Publisher: Elsevier

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Volume 12, Number 18, 16 September 2002

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Contents List
pp. ii

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Graphical Abstracts
pp. 2491-2499(9)

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Peptide inhibitors of CDK2-cyclin A that target the cyclin recruitment-Site: structural variants of the C-Terminal Phe
pp. 2501-2505(5)
Authors: Atkinson, G.E.; Cowan, A.; McInnes, C.; Zheleva, D.I.; Fischer, P.M.; Chan, W.C.

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Synthesis of tag introducible (3-Trifluoromethyl)phenyldiazirine based photoreactive phenylalanine
pp. 2507-2510(4)
Authors: Hashimoto, M.; Hatanaka, Y.; Sadakane, Y.; Nabeta, K.

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Synthesis and antiaggregant properties of Stabilized analogues of polyunsaturated fatty acid metabolites
pp. 2511-2514(4)
Authors: Hachem, A.; Roussel, P.; Menager, E.; Gree, D.; Le Floc'h, Y.; Gree, R.; Cerletti, C.; Rolland, Y.; Simonet, S.; Verbeuren, T.

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Spirocyclic NK1 antagonists I: [4.5] and [5.5]-Spiroketals
pp. 2515-2518(4)
Authors: Seward, E.M.; Carlson, E.; Harrison, T.; Haworth, K.E.; Herbert, R.; Kelleher, F.J.; Kurtz, M.M.; Moseley, J.; Owen, S.N.; Owens, A.P.; Sadowski, S.J.; Swain, C.J.; Williams, B.J.

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Parallel solution- and solid-Phase synthesis of spirohydantoin derivatives as neurokinin-1 receptor ligands
pp. 2519-2522(4)
Authors: Bleicher, K.H.; Wuthrich, Y.; de Boni, M.; Kolczewski, S.; Hoffmann, T.; Sleight, A.J.

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Perylene diimides with different side chains are selective in inducing different G-Quadruplex DNA structures and in inhibiting telomerase
pp. 2527-2533(7)
Authors: Rossetti, L.; Franceschin, M.; Bianco, A.; Ortaggi, G.; Savino, M.

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A new series of M3 muscarinic antagonists based on the 4-amino-piperidine scaffold
pp. 2535-2539(5)
Authors: Diouf, O.; Gadeau, S.; Chelle, F.; Gelbcke, M.; Talaga, P.; Christophe, B.; Gillard, M.; Massingham, R.; Guyaux, M.

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New N-Alkyl-1,2-dihydro-2-thioxo-3-pyridinecarbothioamides as antituberculous agents with improved pharmacokinetics
pp. 2541-2544(4)
Authors: Ubiali, D.; Pagani, G.; Pregnolato, M.; Piersimoni, C.; Pedraz Munoz, J.L.; Rodrguez Gascon, A.; Terreni, M.

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Novel phenolic antioxidants as multifunctional inhibitors of inducible VCAM-1 expression for use in atherosclerosis
pp. 2545-2548(4)
Authors: Meng, C.Q.; Somers, P.K.; Rachita, C.L.; Holt, L.A.; Hoong, L.K.; Zheng, X.S.; Simpson, J.E.; Hill, R.R.; Olliff, L.K.; Kunsch, C.A.; Sundell, C.L.; Parthasarathy, S.; Saxena, U.; Sikorski, J.A.; Wasserman, M.A.

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Tetrahydrothienopyridylbutyl-tetrahydrobenzindoles: New Selective Ligands of the 5-HT7 Receptor
pp. 2549-2552(4)
Authors: Kikuchi, C.; Hiranuma, T.; Koyama, M.

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Glutathione-like tripeptides as inhibitors of glutathionylspermidine synthetase. Part 1: Substitution of the glycine carboxylic acid group
pp. 2553-2556(4)
Authors: Amssoms, K.; Oza, S.L.; Ravaschino, E.; Yamani, A.; Lambeir, A.; Rajan, P.; Bal, G.; Rodriguez, J.B.; Fairlamb, A.H.; Augustyns, K.; Haemers, A.

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Silica-Based Artificial Protease Exploiting Aldehyde Groups as Catalytic Elements
pp. 2557-2560(4)
Authors: Kim, H.; Paik, H.; Kim, M.; Chung, Y.; Suh, J.

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Dihydroquinolines as Novel n-NOS Inhibitors
pp. 2561-2564(4)
Authors: Jaroch, S.; Holscher, P.; Rehwinkel, H.; Sulzle, D.; Burton, G.; Hillmann, M.; McDonald, F.M.

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Quaternary Salts of E2020 Analogues as Acetylcholinesterase Inhibitors for the Reversal of Neuromuscular Block
pp. 2565-2568(4)
Authors: Clark, J.K.; Cowley, P.; Muir, A.W.; Palin, R.; Pow, E.; Prosser, A.B.; Taylor, R.; Zhang, M.

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Novel Piperidinium and Pyridinium Agents as Water-Soluble Acetylcholinesterase Inhibitors for the Reversal of Neuromuscular Blockade
pp. 2569-2572(4)
Authors: Palin, R.; Clark, J.K.; Cowley, P.; Muir, A.W.; Pow, E.; Prosser, A.B.; Taylor, R.; Zhang, M.

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Structure-Activity Relationship Studies of Ethyl 2-[(3-Methyl-2,5-dioxo(3-pyrrolinyl))amino]-4-(trifluoromethyl)pyrimidine-5- carboxylate: An Inhibitor of AP-1 and NF-B Mediated Gene Expression
pp. 2573-2577(5)
Authors: Palanki, M.S.S.; Gayo-Fung, L.M.; Shevlin, G.I.; Erdman, P.; Sato, M.; Goldman, M.; Ransone, L.J.; Spooner, C.

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Comparison of the Prevention of Aflatoxin B1-Induced Genotoxicity by Quercetin and Quercetin Pentaacetate
pp. 2579-2582(4)
Authors: Kohli, E.; Raj, H.G.; Kumari, R.; Rohil, V.; Kaushik, N.K.; Prasad, A.K.; Parmar, V.S.

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Structure-Activity Relationship of Biaryl Acylsulfonamide Analogues on the Human EP3 Prostanoid Receptor
pp. 2583-2586(4)
Authors: Gallant, M.; Carriere, M.C.; Chateauneuf, A.; Denis, D.; Gareau, Y.; Godbout, C.; Greig, G.; Juteau, H.; Lachance, N.; Lacombe, P.; Lamontagne, S.; Metters, K.M.; Rochette, C.; Ruel, R.; Slipetz, D.; Sawyer, N.; Tremblay, N.; Labelle, M.

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8-Aryl xanthines potent inhibitors of phosphodiesterase 5
pp. 2587-2590(4)
Authors: Arnold, R.; Beer, D.; Bhalay, G.; Baettig, U.; Collingwood, S.P.; Craig, S.; Devereux, N.; Dunstan, A.; Glen, A.; Gomez, S.; Haberthuer, S.; Howe, T.; Jelfs, S.; Moser, H.; Naef, R.; Nicklin, P.; Sandham, D.; Stringer, R.; Turner, K.; Watson, S.; Zurini, M.

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DNA Binding Ligands with Excellent Antibiotic Potency Against Drug-Resistant Gram-Positive Bacteria
pp. 2591-2594(4)
Authors: Burli, R.W.; Ge, Y.; White, S.; Baird, E.E.; Touami, S.M.; Taylor, M.; Kaizerman, J.A.; Moser, H.E.

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Parallel Synthesis and Anti-Malarial Activity of a Sulfonamide Library
pp. 2595-2598(4)
Authors: Ryckebusch, A.; Deprez-Poulain, R.; Debreu-Fontaine, M.; Vandaele, R.; Mouray, E.; Grellier, P.; Sergheraert, C.

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Synthesis and Evaluation of 4-Hydroxyphenylacetic Acid Amides and 4-Hydroxycinnamamides as Antioxidants
pp. 2599-2602(4)
Authors: Jung, Y.; Kang, T.; Yoon, J.; Joe, B.; Lim, H.; Seong, C.; Park, W.; Kong, J.; Cho, J.; Park N.-S.

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The discovery of SB-435495 - A potent, orally active inhibitor of lipoprotein-Associated phospholipase A2 for evaluation in man
pp. 2603-2606(4)
Authors: Blackie, J.A.; Bloomer, J.C.; Brown, M.J.B.; Cheng, H.; Elliott, R.L.; Hammond, B.; Hickey, D.M.B.; Ife, R.J.; Leach, C.A.; Lewis, V.A.; Macphee, C.H.; Milliner, K.J.; Moores, K.E.; Pinto, I.L.; Smith, S.A.; Stansfield, I.G.; Stanway, S.J.; Taylor, M.A.; Theobald, C.J.; Whittaker, C.M.

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Synthesis and Characterization of a New RXR Agonist Based on the 6-tert-Butyl-1,1-dimethylindanyl Structure
pp. 2607-2609(3)
Authors: Domnguez, B.; Jesus Vega, M.; Sussman, F.; de Lera, A.R.

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Synthesis and Cytotoxic Activity of pyridazino[1',6':1,2]pyrido[3,4-b]indol-5-inium derivatives as anti-cancer agents
pp. 2611-2614(4)
Authors: Fontana, A.; Benito, E.J.; Martn, M.J.; Sanchez, N.; Alajarn, R.; Vaquero, J.J.; Alvarez-Builla, J.; Lambel-Giraudet, S.; Leonce, S.; Pierre, A.; Caignard, D.

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4-Aminoquinolines as a novel class of NR1/2B subtype selective NMDA receptor antagonists
pp. 2615-2619(5)
Authors: Pinard, E.; Alanine, A.; Bourson, A.; Buttelmann, B.; Heitz, M.; Mutel; Trube, G.; Wyler, R.

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Long-Chain Aminoalcohol and Diamine Derivatives Induce Apoptosis through a Caspase-3 Dependent Pathway
pp. 2621-2626(6)
Authors: del Olmo, E.; Macho, A.; Alves, M.; Lopez, J.L.; el Banoua, F.; Munoz, E.; San Feliciano, A.

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Design, synthesis and biological evaluation of cyclic angiotensin II analogues with 3,5 side-Chain bridges - Role of C-Terminal aromatic residue and ring cluster for activity and implications in the drug design of AT1 non-peptide antagonists
pp. 2627-2633(7)
Authors: Roumelioti, P.; Polevaya, L.; Zoumpoulakis, P.; Giatas, N.; Mutule, I.; Keivish, T.; Zoga, A.; Vlahakos, D.; Iliodromitis, E.; Kremastinos, D.; Grdadolnik, S.G.; Mavromoustakos, T.; Matsoukas, J.

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Syntheses of Polycationic Dendrimers on Lipophilic Peptide Core for Complexation and Transport of Oligonucleotides
pp. 2635-2637(3)
Authors: Wimmer, N.; Marano, R.J.; Kearns, P.S.; Rakoczy, E.P.; Toth, I.

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The Synthesis of Substituted Fluorenes as Novel Non-Imidazole Histamine H3 Inhibitors
pp. 2643-2646(4)
Authors: Ting, P.C.; Lee, J.F.; Albanese, M.M.; Tom, W.C.; Solomon, D.M.; Aslanian, R.; Shih, N.; West, R.

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Synthesis and DNA binding properties of saturated distamycin analogues
pp. 2647-2650(4)
Authors: Woods, C.R.; Faucher, N.; Eschgfaller, B.; Bair, K.W.; Boger, D.L.

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