Search Results

Novel diphenyl esters of peptidyl α-aminoalkylphosphonates as inhibitors of chymotrypsin and subtilisin

Authors: Pietrusewicz, Ewa; Sieńczyk, Marcin; Oleksyszyn, Józef

Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 24, Number 6, December 2009 , pp. 1229-1236(8)

Publisher: Informa Healthcare

Trioxsalen derivatives with lipoxygenase inhibitory activity

Authors: Hadjipavlou-Litina, D.; E. Bariamis, S.; Militsopoulou, M.; Athanassopoulos, C. M.; Papaioannou, D.

Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 24, Number 6, December 2009 , pp. 1351-1356(6)

Publisher: Informa Healthcare

Synthesis and Biological Activity of Wuweizisu C and Analogs

Authors: Chang, J. B.; Wang, Q.; Li, Y. F.

Source: Current Topics in Medicinal Chemistry, Volume 9, Number 17, November 2009 , pp. 1660-1675(16)

Publisher: Bentham Science Publishers

Inhibition of platelet activation by peptide analogs of the β₃-intracellular domain of platelet integrin α_IIbβ₃ conjugated to the cell-penetrating peptide Tat(48-60)

Authors: Dimitriou, Andromaxi A.; Stathopoulos, Panagiotis; Mitsios, John V.; Sakarellos-Daitsiotis, Maria; Goudevenos, John; Tsikaris, Vassilios; Tselepis, Alexandros D.

Source: Platelets, Volume 20, Number 8, June 2009 , pp. 539-547(9)

Publisher: Informa Healthcare

Studies on peptidyl nucleoside antibiotics: synthesis and antifungal evaluation of pyranosyl nucleoside analogs of nikkomycin

Authors: Stauffer, Christina S; Fothergill, Annette W; Rinaldi, Michael G; Dutta, Apurba

Source: Future Medicinal Chemistry, Volume 1, Number 2, May 2009 , pp. 379-389(11)

Publisher: Future Science

Update and commentary on the pro-drug bimatoprost and a putative `prostamide receptor'

Authors: Sharif, Najam A; Klimko, Peter

Source: Expert Review of Ophthalmology, Volume 4, Number 5, October 2009 , pp. 477-489(13)

Publisher: Expert Reviews

Pituitary Adenylate Cyclase-Activating Polypeptide: Focus on Structure- Activity Relationships of a Neuroprotective Peptide

Authors: Bourgault, S.; Vaudry, D.; Dejda, A.; Doan, N. D.; Vaudry, H.; Fournier, A.

Source: Current Medicinal Chemistry, Volume 16, Number 33, November 2009 , pp. 4462-4480(19)

Publisher: Bentham Science Publishers

Kukoamine A analogs with lipoxygenase inhibitory activity

Authors: Hadjipavlou-Litina, Dimitra; Garnelis, Thomas; Athanassopoulos, Constantinos M.; Papaioannou, Dionissios

Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 24, Number 5, October 2009 , pp. 1188-1193(6)

Publisher: Informa Healthcare

Roscovitine Triggers Apoptosis in B-Cell Chronic Lymphocytic Leukemia Cells with Similar Efficiency as Combinations of Conventional Purine Analogs with Cyclophosphamide

Authors: Zolnierczyk, Jolanta D.; Błoński, Jerzy Z.; Robak, Tadeusz; Kiliańska, Zofia M.; Węsierska-Gadek, Józefa

Source: Annals of the New York Academy of Sciences, Volume 1171, Number 1, August 2009 , pp. 124-131(8)

Publisher: Blackwell Publishing

Prevention of hepatocellular carcinoma in hepatitis B virus infection

Authors: Lim, Seng Gee; Mohammed, Rosmawati; Yuen, Man-Fung; Kao, Jia-Horng

Source: Journal of Gastroenterology and Hepatology, Volume 24, Number 8, August 2009 , pp. 1352-1357(6)

Publisher: Blackwell Publishing

Synthesis and Evaluation of Anthelmintic and Cytotoxic Properties of [2,5']Bis-1,3-Azole Analogs of Bengazoles

Authors: Scarone, Laura; Fajardo, Jose; Saldana, Jenny; Dominguez, Laura; Esposito, Pablo; Demastteis, Sylvia; Wipf, Peter; Manta, Eduardo; Serra, Gloria

Source: Letters in Drug Design & Discovery, Volume 6, Number 6, September 2009 , pp. 413-419(7)

Publisher: Bentham Science Publishers

Acronycine Derivatives: A Promising Series of Anti-Cancer Agents

Authors: Nguyen, Q. C.; Nguyen, T. T.; Yougnia, R.; Gaslonde, T.; Dufat, H.; Michel, S.; Tillequin, F.

Source: Anti-Cancer Agents in Medicinal Chemistry (Formerly Current Medicinal Chemistry, Volume 9, Number 7, September 2009 , pp. 804-815(12)

Publisher: Bentham Science Publishers

On the Synthesis and Anticancer Testing of α,β-Unsaturated Ketones as Analogs of Combretastatin-A4

Authors: Chavda, Sameer; Davis, Ryan; Ferguson, Amanda; Riddering, Camille; Dittenhafer, Kristin; Mackay, Hilary; Babu, Balaji; Lee, Moses; Siegfried, Adam; Pennington, William; Shadfan, Miriam; Mooberry, Susan L.; Mishra, Bijay K.; Pati, Hari N.

Source: Letters in Drug Design & Discovery, Volume 6, Number 7, October 2009 , pp. 531-537(7)

Publisher: Bentham Science Publishers

The Current Status and Future Perspectives of Studies of Cannabinoid Receptor 1 Antagonists as Anti-Obesity Agents

Authors: Lee, Hyeon-Kyu; Choi, Eun B.; Pak, Chwang S.i.e.k.

Source: Current Topics in Medicinal Chemistry, Volume 9, Number 6, April 2009 , pp. 482-503(22)

Publisher: Bentham Science Publishers

Kynuramines, metabolites of melatonin and other indoles: the resurrection of an almost forgotten class of biogenic amines

Authors: Hardeland, Rüdiger; Tan, Dun-Xian; Reiter, Russel J.

Source: Journal of Pineal Research, Volume 47, Number 2, September 2009 , pp. 109-126(18)

Publisher: Blackwell Publishing

Molecular targets for antiviral therapy of cytomegalovirus infections

Authors: Marschall, Manfred; Stamminger, Thomas

Source: Future Microbiology, Volume 4, Number 6, August 2009 , pp. 731-742(12)

Publisher: Future Medicine

Fentanyl Analogs: Structure-Activity-Relationship Study

Authors: Vuckovic, S.; Prostran, M.; Ivanovic, M.; Dosen-Micovic, Lj.; Todorovic, Z.; Nesic, Z.; Stojanovic, R.; Divac, N.; Mikovic, Z.

Source: Current Medicinal Chemistry, Volume 16, Number 19, July 2009 , pp. 2468-2474(7)

Publisher: Bentham Science Publishers

Insights through AM1 calculations into the structural requirement of N-hydroxythiosemicarbazone analogs as anti-tubercular agents

Authors: Gupta, Revathi A.; Gupta, Arun Kumar; Soni, Love Kumar; Kaskhedikar, S. G.

Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 24, Number 3, June 2009 , pp. 850-858(9)

Publisher: Informa Healthcare

Design, synthesis and pharmacological evaluation of 6-hydroxy-4-methylquinolin-2(1H)-one derivatives as inotropic agents

Authors: Sadeghian, Hamid; Seyedi, Seyed Mohammad; Saberi, Mohammad Reza; Nick, Reza Shafiee; Hosseini, Azar; Bakavoli, Mehdi; Mansouri, Seyed Mohammad Taghi; Parsaee, Heydar

Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 24, Number 4, August 2009 , pp. 918-929(12)

Publisher: Informa Healthcare

Potent Triazolothione Inhibitor of Heat-Shock Protein-90

Authors: Feldman, Richard I.; Mintzer, Bob; Zhu, Daguang; Wu, James M.; Biroc, Sandra L.; Yuan, Shendong; Emayan, Kumar; Chang, Zheng; Chen, Deborah; Arnaiz, Damian O.; Bryant, Judi; Ge, Xue Snow; Whitlow, Marc; Adler, Marc; Polokoff, Mark A.; Li, Wei-Wei; Ferrer, Mike; Sato, Takashi; Gu, Jian-Ming; Shen, Jun; Tseng, Jih-Lie; Dinter, Harald; Buckman, Brad

Source: Chemical Biology & Drug Design, Volume 74, Number 1, July 2009 , pp. 43-50(8)

Publisher: Blackwell Publishing