Number 5, November 2009 , pp. 1375-1386(12)

Publisher: Blackwell Publishing

Role of channel activation in cognitive enhancement mediated by α7 nicotinic acetylcholine receptors

Authors: Briggs, Clark A; Grønlien, Jens Halvard; Curzon, Peter; Timmermann, Daniel B; Ween, Hilde; Thorin-Hagene, Kirsten; Kerr, Paige; Anderson, David J; Malysz, John; Dyhring, Tino; Olsen, Gunnar M; Peters, Dan; Bunnelle, William H; Gopalakrishnan, Murali

Source: British Journal of Pharmacology, Volume 158, Number 6, November 2009 , pp. 1486-1494(9)

Publisher: Blackwell Publishing

Cloning and pharmacological characterization of the dog P2X7 receptor

Authors: Roman, S; Cusdin, FS; Fonfria, E; Goodwin, JA; Reeves, J; Lappin, SC; Chambers, L; Walter, DS; Clay, WC; Michel, AD

Source: British Journal of Pharmacology, Volume 158, Number 6, November 2009 , pp. 1513-1526(14)

Publisher: Blackwell Publishing

Cytoprotective effects of adenosine and inosine in an in vitro model of acute tubular necrosis

Authors: Módis, Katalin; Gerő, Domokos; Nagy, Nóra; Szoleczky, Petra; Tóth, Zoltán Dóri; Szabó, Csaba

Source: British Journal of Pharmacology, Volume 158, Number 6, November 2009 , pp. 1565-1578(14)

Publisher: Blackwell Publishing

Memantine binding to a superficial site on NMDA receptors contributes to partial trapping

Authors: Kotermanski, Shawn E.; Wood, Jesse T.; Johnson, Jon W.

Source: The Journal of Physiology, Volume 587, Number 19, October 2009 , pp. 4589-4604(16)

Publisher: Blackwell Publishing

Increased colonic transit in rats produced by a combination of a cholinesterase inhibitor with a 5-HT₄ receptor agonist

Authors: campbell-dittmeyer, k.; hicks, g. a.; earnest, d. l.; greenwood-van meerveld, b.

Source: Neurogastroenterology and Motility, Volume 21, Number 11, November 2009 , pp. 1197-e108(-1196)

Publisher: Blackwell Publishing

Cost Effectiveness of Varenicline in Belgium, Compared with Bupropion, Nicotine Replacement Therapy, Brief Counselling and Unaided Smoking Cessation: A BENESCO Markov Cost-Effectiveness Analysis

Authors: Annemans, Lieven; Nackaerts, Kristiaan; Bartsch, Pierre; Prignot, Jacques; Marbaix, Sophie

Source: Clinical Drug Investigation, Volume 29, Number 10, 1 October 2009 , pp. 655-665(11)

Publisher: Adis International

Varenicline increases striatal dopamine D_2/3 receptor binding in rats

Authors: Crunelle, Cleo L.; Miller, Michelle L.; de Bruin, Kora; van den Brink, Wim; Booij, Jan

Source: Addiction Biology, Volume 14, Number 4, October 2009 , pp. 500-502(3)

Publisher: Blackwell Publishing

Spotlight on Buprenorphine/Naloxone in the Treatment of Opioid Dependence†

Authors: Orman, Jennifer S.; Keating, Gillian M.

Source: CNS Drugs, Volume 23, Number 10, 1 October 2009 , pp. 899-902(4)

Publisher: Adis International

Cyclic Opioid Peptide Agonists and Antagonists Obtained Via Ring-Closing Metathesis

Authors: Berezowska, Irena; Lemieux, Carole; Chung, Nga N.; Wilkes, Brian C.; Schiller, Peter W.

Source: Chemical Biology & Drug Design, Volume 74, Number 4, October 2009 , pp. 329-334(6)

Publisher: Blackwell Publishing

The Use of Iontophoresis in the Administration of Nicotine and New Non-Nicotine Drugs through the Skin for Smoking Cessation

Authors: Escobar-Chavez, Jose J.; Merino, Virginia; Lopez-Cervantes, Miriam; Rodriguez-Cruz, Isabel M.a.r.l.e.n.; Quintanar-Guerrero, David; Ganem-Quintanar, Adriana

Source: Current Drug Discovery Technologies, Volume 6, Number 3, September 2009 , pp. 171-185(15)

Publisher: Bentham Science Publishers

Involvement of PKCα and G-protein-coupled receptor kinase 2 in agonist-selective desensitization of µ-opioid receptors in mature brain neurons

Authors: Bailey, CP; Oldfield, S; Llorente, J; Caunt, CJ; Teschemacher, AG; Roberts, L; McArdle, CA; Smith, FL; Dewey, WL; Kelly, E; Henderson, G

Source: British Journal of Pharmacology, Volume 158, Number 1, September 2009 , pp. 157-164(8)

Publisher: Blackwell Publishing

Agonist efficacy and receptor desensitization: from partial truths to a fuller picture

Author: Charlton, Steven J

Source: British Journal of Pharmacology, Volume 158, Number 1, September 2009 , pp. 165-168(4)

Publisher: Blackwell Publishing

The long-acting β-adrenoceptor agonist, indacaterol, inhibits IgE-dependent responses of human lung mast cells

Authors: Scola, Anne-Marie; Loxham, Matthew; Charlton, Steven J; Peachell, Peter T

Source: British Journal of Pharmacology, Volume 158, Number 1, September 2009 , pp. 267-276(10)

Publisher: Blackwell Publishing

Constitutive activity of cannabinoid-2 (CB₂) receptors plays an essential role in the protean agonism of (+)AM1241 and L768242

Authors: Mancini, I; Brusa, R; Quadrato, G; Foglia, C; Scandroglio, P; Silverman, LS; Tulshian, D; Reggiani, A; Beltramo, M

Source: British Journal of Pharmacology, Volume 158, Number 1, September 2009 , pp. 382-391(10)

Publisher: Blackwell Publishing