Search Results

The X-Ray Structure of Carboxypeptidase A Inhibited by a Thiirane Mechanism-Based Inhibitor

Authors: Fernández, Daniel; Testero, Sebastian; Vendrell, Josep; Avilés, Francesc X.; Mobashery, Shahriar

Source: Chemical Biology & Drug Design, Volume 75, Number 1, January 2010 , pp. 29-34(6)

Publisher: Blackwell Publishing

Heme Oxygenase Inhibition by 2-Oxy-substituted 1-Azolyl-4-phenylbutanes: Effect of Variation of the Azole Moiety. X-Ray Crystal Structure of Human Heme Oxygenase-1 in Complex with 4-Phenyl-1-(1H-1,2,4-triazol-1-yl)-2-butanone

Authors: Roman, Gheorghe; Rahman, Mona N.; Vukomanovic, Dragic; Jia, Zongchao; Nakatsu, Kanji; Szarek, Walter A.

Source: Chemical Biology & Drug Design, Volume 75, Number 1, January 2010 , pp. 68-90(23)

Publisher: Blackwell Publishing

Cámaraite, Ba₃NaTi₄(Fe²⁺,Mn)₈(Si₂O₇)₄O₄(OH,F)₇. I. A new Ti-silicate mineral from the Verkhnee Espe Deposit, Akjailyautas Mountains, Kazakhstan

Authors: Sokolova, E.; Abdu, Y.; Hawthorne, F.C.; Stepanov, A.V.; Bekenova, G.K.; Kotel'nikov, P.E.

Source: Mineralogical Magazine, Volume 73, Number 5, October 2009 , pp. 847-854(8)

Publisher: Mineralogical Society

Tautomeric forms study of 1H-(2′-pyridyl)-3-methyl-5-hydroxypyrazole and 1H-(2′-pyridyl)-3-phenyl-5-hydroxypyrazole. Synthesis, structure, and cytotoxic activity of their complexes with palladium(II) ions

Authors: Ciolkowski, Michal; Paneth, Piotr; Lorenz, Ingo-Peter; Mayer, Peter; Rozalski, Marek; Krajewska, Urszula; Budzisz, Elzbieta

Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 24, Number 6, December 2009 , pp. 1257-1268(12)

Publisher: Informa Healthcare

Novel factor Xa inhibitors: a patent review

Authors: de Candia, Modesto; Lopopolo, Gianfranco; Altomare, Cosimo

Source: Expert Opinion on Therapeutic Patents, Volume 19, Number 11, November 2009 , pp. 1535-1580(46)

Publisher: Informa Healthcare

The Status of the Australian Synchrotron

Authors: Hobbs, Robert; Gower, Steve; Lamb, Robert

Source: Synchrotron Radiation News, Volume 22, Number 4, July 2009 , pp. 29-33(5)

Publisher: Taylor and Francis Ltd

Advances in fragment-based drug discovery platforms

Authors: Orita, Masaya; Warizaya, Masaichi; Amano, Yasushi; Ohno, Kazuki; Niimi, Tatsuya

Source: Expert Opinion on Drug Discovery, Volume 4, Number 11, November 2009 , pp. 1125-1144(20)

Publisher: Informa Healthcare

Editorial [Hot topic: Exploring Novel Chemical Space Through the Use of Computational and Structural Biology (Guest Editor: Alan C. Rigby)]

Author: Rigby, Alan C.

Source: Combinatorial Chemistry & High Throughput Screening, Volume 12, Number 10, December 2009 , pp. 927-928(2)

Publisher: Bentham Science Publishers

Structure-Based Virtual Ligand Screening: Recent Success Stories

Authors: Villoutreix, Bruno O.; Eudes, Richard; Miteva, Maria A.

Source: Combinatorial Chemistry & High Throughput Screening, Volume 12, Number 10, December 2009 , pp. 1000-1016(17)

Publisher: Bentham Science Publishers

Editorial [Hot topic: In Silico Approaches in G Protein-Coupled Receptors (GPCRs) Drug Discovery: Quo Vadis? (Executive Editor: Stefano Moro)]

Author: Moro, Stefano

Source: Current Pharmaceutical Design, Volume 15, Number 35, December 2009 , pp. 3992-3993(2)

Publisher: Bentham Science Publishers

Fast Binding Kinetics and Conserved 3D Structure Underlie the Antagonistic Activity of Mutant TNF: Useful Information for Designing Artificial Proteo-Antagonists

Authors: Mukai, Yohei; Nakamura, Teruya; Yoshioka, Yasuo; Shibata, Hiroko; Abe, Yasuhiro; Nomura, Tetsuya; Taniai, Madoka; Ohta, Tsunetaka; Nakagawa, Shinsaku; Tsunoda, Shin-ichi; Kamada, Haruhiko; Yamagata, Yuriko; Tsutsumi, Yasuo

Source: The Journal of Biochemistry, Volume 146, Number 2, 7 August 2009 , pp. 167-172(6)

Publisher: Oxford University Press

Tetrameric Acetylcholinesterase: The Effects of Substrates Acetylcholine and Butyrocholine on Its Submolecular Structure Observed by Atomic Force Microscope

Authors: Jiang, Shuang; Zhang, Yingge; Zhang, Sa

Source: Journal of Scientific Conference Proceedings, Volume 1, Numbers 2-3, June 2009 , pp. 167-172(6)

Publisher: American Scientific Publishers

Quinolones: Action and Resistance Updated

Authors: Drlica, Karl; Hiasa, Hiroshi; Kerns, Robert; Malik, Muhammad; Mustaev, Arkady; Zhao, Xilin

Source: Current Topics in Medicinal Chemistry, Volume 9, Number 11, August 2009 , pp. 981-998(18)

Publisher: Bentham Science Publishers

Ternary oxovanadium(IV) complexes of ONO-donor Schiff base and polypyridyl derivatives as protein tyrosine phosphatase inhibitors: synthesis, characterization, and biological activities

Authors: Yuan, Caixia; Lu, Liping; Gao, Xiaoli; Wu, Yanbo; Guo, Maolin; Li, Ying; Fu, Xueqi; Zhu, Miaoli

Source: JBIC Journal of Biological Inorganic Chemistry, Volume 14, Number 6, August 2009 , pp. 841-851(11)

Publisher: Springer

Yeast as a tool for characterizing mono-ADP-ribosyltransferase toxins

Authors: Turgeon, Zachari; White, Dawn; Jørgensen, René; Visschedyk, Danielle; Fieldhouse, Robert J.; Mangroo, Dev; Merrill, A. Rod

Source: FEMS Microbiology Letters, Volume 300, Number 1, November 2009 , pp. 97-106(10)

Publisher: Blackwell Publishing

The capsid protein of human immunodeficiency virus: designing inhibitors of capsid assembly

Author: Neira, José L.

Source: FEBS Journal, Volume 276, Number 21, November 2009 , pp. 6110-6117(8)

Publisher: Blackwell Publishing

Structural and mutational analysis of TenA protein (HP1287) from the Helicobacter pylori thiamin salvage pathway - evidence of a different substrate specificity

Authors: Barison, Nicola; Cendron, Laura; Trento, Alberto; Angelini, Alessandro; Zanotti, Giuseppe

Source: FEBS Journal, Volume 276, Number 21, November 2009 , pp. 6227-6235(9)

Publisher: Blackwell Publishing

An engineered right-handed coiled coil domain imparts extreme thermostability to the KcsA channel

Authors: Yuchi, Zhiguang; Pau, Victor P. T.; Lu, Bridget X.; Junop, Murray; Yang, Daniel S. C.

Source: FEBS Journal, Volume 276, Number 21, November 2009 , pp. 6236-6246(11)

Publisher: Blackwell Publishing

Low temperature growth of Si nanowires via vapour-liquid-solid mechanism

Authors: Ng, I.K.; Suzuki, H.

Source: Materials Research Innovations, Volume 13, Number 3, September 2009 , pp. 192-195(4)

Publisher: Maney Publishing

Editorial [Hot topic: Structure- and Ligand-Based Drug Design: Advances and Perspectives (Guest Editor: Adriano D. Andricopulo)]

Author: Andricopulo, Adriano D.

Source: Current Topics in Medicinal Chemistry, Volume 9, Number 9, June 2009 , pp. 754-754(1)

Publisher: Bentham Science Publishers