Publisher: Elsevier

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Volume 13, Number 2, 20 January 2003

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Editorial Board
pp. CO2-CO2(1)

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Contents List
pp. iii

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Graphical Abstracts
pp. 153-160(8)

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Small, low nanomolar, noncovalent thrombin inhibitors lacking a group to fill the 'Distal binding pocket'
pp. 161-164(4)
Authors: Sanderson, P.E.J.; Cutrona, K.J.; Dyer, D.L.; Krueger, J.A.; Kuo, L.C.; Lewis, S.D.; Lucas, B.J.; Yan, Y.

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Highly potent and selective αV3-receptor antagonists: solid-phase synthesis and SAR of 1-substituted 4-amino-1H-pyrimidin-2-ones
pp. 165-169(5)
Authors: Zechel, C.; Backfisch, G.; Delzer, J.; Geneste, H.; Graef, C.; Hornberger, W.; Kling, A.; Lange, U.E.W.; Lauterbach, A.; Seitz, W.; Subkowski, T.

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New arylpiperazine derivatives with high affinity for α1A, D2 and 5-HT2A receptors
pp. 175-178(4)
Authors: Gonzalez-Gomez, J.C.; Santana, L.; Uriarte, E.; Brea, J.; Villazon, M.; Loza, M.I.; de Luca, M.; Rivas, M.E.; Montenegro, G.Y.; Fontenla, J.A.

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A new series of potent benzodiazepine -secretase inhibitors
pp. 179-183(5)
Authors: Churcher, I.; Ashton, K.; Butcher, J.W.; Clarke, E.E.; Harrison, T.; Lewis, H.D.; Owens, A.P.; Teall, M.R.; Williams, S.; Wrigley, J.D.J.

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New highly active taxoids from 9-dihydrobaccatin-9,10-acetals. Part 3
pp. 185-190(6)
Authors: Takeda, Y.; Yoshino, T.; Uoto, K.; Chiba, J.; Ishiyama, T.; Iwahana, M.; Jimbo, T.; Tanaka, N.; Terasawa, H.; Soga, T.

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Design, synthesis and antifungal activity of a novel water soluble prodrug of antifungal triazole
pp. 191-196(6)
Authors: Ohwada, J.; Tsukazaki, M.; Hayase, T.; Oikawa, N.; Isshiki, Y.; Fukuda, H.; Mizuguchi, E.; Sakaitani, M.; Shiratori, Y.; Yamazaki, T.; Ichihara, S.; Umeda, I.; Shimma, N.

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Synthesis of 2-substituted-pyrrolidinethiourea derivatives and their antagonist effect on vanilloid receptor
pp. 197-200(4)
Authors: Park, H.; Park, M.; Choi, J.; Choi, S.; Lee, J.; Suh, Y.; Oh, U.; Lee, J.; Kim, H.; Park, Y.; Jeong, Y.S.; Choi, J.K.; Jew S.-s.

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[18F]FMDAA1106 and [18F]FEDAA1106: two positron-Emitter labeled ligands for peripheral benzodiazepine receptor (PBR)
pp. 201-204(4)
Authors: Zhang M.-R.; Maeda, J.; Furutsuka, K.; Yoshida, Y.; Ogawa, M.; Suhara, T.; Suzuki, K.

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Novel inhibitors of neuronal nitric oxide synthase with potent antioxidant properties
pp. 209-212(4)
Authors: Auvin, S.; Auguet, M.; Navet, E.; Harnett, J.J.; Viossat, I.; Schulz, J.; Bigg, D.; Chabrier, P.

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Affinity labeling of the nuclear vitamin D receptor with nonsteroidal alkylating agents
pp. 213-216(4)
Authors: Fernandez-Gacio, A.; Fernandez-Marcos, C.; Swamy, N.; Ray, R.

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4-Alkoxy-2,6-diaminopyrimidine derivatives: inhibitors of cyclin dependent kinases 1 and 2
pp. 217-222(6)
Authors: Mesguiche, V.; Parsons, R.J.; Arris, C.E.; Bentley, J.; Boyle, F.T.; Curtin, N.J.; Davies, T.G.; Endicott, J.A.; Gibson, A.E.; Golding, B.T.; Griffin, R.J.; Jewsbury, P.; Johnson, L.N.; Newell, D.R.; Noble, M.E.M.; Wang, L.Z.; Hardcastle, I.R.

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Anti-Hyperlipidemic sesquiterpenes and new sesquiterpene glycosides from the leaves of artichoke (Cynara scolymus L.): structure requirement and mode of action
pp. 223-228(6)
Authors: Shimoda, H.; Ninomiya, K.; Nishida, N.; Yoshino, T.; Morikawa, T.; Matsuda, H.; Yoshikawa, M.

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Synthesis of non-competitive inhibitors of Sphingomyelinases with significant activity
pp. 229-236(8)
Authors: Yokomatsu, T.; Murano, T.; Akiyama, T.; Koizumi, J.; Shibuya, S.; Tsuji, Y.; Soeda, S.; Shimeno, H.

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Dihydropyrimidinones-a new class of anti-Staphylococcal antibiotics
pp. 241-245(5)
Authors: Brands, M.; Endermann, R.; Gahlmann, R.; Kruger, J.; Raddatz, S.

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-Homolysine Oligomers: A New Class of Trojan Carriers
pp. 247-251(5)
Authors: Garca-Echeverra, C.; Ruetz, S.

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Methylphosphonate LNA: a locked nucleic acid with a methylphosphonate linkage
pp. 253-256(4)
Authors: Lauritsen, A.; Dahl, B.M.; Dahl, O.; Vester, B.; Wengel, J.

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Design and synthesis of novel PPARα// triple activators using a known PPARα/ dual activator as structural template
pp. 257-260(4)
Authors: Mogensen, J.P.; Jeppesen, L.; Bury, P.S.; Pettersson, I.; Fleckner, J.; Nehlin, J.; Frederiksen, K.S.; Albrektsen, T.; Din, N.; Mortensen, S.B.; Svensson, L.A.; Wassermann, K.; Wulff, E.M.; Ynddal, L.; Sauerberg, P.

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Retinoic acid receptor ligands based on the 6-cyclopropyl-2,4-hexadienoic acid
pp. 261-264(4)
Authors: Farmer, L.J.; Zhi, L.; Jeong, S.; Lamph, W.W.; Osburn, D.L.; Croston, G.; Flatten, K.S.; Heyman, R.A.; Nadzan, A.M.

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The preparation of (S)-Aspartate semi-aldehyde appropriate for use in biochemical studies
pp. 265-267(3)
Authors: Roberts, S.J.; Morris, J.C.; Dobson, R.C.J.; Gerrard, J.A.

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Discovery of a series of (4,5-Dihydroimidazol-2-yl)-biphenylamine 5-HT7 agonists
pp. 269-271(3)
Authors: Parikh, V.; Welch, W.M.; Schmidt, A.W.

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p38MAP kinase inhibitors. part 1: design and development of a new class of potent and highly selective inhibitors based on 3,4-dihydropyrido[3,2-d]pyrimidone scaffold
pp. 273-276(4)
Authors: Natarajan, S.R.; Wisnoski, D.D.; Singh, S.B.; Stelmach, J.E.; O'Neill, E.A.; Schwartz, C.D.; Thompson, C.M.; Fitzgerald, C.E.; O'Keefe, S.J.; Kumar, S.; Hop, C.E.C.A.; Zaller, D.M.; Schmatz, D.M.; Doherty, J.B.

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Design and synthesis of potent, orally bioavailable dihydroquinazolinone inhibitors of p38 MAP kinase
pp. 277-280(4)
Authors: Stelmach, J.E.; Liu, L.; Patel, S.B.; Pivnichny, J.V.; Scapin, G.; Singh, S.; Hop, C.E.C.A.; Wang, Z.; Strauss, J.R.; Cameron, P.M.; Nichols, E.A.; O'Keefe, S.J.; O'Neill, E.A.; Schmatz, D.M.; Schwartz, C.D.; Thompson, C.M.; Zaller, D.M.; Doherty, J.B.

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A novel solid support for synthesis of oligonucleotide 3'-phosphorothioate monoesters
pp. 281-284(4)
Authors: Cheruvallath, Z.S.; Cole, D.L.; Ravikumar, V.T.

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Development of a presynaptic 5-HT1A antagonist
pp. 285-288(4)
Authors: Mattson, R.J.; Catt, J.D.; Sloan, C.P.; Gao, Q.; Carter, R.B.; Gentile, A.; Mahle, C.D.; Matos, F.F.; McGovern, R.; VanderMaelen, C.P.; Yocca, F.D.

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CRF Ligands via suzuki and negishi couplings of 3-pyridyl boronic acids or halides with 2-benzyloxy-4-chloro-3-nitropyridine
pp. 289-291(3)
Authors: Arvanitis, A.G.; Arnold, C.R.; Fitzgerald, L.W.; Frietze, W.E.; Olson, R.E.; Gilligan, P.J.; Robertson, D.W.

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Design and synthesis of factor Xa inhibitors and their prodrugs
pp. 297-300(4)
Authors: Song, Y.; Clizbe, L.; Bhakta, C.; Teng, W.; Wong, P.; Huang, B.; Tran, K.; Sinha, U.; Park, G.; Reed, A.; Scarborough, R.M.; Zhu, B.

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Synthesis and evaluation of phosphoramidate amino acid-based inhibitors of sialyltransferases
pp. 301-304(4)
Authors: Whalen, L.J.; McEvoy, K.A.; Halcomb, R.L.

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