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Publisher: Elsevier

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Volume 13, Number 8, 17 April 2003

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Editorial board
pp. CO2-CO2(1)

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Peptide nucleic acid-metal complex conjugates: facile modulation of PNA-DNA duplex stability
pp. 1399-1401(3)
Authors: Mokhir, A.; Stiebing, R.; Kraemer, R.

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3D-QSAR Studies on thieno[3,2-d]pyrimidines as Phosphodiesterase IV Inhibitors
pp. 1403-1408(6)
Authors: Chakraborti, A.K.; Gopalakrishnan, B.; Sobhia, M.E.; Malde, A.

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Peptoid mimics of agouti related protein
pp. 1409-1413(5)
Authors: Thompson, D.A.; Chai, B.; Rood, H.L.E.; Siani, M.A.; Douglas, N.R.; Gantz, I.; Millhauser, G.L.

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Discovery and SAR of novel Naphthyridines as potent inhibitors of spleen tyrosine kinase (SYK)
pp. 1415-1418(4)
Authors: Cywin, C.L.; Zhao, B.; McNeil, D.W.; Hrapchak, M.; Prokopowicz, A.S.; Goldberg, D.R.; Morwick, T.M.; Gao, A.; Jakes, S.; Kashem, M.; Magolda, R.L.; Soll, R.M.; Player, M.R.; Bobko, M.A.; Rinker, J.; DesJarlais, R.L.; Winters, M.P.

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Identification of a broad-Spectrum azasordarin with improved pharmacokinetic properties
pp. 1419-1423(5)
Authors: Serrano-Wu, M.H.; Laurent, D.R.S.; Carroll, T.M.; Dodier, M.; Gao, Q.; Gill, P.; Quesnelle, C.; Marinier, A.; Mazzucco, C.E.; Regueiro-Ren, A.; Stickle, T.M.; Wu, D.; Yang, H.; Yang, Z.; Zheng, M.; Zoeckler, M.E.; Vyas, D.M.; Balasubramanian, B.N.

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Design, synthesis and biological activity of -carboline-based type-5 phosphodiesterase inhibitors
pp. 1425-1428(4)
Authors: Maw, G.N.; Allerton, C.M.N.; Gbekor, E.; Million, W.A.

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Design and synthesis of S-(-)-2-[[4-(napht-1-yl)piperazin-1-yl]methyl]-1,4-dioxoperhydropyrrolo[1,2- a]pyrazine (CSP-2503) using computational simulation. A 5-HT1A receptor agonist
pp. 1429-1432(4)
Authors: Lopez-Rodrguez, M.L.; Morcillo, M.J.; Fernandez, E.; Benhamu, B.; Tejada, I.; Ayala, D.; Viso, A.; Olivella, M.; Pardo, L.; Delgado, M.; Manzanares, J.; Fuentes, J.A.

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Leporin B: a novel hexokinase II gene inducing agent from an unidentified fungus
pp. 1433-1435(3)
Authors: Zhang, C.; Jin, L.; Mondie, B.; Mitchell, S.S.; Castelhano, A.L.; Cai, W.; Bergenhem, N.

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Novel Openers of Ca2+-Dependent Large-Conductance Potassium Channels: Symmetrical Pharmacophore and Electrophysiological Evaluation of Bisphenols
pp. 1437-1439(3)
Authors: Li, Y.; Johnson, G.; Romine, J.L.; Meanwell, N.A.; Martin, S.W.; Dworetzky, S.I.; Boissard, C.G.; Gribkoff, V.K.; Starrett, J.E.

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3-Amino-4-sulfonylpyridinone acetamide and related pyridothiadiazine thrombin inhibitors
pp. 1441-1444(4)
Authors: Sanderson, P.E.J.; Cutrona, K.J.; Savage, K.L.; Naylor-Olsen, A.M.; Bickel, D.J.; Bohn, D.L.; Clayton, F.C.; Krueger, J.A.; Lewis, S.D.; Lucas, B.J.; Lyle, E.A.; Wallace, A.A.; Welsh, D.C.; Yan, Y.

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High-throughput synthesis and optimization of thrombin inhibitors via urazole α-addition and Michael addition
pp. 1445-1449(5)
Authors: Boatman, P.D.; Urban, J.; Nguyen, M.; Qabar, M.; Kahn, M.

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Analogues of dealanylalahopcin are inhibitors of human HIF prolyl hydroxylases
pp. 1451-1454(4)
Authors: Schlemminger, I.; Mole, D.R.; McNeill, L.A.; Dhanda, A.; Hewitson, K.S.; Tian, Y.; Ratcliffe, P.J.; Pugh, C.W.; Schofield, C.J.

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Synthesis and evaluation of a novel series of farnesyl protein transferase inhibitors as non-peptidic CAAX tetrapeptide analogues
pp. 1455-1458(4)
Authors: Perez, M.; Maraval, C.; Dumond, S.; Lamothe, M.; Schambel, P.; Etievant, C.; Hill, B.

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From pure FPP to mixed FPP and CAAX competitive inhibitors of farnesyl protein transferase
pp. 1459-1462(4)
Authors: Lannuzel, M.; Lamothe, M.; Schambel, P.; Etievant, C.; Hill, B.; Perez, M.

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Design, synthesis, and structure-activity relationship of a new class of amidinophenylurea-based factor VIIa inhibitors
pp. 1463-1467(5)
Authors: Klingler, O.; Matter, H.; Schudok, M.; Bajaj, S.P.; Czech, J.; Lorenz, M.; Nestler, H.P.; Schreuder, H.; Wildgoose, P.

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Structure-based design of inhibitors of human l-xylulose reductase modelled into the active site of the enzyme
pp. 1469-1474(6)
Authors: Carbone, V.; Darmanin, C.; Ishikura, S.; Hara, A.; El-Kabbani, O.

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First enantiodivergent Baeyer-Villiger oxidation by recombinant whole-Cells expressing two monooxygenases from Brevibacterium
pp. 1479-1482(4)
Authors: Mihovilovic, M.D.; Rudroff, F.; Muller, B.; Stanetty, P.

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Phenylbutyrates as potent, orally bioavailable vitronectin receptor (integrin αv3) antagonists
pp. 1483-1486(4)
Authors: Miller, W.H.; Manley, P.J.; Cousins, R.D.; Erhard, K.F.; Heerding, D.A.; Kwon, C.; Ross, S.T.; Samanen, J.M.; Takata, D.T.; Uzinskas, I.N.; Yuan, C.C.K.; Haltiwanger, R.C.; Gress, C.J.; Lark, M.W.; Hwang, S.; James, I.E.; Rieman, D.J.; Willette, R.N.; Yue, T.; Azzarano, L.M.; Salyers, K.L.; Smith, B.R.; Ward, K.W.; Johanson, K.O.; Huffman, W.F.

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Synthesis and SAR of bicyclic heteroaryl hydroxamic acid MMP and TACE inhibitors
pp. 1487-1490(4)
Authors: Zask, A.; Gu, Y.; Albright, J.D.; Du, X.; Hogan, M.; Levin, J.I.; Chen, J.M.; Killar, L.M.; Sung, A.; DiJoseph, J.F.; Sharr, M.A.; Roth, C.E.; Skala, S.; Jin, G.; Cowling, R.; Mohler, K.M.; Barone, D.; Black, R.; March, C.; Skotnicki, J.S.

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Photo-oxidation of duplex DNA with the stable trioxatriangulenium ion
pp. 1491-1494(4)
Authors: Pothukuchy, A.; Ellapan, S.; Gopidas, K.R.; Salazar, M.

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Oxyguanidines: application to non-peptidic phenyl-based thrombin inhibitors
pp. 1495-1498(4)
Authors: Tomczuk, B.; Lu, T.; Soll, R.M.; Fedde, C.; Wang, A.; Murphy, L.; Crysler, C.; Dasgupta, M.; Eisennagel, S.; Spurlino, J.; Bone, R.

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