Publisher: Elsevier

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Volume 12, Number 23, 2 December 2002

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Inside (Editorial Board
pp. CO2-CO2(1)

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Contents List
pp. iii

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Graphical Abstracts
pp. 3351-3358(8)

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Design and synthesis of ethyl pyrrolidine-5,5-trans-lactams as inhibitors of hepatitis C virus NS3/4A protease
pp. 3359-3362(4)
Authors: Slater, M.J.; Andrews, D.M.; Baker, G.; Bethell, S.S.; Carey, S.; Chaignot, H.; Clarke, B.; Coomber, B.; Ellis, M.; Good, A.; Gray, N.; Hardy, G.; Jones, P.; Mills, G.; Robinson, E.

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Chemical modification of reveromycin A and its biological activities
pp. 3363-3366(4)
Authors: Shimizu, T.; Usui, T.; Machida, K.; Furuya, K.; Osada, H.; Nakata, T.

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Novel 2,5-dideoxystreptamine derivatives targeting the ribosomal decoding site RNA
pp. 3367-3372(6)
Authors: Vourloumis, D.; Takahashi, M.; Winters, G.C.; Simonsen, K.B.; Ayida, B.K.; Barluenga, S.; Qamar, S.; Shandrick, S.; Zhao, Q.; Hermann, T.

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A glucose-selective fluorescence sensor based on boronicacid-diol recognition
pp. 3373-3377(5)
Authors: Karnati, V.V.R.; Gao, X.; Gao, S.; Yang, W.; Ni, W.; Sankar, S.; Wang, B.

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Structure-activity relationships for a series of thiobenzamide influenza fusion inhibitors derived from 1,3,3-Trimethyl-5-hydroxy-cyclohexylmethylamine
pp. 3379-3382(4)
Authors: Yu, K.; Torri, A.F.; Luo, G.; Cianci, C.; Grant-Young, K.; Danetz, S.; Tiley, L.; Krystal, M.; Meanwell, N.A.

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Pyrrolidine and piperidine analogues of SC-57461A as potent, orally active inhibitors of leukotriene A4 hydrolase
pp. 3383-3386(4)
Authors: Penning, T.D.; Chandrakumar, N.S.; Desai, B.N.; Djuric, S.W.; Gasiecki, A.F.; Liang, C.; Miyashiro, J.M.; Russell, M.A.; Askonas, L.J.; Gierse, J.K.; Harding, E.I.; Highkin, M.K.; Kachur, J.F.; Kim, S.H.; Villani-Price, D.; Pyla, E.Y.; Ghoreishi-Haack, N.S.; Smith, W.G.

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Natural PTP1B Inhibitors from broussonetia papyrifera
pp. 3387-3390(4)
Authors: Chen, R.M.; Hu, L.H.; An, T.Y.; Li, J.; Shen, Q.

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in vitro inhibition of the measles virus by novel ring-expanded ('fat') nucleoside analogues containing the imidazo[4,5-e]diazepine ring system
pp. 3391-3394(4)
Authors: Zhang, N.; Chen, H.; Sood, R.; Kalicharran, K.; Fattom, A.I.; Naso, R.B.; Barnard, D.L.; Sidwell, R.W.; Hosmane, R.S.

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Design and synthesis of a -amino phosphotyrosyl mimetic suitably protected for peptide synthesis
pp. 3399-3401(3)
Authors: Lee, K.; Zhang, M.; Yang, D.; Burke, T.R.

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Core-modified sordaricin derivatives: Synthesis and antifungal activity
pp. 3403-3405(3)
Authors: Regueiro-Ren, A.; Carroll, T.M.; Chen, Y.; Matson, J.A.; Huang, S.; Mazzucco, C.E.; Stickle, T.M.; Vyas, D.M.; Balasubramanian, B.N.

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Design and synthesis of 6-substituted amino-4-oxa-1-azabicyclo[3,2,0]heptan-7-one derivatives as cysteine proteases inhibitors
pp. 3413-3415(3)
Authors: Zhou, N.E.; Guo, D.; Kaleta, J.; Purisima, E.; Menard, R.; Micetich, R.G.; Singh, R.

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6-Acylamino-penam derivatives: synthesis and inhibition of cathepsins B, L, K, and S
pp. 3417-3419(3)
Authors: Zhou, N.E.; Kaleta, J.; Purisima, E.; Menard, R.; Micetich, R.G.; Singh, R.

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Integration of optimized substituent patterns to produce highly potent 4-aryl-pyridine glucagon receptor antagonists
pp. 3421-3424(4)
Authors: Ladouceur, G.H.; Cook, J.H.; Hertzog, D.L.; Jones, J.H.; Hundertmark, T.; Korpusik, M.; Lease, T.G.; Livingston, J.N.; MacDougall, M.L.; Osterhout, M.H.; Phelan, K.; Romero, R.H.; Schoen, W.R.; Shao, C.; Smith, R.A.

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Design, synthesis, and neuraminidase inhibitory activity of GS-4071 analogues that utilize a novel hydrophobic paradigm
pp. 3425-3429(5)
Authors: Hanessian, S.; Wang, J.; Montgomery, D.; Stoll, V.; Stewart, K.D.; Kati, W.; Maring, C.; Kempf, D.; Hutchins, C.; Laver, W.G.

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Novel spirocyclic pyrrolidones as P2/P1 mimetics in potent inhibitors of HIV-1 protease
pp. 3431-3433(3)
Authors: Kazmierski, W.M.; Furfine, E.; Spaltenstein, A.; Wright, L.L.

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Trifluoromethyl ketones as inhibitors of histone deacetylase
pp. 3443-3447(5)
Authors: Frey, R.R.; Wada, C.K.; Garland, R.B.; Curtin, M.L.; Michaelides, M.R.; Li, J.; Pease, L.J.; Glaser, K.B.; Marcotte, P.A.; Bouska, J.J.; Murphy, S.S.; Davidsen, S.K.

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α1-Adrenoceptor activation: A comparison of 4-(Anilinomethyl)imidazoles and 4-(Phenoxymethyl)imidazoles to related 2-imidazolines
pp. 3449-3452(4)
Authors: Hodson, S.J.; Bigham, E.C.; Garrison, D.T.; Gobel, M.J.; Irving, P.E.; Liacos, J.A.; Navas, I.; Saussy, D.L.; Sherman, B.W.; Speake, J.D.; Bishop, M.J.

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Six-membered cyclic ureas as HIV-1 protease inhibitors: A QSAR study based on CODESSA PRO approach
pp. 3453-3457(5)
Authors: Katritzky, A.R.; Oliferenko, A.; Lomaka, A.; Karelson, M.

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Inhibitors of NF-B signaling: design and synthesis of a biotinylated isopanepoxydone affinity reagent
pp. 3463-3466(4)
Authors: Shotwell, J.B.; Koh, B.; Choi, H.W.; Wood, J.L.; Crews, C.M.

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The discovery of novel small molecule non-peptide gonadotropin releasing hormone (GnRH) receptor antagonists
pp. 3467-3470(4)
Authors: Luthin, D.R.; Hong, Y.; Pathak, V.P.; Paderes, G.; Nared-Hood, K.D.; Castro, M.A.; Vazir, H.; Li, H.; Tompkins, E.; Christie, L.; May, J.M.; Anderson, M.B.

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Synthesis and in vitro antiprotozoal activity of 5-nitrothiophene-2-carboxaldehyde thiosemicarbazone derivatives
pp. 3475-3478(4)
Authors: Bharti, N.; Husain, K.; Gonzalez Garza, M.T.; Cruz-Vega, D.E.; Castro-Garza, J.; Mata-Cardenas, B.D.; Naqvi, F.; Azam, A.

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Enhancement of pharmacokinetic properties and in vivo efficacy of benzylidene ketal M2 muscarinic receptor antagonists via benzamide modification
pp. 3479-3482(4)
Authors: Boyle, C.D.; Vice, S.F.; Campion, J.; Chackalamannil, S.; Lankin, C.M.; McCombie, S.W.; Billard, W.; Binch, I.; Crosby, G.; Williams, M.; Coffin, V.L.; Cox, K.A.; Grotz, D.E.; Duffy, R.A.; Ruperto, V.; Lachowicz, J.E.

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Non-peptide αv3 antagonists. Part 5: identification of potent RGD mimetics incorporating 2-aryl -amino acids as aspartic acid replacements
pp. 3483-3486(4)
Authors: Brashear, K.M.; Hunt, C.A.; Kucer, B.T.; Duggan, M.E.; Hartman, G.D.; Rodan, G.A.; Rodan, S.B.; Leu, C.; Prueksaritanont, T.; Fernandez-Metzler, C.; Barrish, A.; Homnick, C.F.; Hutchinson, J.H.; Coleman, P.J.

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New progesterone receptor antagonists: 3,3-disubstituted-5-aryloxindoles
pp. 3487-3490(4)
Authors: Fensome, A.; Bender, R.; Cohen, J.; Collins, M.A.; Mackner, V.A.; Miller, L.L.; Ullrich, J.W.; Winneker, R.; Wrobel, J.; Zhang, P.; Zhang, Z.; Zhu, Y.

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A novel synthesis of 7-aryl-8-fluoro-pyrrolo[1,2-a]pyrimid-4-ones as potent, stable GnRH receptor antagonists
pp. 3491-3495(5)
Authors: Tucci, F.C.; Zhu, Y.; Guo, Z.; Gross, T.D.; Connors, P.J.; Struthers, R.S.; Reinhart, G.J.; Wang, X.; Saunders, J.; Chen, C.

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