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Volume 12, Number 6, 25 March 2002

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Graphical Abstracts
pp. xi-xx(10)

Parallel suspension polymerization for high-throughput resin synthesis
pp. 837-840(4)
Authors: Reger, T.S.; Janda, K.D.

Synthesis of iodinated 3-aryltropanes with selective binding to either the dopamine or serotonin transporters
pp. 845-847(3)
Authors: Davies, H.M.L.; Ren, P.; Kong, N.X.; Sexton, T.; Childers, S.R.

Antibacterial activity of G6-quaternary ammonium derivatives of a lipophilic vancomycin analogue
pp. 849-852(4)
Authors: Blizzard, T.A.; Kim, R.M.; Morgan; Chang, J.; Kohler, J.; Kilburn, R.; Chapman, K.; Hammond, M.L.

Synthesis and photochemical protein crosslinking studies of hydrophilic naphthalimides
pp. 853-856(4)
Authors: Zhang, J.; Woods, R.J.; Brown, P.B.; Lee, K.; Kane, R.R.

Synthesis and antibacterial activity of linezolid analogues
pp. 857-859(3)
Authors: Yu, D.Y.G.; Huiyuan, G.

Imidazo[5,1-f][1,2,4]triazin-4(3H)-ones, a new class of potent PDE 5 inhibitors
pp. 865-868(4)
Authors: Haning, H.; Niewohner, U.; Schenke, T.; Es-Sayed, M.; Schmidt, G.; Lampe, T.; Bischoff, E.

Synthesis, Characterization and Antiamoebic Activity of Benzimidazole Derivatives and Their Vanadium and Molybdenum Complexes
pp. 869-871(3)
Authors: Bharti, N.; Shailendra; Gonzalez Garza, M.T.; Cruz-Vega, D.E.; Castro-Garza, J.; Saleem, K.; Naqvi, F.; Maurya, M.R.; Azam, A.

Dermorphin and deltorphin heptapeptide analogues: replacement of Phe residue by Dmp greatly improves opioid receptor affinity and selectivity
pp. 879-881(3)
Authors: Ambo, A.; Murase, H.; Niizuma, H.; Ouchi, H.; Yamamoto, Y.; Sasaki, Y.

Tricyclic isoxazoles are novel inhibitors of the multidrug resistance protein (MRP1)
pp. 883-886(4)
Authors: Norman, B.H.; Gruber, J.M.; Hollinshead, S.P.; Wilson, J.W.; Starling, J.J.; Law, K.L.; Self, T.D.; Tabas, L.B.; Williams, D.C.; Paul, D.C.; Wagner, M.M.; Dantzig, A.H.

Chemical synthesis and calcium release activity of N1-ether strand substituted cADPR mimic
pp. 887-889(3)
Authors: Huang, L.; Zhao, Y.; Yuan, L.; Min, J.; Zhang L.-H.

Biphenyls as potential mimetics of protein α-helix
pp. 891-893(3)
Author: Jacoby, E.

Highly Potent Inhibitors of TNF-α Production. Part 1: Discovery of Chemical Leads
pp. 903-905(3)
Authors: Matsui, T.; Kondo, T.; Nishita, Y.; Itadani, S.; Nakatani, S.; Omawari, N.; Sakai, M.; Nakazawa, S.; Ogata, A.; Ohno, H.; Obata, T.; Nakai, H.; Toda, M.

Highly potent inhibitors of TNF-α production. Part 2: identification of drug candidates
pp. 907-910(4)
Authors: Matsui, T.; Kondo, T.; Nishita, Y.; Itadani, S.; Tsuruta, H.; Fujita, S.; Omawari, N.; Sakai, M.; Nakazawa, S.; Ogata, A.; Mori, H.; Ohno, H.; Obata, T.; Nakai, H.; Toda, M.

Hydrophobic modifications at 1-phosphate of inositol 1,4,5-Trisphosphate analogues enhance receptor binding
pp. 911-913(3)
Authors: Nakanishi, W.; Kikuchi, K.; Inoue, T.; Hirose, K.; Iino, M.; Nagano, T.

Structure-Activity Study of l-Cysteine-Based N-Type Calcium Channel Blockers: Optimization of N- and C-Terminal Substituents
pp. 915-918(4)
Authors: Seko, T.; Kato, M.; Kohno, H.; Ono, S.; Hashimura, K.; Takimizu, H.; Nakai, K.; Maegawa, H.; Katsube, N.; Toda, M.

Benzimidazoles and isosteric compounds as potent and selective factor Xa inhibitors
pp. 919-922(4)
Authors: He, W.; Hanney, B.; Myers, M.R.; Condon, S.; Becker, M.R.; Spada, A.P.; Burns, C.; Brown, K.; Colussi, D.; Chu, V.

Synthesis and evaluation of pseudopeptide analogues of a specific CXCR4 inhibitor, T140: The insertion of an (E)-alkene dipeptide isostere into the II'-turn moiety
pp. 923-928(6)
Authors: Tamamura, H.; Hiramatsu, K.; Miyamoto, K.; Omagari, A.; Oishi, S.; Nakashima, H.; Yamamoto, N.; Kuroda, Y.; Nakagawa, T.; Otaka, A.; Fujii, N.

Identification of a novel, orally bioavailable histamine H3 receptor antagonist based on the 4-benzyl-(1H-imidazol-4-yl) template
pp. 937-941(5)
Authors: Aslanian, R.; Mutahi, M.W.; Shih, N.; McCormick, K.D.; Piwinski, J.J.; Ting, P.C.; Albanese, M.M.; Berlin, M.Y.; Zhu, X.; Wong, S.; Rosenblum, S.B.; Jiang, Y.; West, R.; She, S.; Williams, S.M.; Bryant, M.; Hey, J.A.

Oxime derivatives of sordaricin as potent antifungal agents
pp. 943-946(4)
Authors: Serrano-Wu, M.H.; St. Laurent, D.R.; Mazzucco, C.E.; Stickle, T.M.; Barrett, J.F.; Vyas, D.M.; Balasubramanian, B.N.

Diaryl-dialkyl-substituted pyrazoles: regioselective synthesis and binding affinity for the estrogen receptor
pp. 947-950(4)
Authors: Nishiguchi, G.A.; Rodriguez, A.L.; Katzenellenbogen, J.A.

Design and synthesis of antiangiogenic/heparin-binding arginine dendrimer mimicking the surface of endostatin
pp. 951-954(4)
Authors: Kasai, S.; Nagasawa, H.; Shimamura, M.; Uto, Y.; Hori, H.

Soluble polymer-supported synthesis of benzodiazepinones
pp. 959-962(4)
Authors: Wu, C.; Sun C.-M.

Novel N-[1-(1-substituted 4-piperidinylmethyl)-4-piperidinyl]benzamides as potent colonic prokinetic agents
pp. 967-970(4)
Authors: Harada, H.; Yamazaki, H.; Toyotomi, Y.; Tateishi, H.; Mine, Y.; Yoshida, N.; Kato, S.

Design, synthesis and bioactivity evaluation of tribactam  lactamase inhibitors
pp. 971-975(5)
Authors: Copar, A.; Prevec, T.; Anzic, B.; Mesar, T.; Selic, L.; Vilar, M.; Solmajer, T.

Benzimidazole-4,7-diones as Inhibitors of Protozoal (Toxoplasma gondii) Purine Nucleoside Phosphorylase
pp. 977-979(3)
Authors: Alvarez, F.; Gherardi, A.; Nebois, P.; Sarciron, M.; Petavy, A.; Walchshofer, N.

Bivalent inhibition of -Tryptase: distance scan of neighboring subunits by dibasic inhibitors
pp. 985-988(4)
Authors: Schaschke, N.; Dominik, A.; Matschiner, G.; Sommerhoff, C.P.

Substrate spectrum of tyrocidine thioesterase probed with randomized peptide N-acetylcysteamine thioesters
pp. 989-992(4)
Authors: Xie, G.; Uttamchandani, M.; Chen, G.Y.J.; Bu, X.; Lin, S.S.; Wong, K.M.; Yan, W.; Yao, S.Q.; Guo, Z.

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