Search Results

Novel effects mediated by bradykinin and pharmacological characterization of bradykinin B₂ receptor antagonism in human synovial fibroblasts

Authors: Bellucci, F; Cucchi, P; Catalani, C; Giuliani, S; Meini, S; Maggi, CA

Source: British Journal of Pharmacology, Volume 158, Number 8, December 2009 , pp. 1996-2004(9)

Publisher: Blackwell Publishing

FTY720 (fingolimod) in Multiple Sclerosis: therapeutic effects in the immune and the central nervous system

Author: Brinkmann, Volker

Source: British Journal of Pharmacology, Volume 158, Number 5, November 2009 , pp. 1173-1182(10)

Publisher: Blackwell Publishing

Functional antagonism of IL-1α induced gene expression profiles define the cAMP/PKA pathway as a unique regulator of IL-1α signaling networks

Authors: Murray, David L.; Johnson, Eric N.; Wang, Ping; Gauthier, Josee; Bing, Nan; Vanderwall, Dana; Xu, Zangwei; Jensen, David; Cox, Richard F.; Kostura, Matthew; Sorensen, Scott D.

Source: Journal of Receptors and Signal Transduction, Volume 29, Number 5, October 2009 , pp. 246-256(11)

Publisher: Informa Healthcare

Ticagrelor binds to human P2Y₁₂ independently from ADP but antagonizes ADP-induced receptor signaling and platelet aggregation

Authors: VAN GIEZEN, J. J. J.; NILSSON, L.; BERNTSSON, P.; WISSING, B.-M.; GIORDANETTO, F.; TOMLINSON, W.; GREASLEY, P. J.

Source: Journal of Thrombosis and Haemostasis, Volume 7, Number 9, September 2009 , pp. 1556-1565(10)

Publisher: Blackwell Publishing

5-HT_1A receptors are involved in the effects of xaliproden on G-protein activation, neurotransmitter release and nociception

Authors: Martel, J-C; Assié, M-B; Bardin, L; Depoortère, R; Cussac, D; Newman-Tancredi, A

Source: British Journal of Pharmacology, Volume 158, Number 1, September 2009 , pp. 232-242(11)

Publisher: Blackwell Publishing

Role of α₁- and β₃-adrenoceptors in the modulation by SR59230A of the effects of MDMA on body temperature in the mouse

Authors: Bexis, Sotiria; Docherty, James R

Source: British Journal of Pharmacology, Volume 158, Number 1, September 2009 , pp. 259-266(8)

Publisher: Blackwell Publishing

SB265610 is an allosteric, inverse agonist at the human CXCR2 receptor

Authors: Bradley, ME; Bond, ME; Manini, J; Brown, Z; Charlton, SJ

Source: British Journal of Pharmacology, Volume 158, Number 1, September 2009 , pp. 328-338(11)

Publisher: Blackwell Publishing

Salicylate, an aspirin metabolite, specifically inhibits the current mediated by glycine receptors containing α1-subunits

Authors: Lu, Y-G; Tang, Z-Q; Ye, Z-Y; Wang, H-T; Huang, Y-N; Zhou, K-Q; Zhang, M; Xu, T-L; Chen, L

Source: British Journal of Pharmacology, Volume 157, Number 8, August 2009 , pp. 1514-1522(9)

Publisher: Blackwell Publishing

Molecular Mechanisms Underlying Female Sex Determination - Antagonism Between Female and Male Pathway

Author: Piprek, Rafał P.

Source: Folia Biologica, Volume 57, Numbers 3-4, June 2009 , pp. 105-113(9)

Publisher: Institute of Systematics and Evolution of Animals, Polish Academy of Sciences

Drugs in development for the treatment of schizophrenia

Author: Emsley, Robin

Source: Expert Opinion on Investigational Drugs, Volume 18, Number 8, August 2009 , pp. 1103-1118(16)

Publisher: Informa Healthcare

Thyroid Hormone Antagonists: Potential Medical Applications and Structure Activity Relationships

Authors: Malm, Johan; Farnegardh, Mathias; Grover, Gary J.; Ladenson, Paul W.

Source: Current Medicinal Chemistry, Volume 16, Number 25, September 2009 , pp. 3258-3266(9)

Publisher: Bentham Science Publishers

Serotonin stimulates platelet receptor shedding by tumor necrosis factor-alpha-converting enzyme (ADAM17)

Authors: DUERSCHMIED, D.; CANAULT, M.; LIEVENS, D.; BRILL, A.; CIFUNI, S. M.; BADER, M.; WAGNER, D. D.

Source: Journal of Thrombosis and Haemostasis, Volume 7, Number 7, July 2009 , pp. 1163-1171(9)

Publisher: Blackwell Publishing

BGC20-1531, a novel, potent and selective prostanoid EP₄ receptor antagonist: a putative new treatment for migraine headache

Authors: Maubach, KA; Davis, RJ; Clark, DE; Fenton, G; Lockey, PM; Clark, KL; Oxford, AW; Hagan, RM; Routledge, C; Coleman, RA

Source: British Journal of Pharmacology, Volume 156, Number 2, January 2009 , pp. 316-327(12)

Publisher: Blackwell Publishing

Antagonism of serotonergic 5-HT_2A/2C receptors: mutual improvement of sleep, cognition and mood?

Authors: Landolt, H.-P.; Wehrle, R.

Source: European Journal of Neuroscience, Volume 29, Number 9, May 2009 , pp. 1795-1809(15)

Publisher: Blackwell Publishing

Endothelin receptor selectivity: evidence from in vitro and pre-clinical models of scleroderma

Authors: Shiwen, X.; Leask, A.; Abraham, D. J.; Fonseca, C.

Source: European Journal of Clinical Investigation, Volume 39, Supplement 2, June 2009 , pp. 19-26(8)

Publisher: Blackwell Publishing

Dopamine D₂-Receptor-Mediated Increase in Vascular and Endothelial NOS Activity Ameliorates Cerebral Vasospasm After Subarachnoid Hemorrhage In Vitro

Authors: Pyne-Geithman, Gail; Caudell, Danielle; Cooper, Matthew; Clark, Joseph; Shutter, Lori

Source: Neurocritical Care, Volume 10, Number 2, April 2009 , pp. 225-231(7)

Publisher: Humana Press

Modelling the human immune response: performance of a 10¹¹ human antibody repertoire against a broad panel of therapeutically relevant antigens

Authors: Lloyd, C.; Lowe, D.; Edwards, B.; Welsh, F.; Dilks, T.; Hardman, C.; Vaughan, T.

Source: Protein Engineering, Design and Selection, Volume 22, Number 3, March 2009 , pp. 159-168(10)

Publisher: Oxford University Press

Endothelin Receptor Antagonism: Role in the Treatment of Pulmonary Arterial Hypertension Related to Scleroderma

Authors: Kabunga, Peter; Coghlan, Gerry

Source: Drugs, Volume 68, Number 12, 2008 , pp. 1635-1645(11)

Publisher: Adis International

Dorothy Hodgkin Lecture 2008 Gastric inhibitory polypeptide (GIP) revisited: a new therapeutic target for obesity-diabetes?

Author: Flatt, P. R.

Source: Diabetic Medicine, Volume 25, Number 7, July 2008 , pp. 759-764(6)

Publisher: Blackwell Publishing

Targets for ethanol action and antagonism in Loop 2 of the extracellular domain of glycine receptors

Authors: Perkins, Daya I.; Trudell, James R.; Crawford, Daniel K.; Alkana, Ronald L.; Davies, Daryl L.

Source: Journal of Neurochemistry, Volume 106, Number 3, August 2008 , pp. 1337-1349(13)

Publisher: Blackwell Publishing