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Publisher: Elsevier

Volume 13, Number 7, 7 April 2003

Editorial board
pp. CO2-CO2(1)

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Graphical Abstracts - 9 pages
pp. 1221-1230(10)

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Synthesis of quinolinyl/isoquinolinyl[a]pyrrolo [3,4-c] carbazoles as cyclin D1/CDK4 inhibitors
pp. 1231-1235(5)
Authors: Zhu, G.; Conner, S.; Zhou, X.; Shih, C.; Brooks, H.B.; Considine, E.; Dempsey, J.A.; Ogg, C.; Patel, B.; Schultz, R.M.; Spencer, C.D.; Teicher, B.; Watkins, S.A.

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A new synthesis of cytoxazone and its diastereomers provides key initial SAR information
pp. 1237-1239(3)
Authors: Carter, P.H.; LaPorte, J.R.; Scherle, P.A.; Decicco, C.P.

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Synthesis and pharmacological activity of fluorescent histamine H1 receptor antagonists related to mepyramine
pp. 1245-1248(4)
Authors: Li, L.; Kracht, J.; Peng, S.; Bernhardt, G.; Buschauer, A.

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Synthesis of low molecular weight compounds with complement inhibition activity
pp. 1249-1251(3)
Authors: Master, H.E.; Khan, S.I.; Poojari, K.A.

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Antimycobacterial pimarane diterpenes from the Fungus Diaporthe sp.
pp. 1253-1255(3)
Authors: Dettrakul, S.; Kittakoop, P.; Isaka, M.; Nopichai, S.; Suyarnsestakorn, C.; Tanticharoen, M.; Thebtaranonth, Y.

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Replacing the pyrophosphate group of HMB-PP by a diphosphonate function abrogates Its potential to activate human  T cells but does not lead to competitive antagonism
pp. 1257-1260(4)
Authors: Reichenberg, A.; Hintz, M.; Kletschek, Y.; Kuhl, T.; Haug, C.; Engel, R.; Moll, J.; Ostrovsky, D.N.; Jomaa, H.; Eberl, M.

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The inhibitory effects of squalene-derived triterpenes on protein phosphatase PP2A
pp. 1261-1264(4)
Authors: Souto, M.L.; Manrquez, C.P.; Norte, M.; Leira, F.; Fernandez, J.J.

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Conformational restriction of methionyl tRNA synthetase inhibitors leading to analogues with potent inhibition and excellent gram-Positive antibacterial activity
pp. 1265-1268(4)
Authors: Jarvest, R.L.; Berge, J.M.; Brown, P.; Houge-Frydrych, C.S.V.; O'Hanlon, P.J.; McNair, D.J.; Pope, A.J.; Rittenhouse, S.

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Novel indole-based inhibitors of IMPDH: introduction of hydrogen bond acceptors at indole C-3
pp. 1273-1276(4)
Authors: Watterson, S.H.; Dhar, T.G.M.; Ballentine, S.K.; Shen, Z.; Barrish, J.C.; Cheney, D.; Fleener, C.A.; Rouleau, K.A.; Townsend, R.; Hollenbaugh, D.L.; Iwanowicz, E.J.

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Phenylacetic acid derivatives as hPPAR agonists
pp. 1277-1280(4)
Authors: Santini, C.; Berger, G.D.; Han, W.; Mosley, R.; MacNaul, K.; Berger, J.; Doebber, T.; Wu, M.; Moller, D.E.; Tolman, R.L.; Sahoo, S.P.

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Synthesis and biological activities of phthalocyanine-estradiol conjugates
pp. 1287-1290(4)
Authors: Khan, E.H.; Ali, H.; Tian, H.; Rousseau, J.; Tessier, G.; Shafiullah; van Lier, J.E.

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[3H]-(R)-NPTS, a radioligand for the type 1 glycine transporter
pp. 1291-1292(2)
Authors: Lowe, J.A.; Drozda, S.E.; Fisher, K.; Strick, C.; Lebel, L.; Schmidt, C.; Hiller, D.; Zandi, K.S.

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Synthesis and biological evaluation of 4-[3-biphenyl-2-yl-1-hydroxy-1-(3-methyl-3H-imidazol-4-yl)-prop-2-ynyl]-1-yl -benzonitrile as novel farnesyltransferase inhibitor
pp. 1293-1296(4)
Authors: Lin N.-H.; Wang, L.; Cohen, J.; Gu, W.; Frost, D.; Zhang, H.; Rosenberg, S.; Sham, H.

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Potent and selective aggrecanase inhibitors containing cyclic P1 substituents
pp. 1297-1300(4)
Authors: Cherney, R.J.; Mo, R.; Meyer, D.T.; Wang, L.; Yao, W.; Wasserman, Z.R.; Liu, R.; Covington, M.B.; Tortorella, M.D.; Arner, E.C.; Qian, M.; Christ, D.D.; Trzaskos, J.M.; Newton, R.C.; Magolda, R.L.; Decicco, C.P.

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Novel and potent human and rat 3-Adrenergic receptor agonists containing substituted 3-indolylalkylamines
pp. 1301-1305(5)
Authors: Harada, H.; Hirokawa, Y.; Suzuki, K.; Hiyama, Y.; Oue, M.; Kawashima, H.; Yoshida, N.; Furutani, Y.; Kato, S.

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Structure-activity relationship of cyclic peptide penta-c[Asp-His6-DPhe7-Arg8-Trp9-Lys ]-NH2 at the human melanocortin-1 and -4 receptors: His6 substitution
pp. 1307-1311(5)
Authors: Cheung A.W.-H.; Danho, W.; Swistok, J.; Qi, L.; Kurylko, G.; Rowan, K.; Yeon, M.; Franco, L.; Chu, X.; Chen, L.; Yagaloff, K.

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Novel 6-aryl-1,4-dihydrobenzo[d]oxazine-2-thiones as potent, selective, and orally active nonsteroidal progesterone receptor agonists
pp. 1313-1316(4)
Authors: Zhang, P.; Terefenko, E.A.; Fensome, A.; Wrobel, J.; Winneker, R.; Zhang, Z.

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Novel 5-aryl-1,3-dihydro-indole-2-thiones - potent, orally active progesterone receptor agonists
pp. 1317-1320(4)
Authors: Fensome, A.; Koko, M.; Wrobel, J.; Zhang, P.; Zhang, Z.; Cohen, J.; Lundeen, S.; Rudnick, K.; Zhu, Y.; Winneker, R.

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Investigation of an antibody-ligase. evidence for strain-induced catalysis
pp. 1321-1324(4)
Authors: Savinov, S.N.; Hirschmann, R.; Benkovic, S.J.; Smith, A.B.

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Synthesis and SAR of aminoalkoxy-biaryl-4-carboxamides: novel and selective histamine H3 receptor antagonists
pp. 1325-1328(4)
Authors: Faghih, R.; Dwight, W.; Pan, J.B.; Fox, G.B.; Krueger, K.M.; A. Esbenshade, T.; McVey, J.M.; Marsh, K.; Bennani, Y.L.; Hancock, A.A.

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Benzo[f]naphtyridones: a new family of topical antibacterial agents active on multi-resistant Gram-positive pathogens
pp. 1329-1331(3)
Authors: Tabart, M.; Picaut, G.; Lavergne, M.; Wentzler, S.; Malleron, J.; Dutka-Malen, S.; Berthaud, N.

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Inhibition of telomerase by BIBR 1532 and related analogues
pp. 1333-1336(4)
Authors: Barma, D.K.; Elayadi, A.; Falck, J.R.; Corey, D.R.

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Microsomal triglyceride transfer protein inhibitors: discovery and synthesis of alkyl phosphonates as potent MTP inhibitors and cholesterol lowering agents
pp. 1337-1340(4)
Authors: Magnin, D.R.; Biller, S.A.; Wetterau, J.; Robl, J.A.; Dickson, J.K.; Taunk, P.; Harrity, T.W.; Lawrence, R.M.; Sun, C.; Wang, T.; Logan, J.; Fryszman, O.; Connolly, F.; Jolibois, K.; Kunselman, L.

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Synthesis and structure-Activity relationships of aroylpyrrole alkylamide bradykinin (B2) antagonists
pp. 1341-1344(4)
Authors: Youngman, M.A.; Carson, J.R.; Lee, J.S.; Dax, S.L.; Zhang, S.; Colburn, R.W.; Stone, D.J.; Codd, E.E.; Jetter, M.C.

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Identification of novel and potent isoquinoline aminooxazole-Based IMPDH inhibitors
pp. 1345-1348(4)
Authors: Chen, P.; Norris, D.; Haslow, K.D.; Murali Dhar, T.G.; Pitts, W.J.; Watterson, S.H.; Cheney, D.L.; Bassolino, D.A.; Fleener, C.A.; Rouleau, K.A.; Hollenbaugh, D.L.; Townsend, R.M.; Barrish, J.C.; Iwanowicz, E.J.

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Reaction of Thiols with 7-Methylbenzopentathiepin
pp. 1349-1352(4)
Authors: Chatterji, T.; Gates, K.S.

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Pharmacokinetic optimization of 3-amino-6-chloropyrazinone acetamide thrombin inhibitors. implementation of P3 pyridine N-Oxides to deliver an orally bioavailable series containing P1 N-Benzylamides
pp. 1353-1357(5)
Authors: Burgey, C.S.; Robinson, K.A.; Lyle, T.A.; Nantermet, P.G.; Selnick, H.G.; Isaacs, R.C.A.; Lewis, S.D.; Lucas, B.J.; Krueger, J.A.; Singh, R.; Miller-Stein, C.; White, R.B.; Wong, B.; Lyle, E.A.; Stranieri, M.T.; Cook, J.J.; McMasters, D.R.; Pellicore, J.M.; Pal, S.; Wallace, A.A.; Clayton, F.C.; Bohn, D.; Welsh, D.C.; Lynch, J.J.; Yan, Y.; Chen, Z.; Kuo, L.; Gardell, S.J.; Shafer, J.A.; Vacca, J.P.

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Aryl tetrahydropyridine inhibitors of farnesyltransferase: glycine, phenylalanine and histidine derivatives
pp. 1359-1362(4)
Authors: Gwaltney, S.L.; O'Connor, S.J.; Nelson, L.T.J.; Sullivan, G.M.; Imade, H.; Wang, W.; Hasvold, L.; Li, Q.; Cohen, J.; Gu, W.; Tahir, S.K.; Bauch, J.; Marsh, K.; Ng, S.; Frost, D.J.; Zhang, H.; Muchmore, S.; Jakob, C.G.; Stoll, V.; Hutchins, C.; Rosenberg, S.H.; Sham, H.L.

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Aryl tetrahydropyridine inhibitors of farnesyltransferase: bioavailable analogues with improved cellular potency
pp. 1363-1366(4)
Authors: Gwaltney, S.L.; O'Connor, S.J.; Nelson, L.T.J.; Sullivan, G.M.; Imade, H.; Wang, W.; Hasvold, L.; Li, Q.; Cohen, J.; Gu, W.; Tahir, S.K.; Bauch, J.; Marsh, K.; Ng, S.; Frost, D.J.; Zhang, H.; Muchmore, S.; Jakob, C.G.; Stoll, V.; Hutchins, C.; Rosenberg, S.H.; Sham, H.L.

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Novel and selective imidazole-containing biphenyl inhibitors of protein farnesyltransferase
pp. 1367-1371(5)
Authors: Curtin, M.L.; Florjancic, A.S.; Cohen, J.; Gu, W.; Frost, D.J.; Muchmore, S.W.; Sham, H.L.

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Azalide 3,6-Ketals: antibacterial activity and structure-Activity relationships of aryl and hetero aryl substituted analogues
pp. 1373-1375(3)
Authors: Sakya, S.M.; Bertinato, P.; Pratt, B.; Suarez-Contreras, M.; Lundy, K.M.; Minich, M.L.; Cheng, H.; Ziegler, C.B.; Kamicker, B.J.; Hayashi, S.F.; Santoro, S.L.; George, D.M.; Bertsche, C.D.

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Adsorbed surfactants for affinity chromatography - end-group modification of ethylene glycol polymers
pp. 1381-1384(4)
Authors: Yanic, C.; Bredenkamp, M.W.; Jacobs, E.P.; Swart, P.

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