Publisher: Elsevier

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Volume 13, Number 1, January 2003

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Antiviral activity of cyclopentenyl nucleosides against orthopox viruses (Smallpox, monkeypox and cowpox)
pp. 9-12(4)
Authors: Chu, C.K.; Jin, Y.H.; Baker, R.O.; Huggins, J.

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Synthesis and antifungal activity of 2,5-disubstituted-6-arylamino-4,7-benzimidazolediones
pp. 17-20(4)
Authors: Ryu C.-K.; Song, E.; Shim, J.; You, H.; Choi, K.U.; Choi, I.H.; Lee, E.Y.; Chae, M.J.

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True interaction mode of porcine pancreatic elastase with FR136706, a potent peptidyl inhibitor
pp. 21-24(4)
Authors: Kinoshita, T.; Nakanishi, I.; Sato, A.; Tada, T.

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Identification of a stable chymase inhibitor using a pharmacophore-Based database search
pp. 25-29(5)
Authors: Koide, Y.; Tatsui, A.; Hasegawa, T.; Murakami, A.; Satoh, S.; Yamada, H.; Kazayama, S.; Takahashi, A.

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Siphonols A-E: Novel nitric oxide inhibitors from Orthosiphon stamineus of Indonesia
pp. 31-35(5)
Authors: Awale, S.; Tezuka, Y.; Banskota, A.H.; Kadota, S.

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Synthesis and -secretase activity of APP substrate-based hydroxyethylene dipeptide isosteres
pp. 37-41(5)
Authors: Nadin, A.; Owens, A.P.; Castro, J.L.; Harrison, T.; Shearman, M.S.

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Homologues and isomers of noladin ether, a putative novel endocannabinoid: interaction with rat cannabinoid CB1 receptors
pp. 43-46(4)
Authors: Appendino, G.; Ligresti, A.; Minassi, A.; Daddario, N.; Bisogno, T.; Di Marzo, V.

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Comparison of library screening techniques used in the development of dsDNA ligands
pp. 47-50(4)
Authors: Chaltin, P.; Borgions, F.; van Aerschot, A.; Herdewijn, P.

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Structural chemistry and In vitro antitubercular activity of acetylpyridine benzoyl hydrazone and its copper complex against Mycobacterium smegmatis
pp. 51-55(5)
Authors: Patole, J.; Sandbhor, U.; Padhye, S.; Deobagkar, D.N.; Anson, C.E.; Powell, A.

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Identification of novel muscarinic M3 selective antagonists with a conformationally restricted Hyp-Pro spacer
pp. 57-60(4)
Authors: Sagara, Y.; Kimura, T.; Fujikawa, T.; Noguchi, K.; Ohtake, N.

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New tetrahydrobenzindoles as potent and selective 5-HT7 antagonists with increased In vitro metabolic stability
pp. 61-64(4)
Authors: Kikuchi, C.; Suzuki, H.; Hiranuma, T.; Koyama, M.

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Synthetic study on the unique dimeric arylpiperazine: access to the minor contaminant of aripiprazole
pp. 65-68(4)
Authors: Torisawa, Y.; Shinhama, K.; Nishi, T.; Minamikawa, J.

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Rational approaches towards reversible inhibition of type B monoamine oxidase. Design and evaluation of a novel 5H-Indeno[1,2-c]pyridazin-5-one derivative
pp. 69-73(5)
Authors: Ooms, F.; Frederick, R.; Durant, F.; Petzer, J.P.; Castagnoli, N.; van der Schyf, C.J.; Wouters, J.

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Synthesis and antimalarial activity of 2-methoxyprop-2-yl peroxides derivatives
pp. 75-77(3)
Authors: Cointeaux, L.; Berrien, J.; Peyrou, V.; Provot, O.; Ciceron, L.; Danis, M.; Robert, A.; Meunier, B.; Mayrargue, J.

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Hepatoprotective pyrrole derivatives of Lycium chinense fruits
pp. 79-81(3)
Authors: Chin, Y.; Lim, S.W.; Kim, S.; Shin, D.; Suh, Y.; Kim, Y.; Kim, Y.C.; Kim, J.

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Fluorescent bioprobes for visualization of puromycin-sensitive aminopeptidase in living cells
pp. 83-86(4)
Authors: Kakuta, H.; Koiso, Y.; Nagasawa, K.; Hashimoto, Y.

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Design and synthesis of novel benzofurans as a new class of antifungal agents targeting fungal N-myristoyltransferase. Part 3
pp. 87-91(5)
Authors: Kawasaki, K.; Masubuchi, M.; Morikami, K.; Sogabe, S.; Aoyama, T.; Ebiike, H.; Niizuma, S.; Hayase, M.; Fujii, T.; Sakata, K.; Shindoh, H.; Shiratori, Y.; Aoki, Y.; Ohtsuka, T.; Shimma, N.

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Design and synthesis of pseudo-Symmetric HIV protease inhibitors containing a novel hydroxymethylcarbonyl (HMC)-Hydrazide isostere
pp. 93-96(4)
Authors: Hidaka, K.; Kimura, T.; Hayashi, Y.; McDaniel, K.F.; Dekhtyar, T.; Colletti, L.; Kiso, Y.

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N,N-Disubstituted piperazines: synthesis and affinities at α42* and α7* neuronal nicotinic acetylcholine receptors
pp. 97-100(4)
Authors: Chen, J.; Norrholm, S.; Dwoskin, L.P.; Crooks, P.A.; Bai, D.

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Structure-activity and crystallographic analysis of benzophenone derivatives-the potential anticancer agents
pp. 101-105(5)
Authors: Hsieh H.-P.; Liou, J.; Lin, Y.; Mahindroo, N.; Chang, J.; Yang, Y.; Chern, S.; Tan, U.; Chang, C.; Chen, T.; Lin, C.; Chang, Y.; Wang, C.

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Design of novel N-(2,4-dioxo-1,2,3,4-tetrahydro-thieno[3,2-d]pyrimidin-7-yl)-guanidines as thymidine phosphorylase inhibitors, and flexible docking to a homology model
pp. 107-110(4)
Authors: Price, M.P.; Guida, W.; Jackson, T.; Nydick, J.; Gladstone, P.; Juarez, J.; Donate, F.; Ternansky, R.

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Development of an orexin-2 receptor selective agonist, [Ala11, d-Leu15]orexin-B
pp. 111-113(3)
Authors: Asahi, S.; Egashira, S.; Matsuda, M.; Iwaasa, H.; Kanatani, A.; Ohkubo, M.; Ihara, M.; Morishima, H.

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Design, synthesis, and biological evaluation of angiogenesis inhibitors: aromatic enone and dienone analogues of curcumin
pp. 115-117(3)
Authors: Robinson, T.P.; Ehlers, T.; Hubbard, I.; Bai, X.; Arbiser, J.L.; Goldsmith, D.J.; Bowen, J.P.

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1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists: modifications of the arylpropylpiperidine side chains
pp. 119-123(5)
Authors: Lynch, C.L.; Willoughby, C.A.; Hale, J.J.; Holson, E.J.; Budhu, R.J.; Gentry, A.L.; Rosauer, K.G.; Caldwell, C.G.; Chen, P.; Mills, S.G.; MacCoss, M.; Berk, S.; Chen, L.; Chapman, K.T.; Malkowitz, L.; Springer, M.S.; Gould, S.L.; DeMartino, J.A.; Siciliano, S.J.; Cascieri, M.A.; Carella, A.; Carver, G.; Holmes, K.; Schleif, W.A.; Danzeisen, R.; Hazuda, D.; Kessler, J.; Lineberger, J.; Miller, M.; Emini, E.A.

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Imidazo[4,5-b]pyridines as corticotropin releasing factor receptor ligands
pp. 125-128(4)
Authors: Arvanitis, A.G.; Rescinito, J.T.; Arnold, C.R.; Wilde, R.G.; Cain, G.A.; Sun, J.H.; Yan, J.; Teleha, C.A.; Fitzgerald, L.W.; McElroy, J.; Zaczek, R.; Hartig, P.R.; Grossman, S.; Arneric, S.P.; Gilligan, P.J.; Olson, R.E.; Robertson, D.W.

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Imidazo[4,5-c]pyridines as corticotropin releasing factor receptor ligands
pp. 129-131(3)
Authors: Arvanitis, A.G.; Rescinito, J.T.; Arnold, C.R.; Wilde, R.G.; Fitzgerald, L.W.; Zaczek, R.; Hartig, P.R.; Grossman, S.; Arneric, S.P.; Gilligan, P.J.; Olson, R.E.; Robertson, D.W.

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Structure-Activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH2 at the human melanocortin-1 and -4 receptors: histidine substitution
pp. 133-137(5)
Authors: Cheung A.W.-H.; Danho, W.; Swistok, J.; Qi, L.; Kurylko, G.; Rowan, K.; Yeon, M.; Franco, L.; Chu, X.; Chen, L.; Yagaloff, K.

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3-Acylamino-azetidin-2-one as a novel class of cysteine proteases inhibitors
pp. 139-141(3)
Authors: Zhou, N.E.; Guo, D.; Thomas, G.; Reddy, A.V.N.; Kaleta, J.; Purisima, E.; Menard, R.; Micetich, R.G.; Singh, R.

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Studies on the synthesis and anti-Osteoporosis of estrogen-GHRPs linkers
pp. 143-146(4)
Authors: Wang, C.; Cui, W.; Zhao, M.; Yang, J.; Peng, S.

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Nodulisporic acid side-Chain modifications: access to the 2'', 3'', 4'', and 6'' registers
pp. 147-150(4)
Authors: Chakravarty, P.K.; Shih, T.L.; Colletti, S.L.; Ayer, M.B.; Snedden, C.; Kuo, H.; Tyagarajan, S.; Gregory, L.; Zakson-Aiken, M.; Shoop, W.L.; Schmatz, D.M.; Wyvratt, M.; Fisher, M.H.; Meinke, P.T.

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