Probing Multidrug Resistance P-glycoprotein Transporter Activity with SPECT Radiopharmaceuticals
Keywords: 11C-verapamil; 99mTc-Furifosmin; 99mTc-Sestamibi; ABC transporters; ATP-binding cassette (ABC); Alzheimer's Disease (AD); Blood-brain barrier; Cancer; Creutzfeldt-Jakob disease; Cyclosporin; Gene therapy; LY335979; Metal complexes; Multidrug Resistance; Multidrug resistance; Multiple myeloma (MM); Nucleotide-binding domains (NBDs); P-glycoprotein; PET; PSC 833; Parkinsonian syndrome; Pgp activity; Pgp expression; Pgp inhibitors; Pgp substrate; Q-complexes; Quinidine; Radiopharmaceuticals; SPECT; Schiff-base Ga(III) complexes; Tariquidar; Technetium-99m; Transmembrane domains; Verapamil; blood-brain barrier; cancer; gene therapy; metal complexes; radiopharmaceuticals; technetium-99m; valspodar
Document Type: Research Article
Affiliations: Mallinckrodt Institute of Radiology, Washington University Medical School, Box 8225, 510 S.Kingshighway Blvd. St. Louis, MO 63110.
Publication date: 01 December 2010
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