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Publisher: Elsevier

Volume 13, Number 16, 18 August 2003

Editorial board
pp. CO2-CO2(1)

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Contents List
pp. iii-v(3)

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Graphical Abstracts
pp. 2613-2623(11)

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Hit-to-Lead studies: The discovery of potent, orally bioavailable triazolethiol CXCR2 receptor antagonists
pp. 2625-2628(4)
Authors: Baxter, A.; Bennion, C.; Bent, J.; Boden, K.; Brough, S.; Cooper, A.; Kinchin, E.; Kindon, N.; McInally, T.; Mortimore, M.; Roberts, B.; Unitt, J.

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Antitumor activity of unsaturated fatty acid esters of 4'-demethyldeoxypodophyllotoxin
pp. 2629-2632(4)
Authors: You, Y.; Kim, Y.; Nam, N.; Ahn B.-Z.

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Facile preparation of DNA-tagged carbohydrates
pp. 2633-2636(4)
Authors: Sando, S.; Matsui, K.; Niinomi, Y.; Sato, N.; Aoyama, Y.

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4-Phenyl-4H-pyrans as IKCa channel blockers
pp. 2637-2639(3)
Authors: Urbahns, K.; Horvath, E.; Stasch, J.; Mauler, F.

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Pyrimidinone antibiotics-heterocyclic analogues with improved antibacterial spectrum
pp. 2641-2645(5)
Authors: Brands, M.; Grande, Y.C.; Endermann, R.; Gahlmann, R.; Kruger, J.; Raddatz, S.

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Sub-Nanomolar hMC1R Agonists by End-Capping of the Melanocortin Tetrapeptide His-d-Phe-Arg-Trp-NH2
pp. 2647-2650(4)
Authors: Koikov, L.N.; Ebetino, F.H.; Solinsky, M.G.; Cross-Doersen, D.; Knittel, J.J.

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Anti-Androgens with full antagonistic activity toward human prostate tumor LNCaP cells with mutated androgen receptor
pp. 2655-2658(4)
Authors: Ishioka, T.; Tanatani, A.; Nagasawa, K.; Hashimoto, Y.

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Design, synthesis and antimalarial activity of novel, quinoline-Based, zinc metallo-aminopeptidase inhibitors
pp. 2659-2662(4)
Authors: Flipo, M.; Florent, I.; Grellier, P.; Sergheraert, C.; Deprez-Poulain, R.

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Hypocholesterolemic activity of hesperetin derivatives
pp. 2663-2665(3)
Authors: Jeong, T.; Kim, E.E.; Lee, C.; Oh, J.; Moon, S.; Lee, W.S.; Oh, G.; Lee, S.; Bok, S.

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Synthesis and antioxidant efficiency of a new amphiphilic spin-trap derived from PBN and lipoic acid
pp. 2673-2676(4)
Authors: Durand, G.; Polidori, A.; Salles, J.P.; Prost, M.; Durand, P.; Pucci, B.

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2-Oxoglutarate analogue inhibitors of hif prolyl hydroxylase
pp. 2677-2680(4)
Authors: Mole, D.R.; Schlemminger, I.; McNeill, L.A.; Hewitson, K.S.; Pugh, C.W.; Ratcliffe, P.J.; Schofield, C.J.

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Anti-atherogenic effects of 3,4-Dihydroxy hydrocinnamides
pp. 2681-2682(2)
Authors: Lee, S.; Lee, C.; Oh, J.; Kim, E.E.; Choi, Y.; Kim, E.; Lee, W.S.; Bok, S.; Jeong T.-S.

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Oxime bond formation for the covalent attachment of oligonucleotides on glass support
pp. 2683-2686(4)
Authors: Defrancq, E.; Hoang, A.; Vinet, F.; Dumy, P.

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Synthesis and preliminary evaluation of (R,R)(S,S) 5-(2-(2-[4-(2-[18F]fluoroethoxy)phenyl]-1-methylethylamino)-1-hydroxy ethyl )-benzene-1,3-diol ([18F]FEFE) for the in vivo visualisation and quantification of the 2-adrenergic receptor status in lung
pp. 2687-2692(6)
Authors: Schirrmacher, E.; Schirrmacher, R.; Thews, O.; Dillenburg, W.; Helisch, A.; Wessler, I.; Buhl, R.; Hohnemann, S.; Buchholz, H.; Bartenstein, P.; Machulla, H.; Rosch, F.

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Search compounds with antimicrobial activity by applying molecular topology to selected quinolones
pp. 2699-2702(4)
Authors: Mut-Ronda, S.; Salabert-Salvador, M.T.; Duart, M.J.; Anton-Fos, G.M.

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A specific anti-Helicobacter pylori agent NE2001: synthesis and its effect on the growth of H. pylori
pp. 2703-2707(5)
Authors: Cheng, N.; Xie, J.; Zhang, M.; Shu, C.; Zhu D.-X.

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Structure-activity relationships of the peptide deformylase inhibitor BB-3497: modification of the methylene spacer and the P1' side chain
pp. 2709-2713(5)
Authors: Davies, S.J.; Ayscough, A.P.; Beckett, R.P.; Bragg, R.A.; Clements, J.M.; Doel, S.; Grew, C.; Launchbury, S.B.; Perkins, G.M.; Pratt, L.M.; Smith, H.K.; Spavold, Z.M.; Thomas, S.W.; Todd, R.S.; Whittaker, M.

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Structure-activity relationships of the peptide deformylase inhibitor BB-3497: modification of the P2' and P3' side chains
pp. 2715-2718(4)
Authors: Davies, S.J.; Ayscough, A.P.; Beckett, R.P.; Clements, J.M.; Doel, S.; Pratt, L.M.; Spavold, Z.M.; Thomas, S.W.; Whittaker, M.

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Synthesis of 3a,4-dihydro-3H-[1]benzopyrano[4,3-c]isoxazoles, displaying combined 5-HT uptake inhibiting and α2-adrenoceptor antagonistic activities: a novel series of potential antidepressants
pp. 2719-2725(7)
Authors: Andres, J.I.; Alcazar, J.; Alonso, J.M.; Alvarez, R.M.; Cid, J.M.; de Lucas, A.I.; Fernandez, J.; Martinez, S.; Nieto, C.; Pastor, J.; Bakker, M.H.; Biesmans, I.; Heylen, L.I.; Megens, A.A.

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Effect of the acyl groups on O->N acyl migration in the water-soluble prodrugs of HIV-1 protease inhibitor
pp. 2727-2730(4)
Authors: Hamada, Y.; Matsumoto, H.; Kimura, T.; Hayashi, Y.; Kiso, Y.

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Synthesis and pharmacological evaluation of novel non-lactone analogues of camptothecin
pp. 2731-2735(5)
Authors: Hautefaye, P.; Cimetiere, B.; Pierre, A.; Leonce, S.; Hickman, J.; Laine, W.; Bailly, C.; Lavielle, G.

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Structure-activity relationships of azasugar-based MMP/ADAM inhibitors
pp. 2737-2740(4)
Authors: Moriyama, H.; Tsukida, T.; Inoue, Y.; Kondo, H.; Yoshino, K.; Nishimura S.-I.

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Design, synthesis and evaluation of novel azasugar-based MMP/ADAM inhibitors
pp. 2741-2744(4)
Authors: Moriyama, H.; Tsukida, T.; Inoue, Y.; Kondo, H.; Yoshino, K.; Nishimura S.-I.

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Topological virtual screening: A way to find new anticonvulsant drugs from chemical diversity
pp. 2749-2754(6)
Authors: Bruno-Blanch, L.; Galvez, J.; Garcia-Domenech, R.

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Conformationally-restricted analogues of efflux pump inhibitors that potentiate the activity of levofloxacin in Pseudomonas aeruginosa
pp. 2755-2758(4)
Authors: Renau, T.E.; Leger, R.; Filonova, L.; Flamme, E.M.; Wang, M.; Yen, R.; Madsen, D.; Griffith, D.; Chamberland, S.; Dudley, M.N.; Lee, V.J.; Lomovskaya, O.; Watkins, W.J.; Ohta, T.; Nakayama, K.; Ishida, Y.

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The imidazo[2,1-a]isoindole system. A new skeletal basis for antiplasmodial compounds
pp. 2769-2772(4)
Authors: del Olmo, E.; Armas, M.G.; Ybarra, M.a.I.; Lopez, J.L.; Oporto, P.; Gimenez, A.; Deharo, E.; San Feliciano, A.

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Novel 3-O-acyl mesquitol analogues as free-Radical scavengers and enzyme inhibitors: synthesis, biological evaluation and structure-activity relationship
pp. 2777-2780(4)
Authors: Jagadeeshwar Rao, R.; Tiwari, A.K.; Kumar, U.S.; Reddy, S.V.; Ali, A.Z.; Rao, J.M.

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Design and synthesis of potent and selective macrocyclic thrombin inhibitors
pp. 2781-2784(4)
Authors: Nantermet, P.G.; Barrow, J.C.; Newton, C.L.; Pellicore, J.M.; Young, M.; Lewis, S.D.; Lucas, B.J.; Krueger, J.A.; McMasters, D.R.; Yan, Y.; Kuo, L.C.; Vacca, J.P.; Selnick, H.G.

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Antiplatelet activity of benzylisoquinoline derivatives oxidized by cerium(IV) ammonium nitrate
pp. 2789-2793(5)
Authors: Kuo, R.; Chang, F.; Wu, C.; Patnam, R.; Wang, W.; Du, Y.; Wu Y.-C.

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5-Aryl thiazolidine-2,4-diones: discovery of PPAR dual α/ agonists as antidiabetic agents
pp. 2795-2798(4)
Authors: Desai, R.C.; Han, W.; Metzger, E.J.; Bergman, J.P.; Gratale, D.F.; MacNaul, K.L.; Berger, J.P.; Doebber, T.W.; Leung, K.; Moller, D.E.; Heck, J.V.; Sahoo, S.P.

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Acetylenic TACE inhibitors. Part 1. SAR of the acyclic sulfonamide hydroxamates
pp. 2799-2803(5)
Authors: Levin, J.I.; Chen, J.M.; Cheung, K.; Cole, D.; Crago, C.; Santos, E.D.; Du, X.; Khafizova, G.; MacEwan, G.; Niu, C.; Salaski, E.J.; Zask, A.; Cummons, T.; Sung, A.; Xu, J.; Zhang, Y.; Xu, W.; Ayral-Kaloustian, S.; Jin, G.; Cowling, R.; Barone, D.; Mohler, K.M.; Black, R.A.; Skotnicki, J.S.

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Synthesis and evaluation of ether and halogenated derivatives of mannopeptimycin glycopeptide antibiotics
pp. 2805-2808(4)
Authors: Sum P.-E.; How, D.; Torres, N.; Petersen, P.J.; Ashcroft, J.; Graziani, E.I.; Koehn, F.E.; Mansour, T.S.

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Pyrrolo[2,3-h]quinolinones: synthesis and photochemotherapic activity
pp. 2809-2811(3)
Authors: Barraja, P.; Diana, P.; Lauria, A.; Montalbano, A.; Almerico, A.M.; Dattolo, G.; Cirrincione, G.; Viola, G.; Dall'Acqua, F.

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