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Publisher: Elsevier

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Volume 12, Number 24, 16 December 2002

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Inside (Editorial Board)
pp. CO2-CO2(1)

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Author Index 2002
pp. IX-XXXIX(31)

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Contributors to this Issue
pp. vii-viii(2)

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Contents List
pp. iii

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Graphical Abstracts
pp. 3497-3504(8)

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Synthesis and cytotoxic activity of a new potent daunomycinone derivative
pp. 3505-3507(3)
Authors: Aligiannis, N.; Pouli, N.; Marakos, P.; Skaltsounis A.-L.; Pratsinis, H.

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Bioactive 4-substituted-6-methyl-2-pyrones with promising cytotoxicity against A2780 and K562 cell lines
pp. 3509-3513(5)
Authors: Marrison, L.R.; Dickinson, J.M.; Fairlamb, I.J.S.

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Synthesis of (+)-Lasonolide A: (-)-Lasonolide A is the biologically active enantiomer
pp. 3519-3520(2)
Authors: Lee, E.; Song, H.Y.; Joo, J.M.; Kang, J.W.; Kim, D.S.; Jung, C.K.; Hong, C.Y.; Jeong, S.; Jeon, K.

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Stereoselective and improved syntheses and anticancer testing of 3'-O-silatranylthymidines
pp. 3521-3523(3)
Authors: Black, C.A.; Ucci, J.W.; Vorpagel, J.S.; Mauck, M.C.; Fenlon, E.E.

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Synthesis of new targretin(R) analogues that induce apoptosis in leukemia HL-60 cells
pp. 3529-3532(4)
Authors: Winum, J.; Baghdiguian, S.; Commes, T.; Leydet, A.; Montero J.-L.

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Design and efficient synthesis of new stable 1α,25-dihydroxy-19-norvitamin D3 analogues containing amide bond
pp. 3533-3536(4)
Authors: Suhara, Y.; Kittaka, A.; Ono, K.; Kurihara, M.; Fujishima, T.; Yoshida, A.; Takayama, H.

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Optimization of a pyrazolo[1,5-a]pyrimidine class of KDR kinase inhibitors: improvements in physical properties enhance cellular activity and pharmacokinetics
pp. 3537-3541(5)
Authors: Fraley, M.E.; Rubino, R.S.; Hoffman, W.F.; Hambaugh, S.R.; Arrington, K.L.; Hungate, R.W.; Bilodeau, M.T.; Tebben, A.J.; Rutledge, R.Z.; Kendall, R.L.; McFall, R.C.; Huckle, W.R.; Coll, K.E.; Thomas, K.A.

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Synthesis of aglycon analogues of sarmentosin and Their bioactivity of lymphocyte proliferation
pp. 3543-3545(3)
Authors: Zhang, H.; Xu, R.; Hu, Z.; He, X.; Bai, D.; Li, X.; Wang, X.

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Natural and synthetic geiparvarins are strong and selective MAO-B inhibitors. synthesis and SAR studies
pp. 3551-3555(5)
Authors: Carotti, A.; Carrieri, A.; Chimichi, S.; Boccalini, M.; Cosimelli, B.; Gnerre, C.; Carotti, A.; Carrupt, P.; Testa, B.

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Synthesis and biological evaluation of aristolactams
pp. 3557-3559(3)
Authors: Couture, A.; Deniau, E.; Grandclaudon, P.; Rybalko-Rosen, H.; Leonce, S.; Pfeiffer, B.; Renard, P.

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Synthesis and biological evaluation of novel 2-(1H-imidazol-4-yl)cyclopropane carboxylic acids: key intermediates for H3 histamine receptor ligands
pp. 3561-3563(3)
Authors: Brana, M.F.; Guisado, C.; Fernando Alguacil, L.; Garrido, E.; Perez-Garca, C.; Ruiz-Gayo, M.

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Synthesis and pharmacological evaluation of a new class of peroxisome proliferator-activated receptor modulators
pp. 3565-3567(3)
Authors: Thor, M.; Beierlein, K.; Dykes, G.; Gustavsson, A.; Heidrich, J.; Jendeberg, L.; Lindqvist, B.; Pegurier, C.; Roussel, P.; Slater, M.; Svensson, S.; Sydow-Backman, M.; Thornstrom, U.; Uppenberg, J.

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17S,20S-Methanofusidic acid, a new potent semi-synthetic fusidane antibiotic
pp. 3569-3572(4)
Authors: Duvold, T.; Jorgensen, A.; Andersen, N.R.; Henriksen, A.S.; Dahl Sorensen, M.; Bjorkling, F.

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2-(Dimethylaminomethyl)-tetrahydroisoxazolopyridobenzazepine derivatives. Synthesis of a new 5-HT2C antagonist with potential anxiolytic properties
pp. 3573-3577(5)
Authors: Andres, J.I.; Alonso, J.M.; Fernandez, J.; Iturrino, L.; Martnez, P.; Meert, T.F.; Sipido, V.K.

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Synthetic studies of cis-4-Amino-l-proline derivatives as novel lipid lowering agents
pp. 3579-3581(3)
Authors: Das, S.K.; Narasimha Rao Krovvidi, V.L.; Jagadheshan, H.; Iqbal, J.

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Novel 1',1'-chain substituted Δ8-tetrahydrocannabinols
pp. 3583-3586(4)
Authors: Papahatjis, D.P.; Nikas, S.P.; Andreou, T.; Makriyannis, A.

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Isolation and antimalarial activity of peroxydisulfate oxidation products of primaquine
pp. 3587-3589(3)
Authors: Dua, V.K.; Sinha, S.N.; Biswas, S.; Valecha, N.; Puri, S.K.; Sharma, V.P.

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Reductively activated disulfide prodrugs of paclitaxel
pp. 3591-3594(4)
Authors: Vrudhula, V.M.; MacMaster, J.F.; Li, Z.; Kerr, D.E.; Senter, P.D.

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Structure-activity relationships of the peptide deformylase inhibitor BB-3497: modification of the metal binding group
pp. 3595-3599(5)
Authors: Smith, H.K.; Beckett, R.P.; Clements, J.M.; Doel, S.; East, S.P.; Launchbury, S.B.; Pratt, L.M.; Spavold, Z.M.; Thomas, W.; Todd, R.S.; Whittaker, M.

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Antitrypanosomal activities and cytotoxicity of 5-nitro-2-furancarbohydrazides
pp. 3601-3604(4)
Authors: Millet, R.; Maes, L.; Landry, V.; Sergheraert, C.; Davioud-Charvet, E.

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Synthesis, radiolabeling and preliminary biological evaluation of radiolabeled 5-methyl-6-nitroquipazine, a potential radioligand for the serotonin transporter
pp. 3611-3613(3)
Authors: Sandell, J.; Yu, M.; Emond, P.; Garreau, L.; Chalon, S.; Nagren, K.; Guilloteau, D.; Halldin, C.

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Silanediol-Based inhibitor of thermolysin
pp. 3625-3627(3)
Authors: Kim, J.; Glekas, A.; Sieburth, S.M.

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Inhibition of amine oxidases activity by 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives
pp. 3629-3633(5)
Authors: Manna, F.; Chimenti, F.; Bolasco, A.; Secci, D.; Bizzarri, B.; Befani, O.; Turini, P.; Mondov, B.; Alcaro, S.; Tafi, A.

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Characterization of mono- and diaminopyrimidine derivatives as novel, nonpeptide gonadotropin releasing hormone (GnRH) receptor antagonists
pp. 3635-3639(5)
Authors: Luthin, D.R.; Hong, Y.; Tompkins, E.; Anderes, K.L.; Paderes, G.; Kraynov, E.A.; Castro, M.A.; Nared-Hood, K.D.; Castillo, R.; Gregory, M.; Vazir, H.; May, J.M.; Anderson, M.B.

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Unique hole-Trapping property of the degenerate base,2-amino-7-deazaadenine
pp. 3641-3643(3)
Authors: Okamoto, A.; Tanaka, K.; Saito, I.

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Erratum to ''Tryptophanyl phosphoramidates as prodrugs of synadenol and its E-isomer: synthesis and biological activity'' [Bioorg. Med. Chem. Lett. 12 (2002) 2467]
pp. 3645-3645(1)
Authors: Wang, R.; Corbett, T.H.; Cheng, Y.; Drach, J.C.; Kern, E.R.; Mitsuya, H.; Zemlicka, J.

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