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Publisher: Elsevier

Volume 12, Number 12, 17 June 2002

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Graphical Abstracts
pp. xi-xix(9)

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The use of dioxygen by HIF prolyl hydroxylase (PHD1)
pp. 1547-1550(4)
Authors: McNeill, L.A.; Hewitson, K.S.; Gleadle, J.M.; Horsfall, L.E.; Oldham, N.J.; Maxwell, P.H.; Pugh, C.W.; Ratcliffe, P.J.; Schofield, C.J.

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Synthesis and pharmacological characterization of a potent, orally active p38 kinase inhibitor
pp. 1559-1562(4)
Authors: Dumas, J.; Hatoum-Mokdad, H.; Sibley, R.N.; Smith, R.A.; Scott, W.J.; Khire, U.; Lee, W.; Wood, J.; Wolanin, D.; Cooley, J.; Bankston, D.; Redman, A.M.; Schoenleber, R.; Caringal, Y.; Gunn, D.; Romero, R.; Osterhout, M.; Paulsen, H.; Housley, T.J.; Wilhelm, S.M.; Pirro, J.; Chien, D.; Ranges, G.E.; Shrikhande, A.; Muzsi, A.; Bortolon, E.; Wakefield, J.; Gianpaolo Ostravage, C.; Bhargava, A.; Chau, T.

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2-Aminothiazoles: A new class of agonist allosteric enhancers of A1 adenosine receptors
pp. 1563-1566(4)
Authors: Chordia, M.D.; Murphree, L.J.; Macdonald, T.L.; Linden, J.; Olsson, R.A.

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Synthesis and biological activity of polygalloyl-dendrimers as stable tannic acid mimics
pp. 1567-1570(4)
Authors: Halkes, S.B.A.; Vrasidas, I.; Rooijer, G.R.; van den Berg, A.J.J.; Liskamp, R.M.J.; Pieters, R.J.

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Solid-phase synthesis of thrombin inhibitors
pp. 1571-1573(3)
Authors: Lange, U.E.W.; Zechel, C.

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Pyridazines. Part 28: 5-alkylidene-6-phenyl-3(2H)-pyridazinones, a new family of platelet aggregation inhibitors
pp. 1575-1577(3)
Authors: Sotelo, E.; Fraiz, N.; Yanez, M.; Laguna, R.; Cano, E.; Brea, J.; Ravina, E.

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Inhibition of glutathione S-transferase in rat hepatocytes by a glycine-tetrazole modified S-alkyl-GSH analogue
pp. 1579-1582(4)
Authors: Burg, D.; Hameetman, L.; Filippov, D.V.; van der Marel, G.A.; Mulder, G.J.

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Synthesis and preliminary biochemical assessment of ethyl-terminated perfluoroalkylamine oxide surfactants
pp. 1587-1590(4)
Authors: Chaudier, Y.; Zito, F.; Barthelemy, P.; Stroebel, D.; Ameduri, B.; Popot, J.; Pucci, B.

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Discovery and evaluation of N-(triazin-1,3,5-yl) phenylalanine derivatives as VLA-4 integrin antagonists
pp. 1591-1594(4)
Authors: Porter, J.R.; Archibald, S.C.; Brown, J.A.; Childs, K.; Critchley, D.; Head, J.C.; Hutchinson, B.; Parton, T.A.H.; Robinson, M.K.; Shock, A.; Warrellow, G.J.; Zomaya, A.

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N-(Pyrimidin-4-yl) and N-(Pyridin-2-yl) phenylalanine derivatives as VLA-4 integrin antagonists
pp. 1595-1598(4)
Authors: Porter, J.R.; Archibald, S.C.; Brown, J.A.; Childs, K.; Critchley, D.; Head, J.C.; Hutchinson, B.; Parton, T.A.H.; Robinson, M.K.; Shock, A.; Warrellow, G.J.; Zomaya, A.

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Development of tripeptidyl farnesyltransferase inhibitors
pp. 1599-1602(4)
Authors: Lee H.-Y.; Sohn, J.; Kwon, B.

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Exploration of peptidyl hydrazones as water-soluble calpain inhibitors
pp. 1603-1606(4)
Authors: Nakamura, M.; Inoue, J.

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8-Methoxyquinoline-5-carboxamides as PDE4 inhibitors: a potential treatment for asthma
pp. 1613-1615(3)
Authors: Buckley, G.M.; Cooper, N.; Dyke, H.J.; Galleway, F.P.; Gowers, L.; Haughan, A.F.; Kendall, H.J.; Lowe, C.; Maxey, R.; Montana, J.G.; Naylor, R.; Oxford, J.; Peake, J.C.; Picken, C.L.; Runcie, K.A.; Sabin, V.; Sharpe, A.; Warneck, J.B.H.

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8-Methoxyquinolines as PDE4 inhibitors
pp. 1617-1619(3)
Authors: Billah, M.; Buckley, G.M.; Cooper, N.; Dyke, H.J.; Egan, R.; Ganguly, A.; Gowers, L.; Haughan, A.F.; Kendall, H.J.; Lowe, C.; Minnicozzi, M.; Montana, J.G.; Oxford, J.; Peake, J.C.; Picken, C.L.; Piwinski, J.J.; Naylor, R.; Sabin, V.; Shih, N.; Warneck, J.B.H.

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Synthesis and profile of SCH351591, a novel PDE4 inhibitor
pp. 1621-1623(3)
Authors: Billah, M.; Cooper, N.; Cuss, F.; Davenport, R.J.; Dyke, H.J.; Egan, R.; Ganguly, A.; Gowers, L.; Hannah, D.R.; Haughan, A.F.; Kendall, H.J.; Lowe, C.; Minnicozzi, M.; Montana, J.G.; Naylor, R.; Oxford, J.; Peake, J.C.; Piwinski, J.J.; Runcie, K.A.; Sabin, V.; Sharpe, A.; Shih, N.; Warneck, J.B.H.

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Syntheses of depsipeptide analogues of the insect neuropeptide proctolin
pp. 1625-1628(4)
Authors: Scherkenbeck, J.; Plant, A.; Stieber, F.; Losel, P.; Dyker, H.

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Vitamin D3: synthesis of seco C-9,11,21-trisnor-17-methyl-1α, 25-dihydroxyvitamin D3 analogues
pp. 1629-1632(4)
Authors: Wu, Y.; Sabbe, K.; de Clercq, P.; Vandewalle, M.; Bouillon, R.; Verstuyf, A.

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Vitamin D3: synthesis of seco-C-9,11-bisnor-17-methyl-1α,25-dihydroxyvitamin D3 analogues
pp. 1633-1636(4)
Authors: Wu, Y.; de Clercq, P.; Vandewalle, M.; Bouillon, R.; Verstuyf, A.

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Preparation, characterization, molecular modeling and In vitro activity of paclitaxel-cyclodextrin complexes
pp. 1637-1641(5)
Authors: Alcaro, S.; Ventura, C.A.; Paolino, D.; Battaglia, D.; Ortuso, F.; Cattel, L.; Puglisi, G.; Fresta, M.

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Design, synthesis and biological activity of novel non-amidine factor Xa inhibitors. Part 1: P1 structure-activity relationships of the substituted 1-(2-Naphthyl)-1H-pyrazole-5-carboxylamides
pp. 1651-1655(5)
Authors: Jia, Z.J.; Wu, Y.; Huang, W.; Goldman, E.; Zhang, P.; Woolfrey, J.; Wong, P.; Huang, B.; Sinha, U.; Park, G.; Reed, A.; Scarborough, R.M.; Zhu B.-Y.

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Design, synthesis, and SAR of monobenzamidines and aminoisoquinolines as factor Xa inhibitors
pp. 1657-1661(5)
Authors: Zhang, P.; Zuckett, J.F.; Woolfrey, J.; Tran, K.; Huang, B.; Wong, P.; Sinha, U.; Park, G.; Reed, A.; Malinowski, J.; Hollenbach, S.; Scarborough, R.M.; Zhu B.-Y.

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Cephalosporin-derived inhibitors of -Lactamase. Part 4: The C3 substituent
pp. 1663-1666(4)
Authors: Buynak, J.D.; Vogeti, L.; Doppalapudi, V.R.; Solomon, G.M.; Chen, H.

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Optimization of the -Aminoester class of factor Xa inhibitors. part 1: P4 and side-Chain modifications for improved In vitro potency
pp. 1667-1670(4)
Authors: Czekaj, M.; Klein, S.I.; Guertin, K.R.; Gardner, C.J.; Zulli, A.L.; Pauls, H.W.; Spada, A.P.; Cheney, D.L.; Brown, K.D.; Colussi, D.J.; Chu, V.; Leadley, R.J.; Dunwiddie, C.T.

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Optimization of the -Aminoester class of factor Xa inhibitors. part 2: Identification of FXV673 as a potent and selective inhibitor with excellent In vivo anticoagulant activity
pp. 1671-1674(4)
Authors: Guertin, K.R.; Gardner, C.J.; Klein, S.I.; Zulli, A.L.; Czekaj, M.; Gong, Y.; Spada, A.P.; Cheney, D.L.; Maignan, S.; Guilloteau, J.; Brown, K.D.; Colussi, D.J.; Chu, V.; Heran, C.L.; Morgan, S.R.; Bentley, R.G.; Dunwiddie, C.T.; Leadley, R.J.; Pauls, H.W.

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Synthesis of novel furo, thieno, and benzazetoazepines and evaluation of their cytotoxicity
pp. 1675-1677(3)
Authors: Martnez, R.; Gustavo Avila Zarraga, J.; Duran, M.S.T.E.; Ramrez Apam, M.T.; Canas, R.

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Focused library approach for identification of new N-acylphenylalanines as VCAM/VLA-4 antagonists
pp. 1679-1682(4)
Authors: Chen, L.; Trilles, R.; Miklowski, D.; Huang, T.; Fry, D.; Campbell, R.; Rowan, K.; Schwinge, V.; Tilley, J.W.

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Pyrrolo[2,3-d]pyrimidines containing diverse N-7 substituents as potent inhibitors of Lck
pp. 1683-1686(4)
Authors: Calderwood, D.J.; Johnston, D.N.; Munschauer, R.; Rafferty, P.

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Pyrazolo[3,4-d]pyrimidines containing an extended 3-substituent as potent inhibitors of Lck - a selectivity insight
pp. 1687-1690(4)
Authors: Burchat, A.F.; Calderwood, D.J.; Friedman, M.M.; Hirst, G.C.; Li, B.; Rafferty, P.; Ritter, K.; Skinner, B.S.

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Development of a genetic selection for catalytic antibodies
pp. 1691-1694(4)
Authors: Gildersleeve, J.; Janes, J.; Ulrich, H.; Yang, P.; Barbas, C.; Schultz, P.G.

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CorrigendumCorrigendum to ''The discovery of acylated -Amino acids as potent and orally bioavailable VLA-4 antagonists''[Bioorg. Med. Chem. Lett. 12 (2002) 611]
pp. 1695-1695(1)
Authors: Lin, L.S.; Kopka, I.E.; Mumford, R.A.; Magriotis, P.A.; Lanza, J.; Durette, P.L.; Kamenecka, T.; Young, D.N.; de Laszlo, S.E.; McCauley, E.; van Riper, G.; Kidambi, U.; Egger, L.A.; Tong, X.; Lyons, K.; Vincent, S.; Stearns, R.; Colletti, A.; Teffera, Y.; Fenyk-Melody, J.; Schmidt, J.A.; MacCoss, M.; Hagmann, W.K.

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