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Design, Synthesis, and Biological Evaluation of 7H-thiazolo[3,2-b]-1,2,4-triazin-7-one Derivatives as Acetylcholinesterase Inhibitors

Authors: Liu, Si-Jie; Yang, Liu; Liu, Xiao-Guang; Luo, Ying; Cao, Zi-Jian; Cheong Wan, David C.; Lin, Huang-Quan; Hu, Chun

Source: Letters in Drug Design & Discovery, Volume 7, Number 1, January 2010 , pp. 5-8(4)

Publisher: Bentham Science Publishers

α-N-Heterocyclic Thiosemicarbazone Derivatives as Potential Antitumor Agents: A Structure-Activity Relationships Approach

Authors: Matesanz, Ana I.; Souza, Pilar

Source: Mini Reviews in Medicinal Chemistry, Volume 9, Number 12, October 2009 , pp. 1389-1396(8)

Publisher: Bentham Science Publishers

Machine Learning Quantitative Structure-Activity Relationships (QSAR) for Peptides Binding to the Human Amphiphysin-1 SH3 Domain

Author: Ivanciuc, Ovidiu

Source: Current Proteomics, Volume 6, Number 4, December 2009 , pp. 289-302(14)

Publisher: Bentham Science Publishers

Overview of Naphthalimide Analogs as Anticancer Agents

Authors: Lv, Min; Xu, Hui

Source: Current Medicinal Chemistry, Volume 16, Number 36, December 2009 , pp. 4797-4813(17)

Publisher: Bentham Science Publishers

Editorial [Hot topic: Natural Products (Guest Editors: Wei-Shuo Fang and Junzeng Zhang)]

Authors: Fang, Wei-Shuo; Zhang, Junzeng

Source: Current Topics in Medicinal Chemistry, Volume 9, Number 16, November 2009 , pp. 1493-1493(1)

Publisher: Bentham Science Publishers

Polyisoprenylated Benzophenones from Clusiaceae: Potential Drugs and Lead Compounds

Authors: Acuna, Ulyana M.; Jancovski, Nikola; Kennelly, Edward J.

Source: Current Topics in Medicinal Chemistry, Volume 9, Number 16, November 2009 , pp. 1560-1580(21)

Publisher: Bentham Science Publishers

Pentacyclic Triterpenoids and Their Saponins with Apoptosis-Inducing Activity

Authors: Wang, Shao-Rong; Fang, Wei-Shuo

Source: Current Topics in Medicinal Chemistry, Volume 9, Number 16, November 2009 , pp. 1581-1596(16)

Publisher: Bentham Science Publishers

Pituitary Adenylate Cyclase-Activating Polypeptide: Focus on Structure- Activity Relationships of a Neuroprotective Peptide

Authors: Bourgault, S.; Vaudry, D.; Dejda, A.; Doan, N. D.; Vaudry, H.; Fournier, A.

Source: Current Medicinal Chemistry, Volume 16, Number 33, November 2009 , pp. 4462-4480(19)

Publisher: Bentham Science Publishers

Extraction of Structure-Activity Relationship Information from High-Throughput Screening Data

Authors: Wawer, M.; Bajorath, J.

Source: Current Medicinal Chemistry, Volume 16, Number 31, November 2009 , pp. 4049-4057(9)

Publisher: Bentham Science Publishers

How to Recognize and Workaround Pitfalls in QSAR Studies:A Critical Review

Authors: Scior, T.; Medina-Franco, J. L.; Do, Q.-T.; Martinez-Mayorga, K.; Yunes Rojas, J. A.; Bernard, P.

Source: Current Medicinal Chemistry, Volume 16, Number 32, November 2009 , pp. 4297-4313(17)

Publisher: Bentham Science Publishers

Calmodulin in Complex with Proteins and Small Molecule Ligands: Operating with the Element of Surprise; Implications for Structure-Based Drug Design

Authors: Menyhard, Dora K.; Keseru, Gyorgy M.; Naray-Szabo, Gabor

Source: Current Computer - Aided Drug Design, Volume 5, Number 4, December 2009 , pp. 264-279(16)

Publisher: Bentham Science Publishers

Prospective Ligand- and Target-Based 3D QSAR: State of the Art 2008

Author: Clark, Robert D.

Source: Current Topics in Medicinal Chemistry, Volume 9, Number 9, June 2009 , pp. 791-810(20)

Publisher: Bentham Science Publishers

Inhibitory activity of isoflavones of Pueraria flowers on nitric oxide production from lipopolysaccharide-activated primary rat microglia

Authors: Yuan, Dan; Xie, Yuan-Yuan; Bai, Xue; Wu, Xia; Yang, Jing-Yu; Wu, Chun-Fu

Source: Journal of Asian Natural Products Research, Volume 11, Number 6, June 2009 , pp. 471-481(11)

Publisher: Taylor and Francis Ltd

Synthesis and SAR Study of Opioid Receptor Ligands: Mono- and Bis-Indolomorphinans

Authors: Li, Fuying; Yin, Chenlei; Chen, Jie; Liu, Jinggen; Xie, Xin; Zhang, Ao

Source: Chemical Biology & Drug Design, Volume 74, Number 4, October 2009 , pp. 335-342(8)

Publisher: Blackwell Publishing

Medicinal Chemistry of Paclitaxel and its Analogues

Authors: Fu, Y.; Li, S.; Zu, Y.; Yang, G.; Yang, Z.; Luo, M.; Jiang, S.; Wink, M.; Efferth, T.

Source: Current Medicinal Chemistry, Volume 16, Number 30, October 2009 , pp. 3966-3985(20)

Publisher: Bentham Science Publishers

QSAR Study of Androstenedione Analogs as Aromatase Inhibitors

Authors: Oliveira, Aline A.; Ramalho, Teodorico C.; da Cunha, Elaine F.F.

Source: Letters in Drug Design & Discovery, Volume 6, Number 8, December 2009 , pp. 554-562(9)

Publisher: Bentham Science Publishers

Recent Studies of QSAR on Inhibitors of Estrogen Receptor and Human Eosinophil Phosphodiesterase

Authors: Xiang, Yuhong; Zhang, Zhuoyong; Xiao, Aijing; Huo, Jinxu

Source: Current Computer - Aided Drug Design, Volume 5, Number 3, September 2009 , pp. 200-214(15)

Publisher: Bentham Science Publishers

Substrates, Inducers, Inhibitors and Structure-Activity Relationships of Human Cytochrome P450 2C9 and Implications in Drug Development

Authors: Zhou, S.-F.; Zhou, Z.-W.; Yang, L.-P.; Cai, J.-P.

Source: Current Medicinal Chemistry, Volume 16, Number 27, September 2009 , pp. 3480-3675(196)

Publisher: Bentham Science Publishers

Translocator Protein Ligands as Promising Therapeutic Tools for Anxiety Disorders

Authors: Taliani, S.; Da Settimo, F.; Da Pozzo, E.; Chelli, B.; Martini, C.

Source: Current Medicinal Chemistry, Volume 16, Number 26, September 2009 , pp. 3359-3380(22)

Publisher: Bentham Science Publishers

Conformational Sampling and Energetics of Drug-Like Molecules

Authors: Foloppe, Nicolas; Chen, I-Jen

Source: Current Medicinal Chemistry, Volume 16, Number 26, September 2009 , pp. 3381-3413(33)

Publisher: Bentham Science Publishers