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Publisher: Elsevier

Volume 12, Number 2, 21 January 2002

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Graphical Abstracts
pp. xi-xx(10)

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Effects of the incorporation of IBTM -turn mimetics into the dipeptoid CCK1 receptor agonist PD 170292
pp. 109-112(4)
Authors: Martn-Martnez, M.; Latorre, M.; Garca-Lopez, M.T.; Cenarruzabeitia, E.; Del Ro, J.; Gonzalez-Muniz, R.

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Anti-MRSA activity of alkyl gallates
pp. 113-116(4)
Authors: Kubo, I.; Xiao, P.; Fujita, K.

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Antifungal sordarins. Synthesis and structure-activity relationships of 3'-O-Substituted derivatives
pp. 117-120(4)
Authors: Arribas, E.M.; Castro, J.; Clemens, I.R.; Cuevas, J.C.; Chicharro, J.; Fraile, M.T.; Garca-Ochoa, S.; Gomez de las Heras, F.; Ruiz, J.R.

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Antifungal sordarins. Synthesis and structure-activity relationships of 3',4'-Fused dioxolane and dioxane derivatives
pp. 121-124(4)
Authors: Bueno, J.M.; Cuevas, J.C.; Fiandor, J.M.; Garca-Ochoa, S.; Gomez de las Heras, F.

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The design and synthesis of a novel series of indole derived selective ETA antagonists
pp. 125-128(4)
Authors: Rawson, D.J.; Dack, K.N.; Dickinson, R.P.; James, K.

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Potent In vitro methicillin-resistant Staphylococcus aureus activity of 2-(1H-indol-3-yl)tetrahydroquinoline derivatives
pp. 129-132(4)
Authors: Hoemann, M.Z.; Xie, R.L.; Rossi, R.F.; Meyer, S.; Sidhu, A.; Cuny, G.D.; Hauske, J.R.

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Specific and dual antagonists of α41 and α47 integrins
pp. 133-136(4)
Authors: Lin, L.S.; Lanza, T.; McCauley, E.; Riper, G.V.; Kidambi, U.; Cao, J.; Egger, L.A.; Mumford, R.; Schmidt, J.A.; MacCoss, M.; Hagmann, W.K.

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N-Acyl-l-phenylalanine derivatives as potent VLA-4 antagonists that mimic a cyclic peptide conformation
pp. 137-140(4)
Authors: Chen, L.; Tilley, J.; Trilles, R.V.; Yun, W.; Fry, D.; Cook, C.; Rowan, K.; Schwinge, V.; Campbell, R.

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Synthesis and structure-activity relationships of oxime neurokinin antagonists: discovery of potent arylamides
pp. 141-145(5)
Authors: Shih N.-Y.; Albanese, M.; Anthes, J.C.; Carruthers?, N.I.; Grice?, C.A.; Lin, L.; Mangiaracina, P.; Reichard, G.A.; Schwerdt, J.; Seidl, V.; Wong, S.; Piwinski, J.J.

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Mixed lineage kinase activity of indolocarbazole analogues
pp. 147-150(4)
Authors: Murakata, C.; Kaneko, M.; Gessner, G.; Angeles, T.S.; Ator, M.A.; O'Kane, T.M.; McKenna, B.A.W.; Thomas, B.A.; Mathiasen, J.R.; Saporito, M.S.; Bozyczko-Coyne, D.; Hudkins, R.L.

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An N1-Hydrogen bonding model for flavin coenzyme
pp. 151-154(4)
Authors: Guo, F.; Chang, B.H.; Rizzo, C.J.

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Evaluation of isotryptamine derivatives at 5-HT2 serotonin receptors
pp. 155-158(4)
Authors: Chang-Fong, J.; Addo, J.; Dukat, M.; Smith, C.; Mitchell, N.A.; Herrick-Davis, K.; Teitler, M.; Glennon, R.A.

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The discovery of small molecule carbamates as potent dual α4147 integrin antagonists
pp. 159-163(5)
Authors: Chang, L.L.; Truong, Q.; Mumford, R.A.; Egger, L.A.; Kidambi, U.; Lyons, K.; McCauley, E.; van Riper, G.; Vincent, S.; Schmidt, J.A.; MacCoss, M.; Hagmann, W.K.

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Synthesis and biological activity of 8-substituted hydrocodone indole and hydromorphone indole derivatives
pp. 165-168(4)
Authors: Yu, H.; Prisinzano, T.; Dersch, C.M.; Marcus, J.; Rothman, R.B.; Jacobson, A.E.; Rice, K.C.

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Facile synthesis of -Cyclodextrin dithiols
pp. 169-170(2)
Authors: Yang, J.; Leung, D.K.

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Solid-Phase synthesis of new saphenamycin analogues with antimicrobial activity
pp. 171-175(5)
Authors: Laursen, J.B.; de Visser, P.C.; Nielsen, H.K.; Jensen, K.J.; Nielsen, J.

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An improved procedure for the synthesis of branched polyethylene glycols (PEGs) with the reporter dipeptide met-ala for protein conjugation
pp. 177-180(4)
Authors: Guiotto, A.; Pozzobon, M.; Sanavio, C.; Schiavon, O.; Orsolini, P.; Veronese, F.M.

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Selective urokinase-type plasminogen activator (uPA) inhibitors. Part 1: 2-Pyridinylguanidines
pp. 181-184(4)
Authors: Barber, C.G.; Dickinson, R.P.; Horne, V.A.

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Synthesis and pharmacology of isoquinuclidine derivatives as 5-HT3 ligands
pp. 189-192(4)
Authors: Iriepa, I.; Villasante, F.J.; Galvez, E.; Labeaga, L.; Innerarity, A.; Orjales, A.

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Oxyaniliniums as acetylcholinesterase inhibitors for the reversal of neuromuscular block
pp. 193-196(4)
Authors: Grove, S.J.A.; Kaur, J.; Muir, A.W.; Pow, E.; Tarver, G.J.; Zhang M.-Q.

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3-Aryl pyridone derivatives. Potent and selective kappa opioid receptor agonists
pp. 197-200(4)
Authors: Semple, G.; Andersson, B.; Chhajlani, V.; Georgsson, J.; Johansson, M.; Lindschoten, M.; Ponten, F.; Rosenquist; Sorensen, H.; Swanson, L.; Swanson, M.

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DNA cleavage by pentadentate iron(II) complexes containing fluoro-substituted phenyl groups
pp. 201-203(3)
Authors: Kurosaki, H.; Maruyama, A.; Koike, H.; Kuroda, N.; Ishikawa, Y.; Goto, M.

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Biphenyls as potent vitronectin receptor antagonists
pp. 205-208(4)
Authors: Urbahns, K.; Harter, M.; Albers, M.; Schmidt, D.; Stelte-Ludwig, B.; Bruggemeier, U.; Vaupel, A.; Gerdes, C.

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New series of aryloxypropanolamines with both human 3-adrenoceptor agonistic activity and free radical scavenging properties
pp. 209-212(4)
Authors: Aubriot, S.; Nicolle, E.; Lattier, M.; Morel, C.; Cao, W.; Daniel, K.W.; Collins, S.; Leclerc, G.; Faure, P.

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Synthesis of an immunoconjugate of camptothecin
pp. 217-219(3)
Authors: Walker, M.A.; Dubowchik, G.M.; Hofstead, S.J.; Trail, P.A.; Firestone, R.A.

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Structure-based design and protein X-ray analysis of a protein kinase inhibitor
pp. 221-224(4)
Authors: Furet, P.; Meyer, T.; Strauss, A.; Raccuglia, S.; Rondeau, J.

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N-Methylbenzanilide derivatives as a novel class of selective V1A receptor antagonists
pp. 229-232(4)
Authors: Kakefuda, A.; Tsukada, J.; Kusayama, T.; Tahara, A.; Tsukamoto, S.

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Polyhydroxylated azepanes as new motifs for DNA minor groove binding agents
pp. 237-241(5)
Authors: Johnson, H.A.; Thomas, N.R.

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Synthesis and structure-activity relationship of 2-(aminoalkyl)-2,3,3a,8-tetrahydrodibenzo[c,f]isoxazolo[2,3-a]azepine derivatives: a novel series of 5-HT2A/2C receptor antagonists. Part 1
pp. 243-248(6)
Authors: Andres, J.I.; Alcazar, J.; Alonso, J.M.; Daz, A.; Fernandez, J.; Gil, P.; Iturrino, L.; Matesanz, E.; Meert, T.F.; Megens, A.; Sipido, V.K.

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Synthesis and structure-Activity relationship of 2-(aminoalkyl)-2,3,3a,8-tetrahydrodibenzo[c,f]isoxazolo[2,3-a]azepine derivatives: a novel series of 5-HT2A/2C receptor antagonists. Part 2
pp. 249-253(5)
Authors: Ignacio Andres, J.; Alcazar, J.; Alonso, J.M.; Daz, A.; Fernandez, J.; Gil, P.; Iturrino, L.; Matesanz, E.; Meert, T.F.; Megens, A.; Sipido, V.K.

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Cyclic acid anhydrides as a new class of potent, selective and non-peptidic inhibitors of geranylgeranyl transferase
pp. 255-259(5)
Authors: Marson, C.M.; Rioja, A.S.; Brooke, G.; Coombes, R.C.; Vigushin, D.M.

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First dual NK1 antagonists-serotonin reuptake inhibitors: synthesis and SAR of a new class of potential antidepressants
pp. 261-264(4)
Authors: Ryckmans, T.; Balancon, L.; Berton, O.; Genicot, C.; Lamberty, Y.; Lallemand, B.; Pasau, P.; Pirlot, N.; Quere, L.; Talaga, P.

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Increase of the adenallene anti-HIV activity in cell culture using its bis(tBuSATE) phosphotriester derivative
pp. 265-266(2)
Authors: Egron, D.; Perigaud, C.; Gosselin, G.; Aubertin, A.; Gatanaga, H.; Mitsuya, H.; Zemlicka, J.; Imbach, J.

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