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Publisher: Elsevier

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Volume 11, Number 18, 17 September 2001

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G-Quadruplex DNA binding by a series of carbocyanine dyes
pp. 2411-2414(4)
Authors: Kerwin, S.M.; Sun, D.; Kern, J.T.; Rangan, A.; Thomas, P.W.

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Stereospecific synthesis of trans-arachidonic acids
pp. 2415-2418(4)
Authors: Krishna, U.M.; Reddy, M.M.; Xia, J.; Falck, J.R.; Balazy, M.

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Synthesis and biological evaluation of clitocine analogues as adenosine kinase inhibitors
pp. 2419-2422(4)
Authors: Lee C.-H.; Daanen, J.F.; Jiang, M.; Yu, H.; Kohlhaas, K.L.; Alexander, K.; Jarvis, M.F.; Kowaluk, E.L.; Bhagwat, S.S.

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Modulation of penicillin acylase properties via immobilization techniques: one-pot chemoenzymatic synthesis of cephamandole from cephalosporin C
pp. 2429-2432(4)
Authors: Terreni, M.; Pagani, G.; Ubiali, D.; Fernandez-Lafuente, R.; Mateo, C.; Guisan, J.M.

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Synthesis of glycosyl phosphoramidates: novel isosteric analogues of glycosyl phosphates
pp. 2433-2435(3)
Authors: Kannan, T.; Vinodhkumar, S.; Varghese, B.; Loganathan, D.

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Solid-phase, single nucleotide primer extension of DNA/RNA hybrids by reverse transcriptases
pp. 2437-2440(4)
Authors: Pirrung, M.C.; Worden, J.D.; Labriola, J.P.; Montague-Smith, M.P.; Weislo, L.J.

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New anti-malarial flavonol glycoside from hydrangeae dulcis folium
pp. 2445-2447(3)
Authors: Murakami, N.; Mostaqul, H.M.; Tamura, S.; Itagaki, S.; Horii, T.; Kobayashi, M.

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Identification of E2F-1/Cyclin A antagonists
pp. 2449-2452(4)
Authors: Sharma, S.K.; Ramsey, T.M.; Chen, Y.; Chen, W.; Martin, M.S.; Clune, K.; Sabio, M.; Bair, K.W.

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Incorporation of 2'-deoxy-5-(trifluoromethyl)uridine and 5-Cyano-2'-deoxyuridine into DNA
pp. 2453-2455(3)
Authors: Markley, J.C.; Chirakul, P.; Sologub, D.; Sigurdsson, S.T.

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Modulation of human mammary cell sensitivity to paclitaxel by new quinoline sulfonamides
pp. 2457-2460(4)
Authors: Chibale, K.; Ojima, I.; Haupt, H.; Geng, X.; Pera, P.; Bernacki, R.J.

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The discovery of novel, potent and selective PDE5 inhibitors
pp. 2461-2464(4)
Authors: Bi, Y.; Stoy, P.; Adam, L.; He, B.; Krupinski, J.; Normandin, D.; Pongrac, R.; Seliger, L.; Watson, A.; Macor, J.E.

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Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 3: A proposed pharmacophore model for 1-[N-(methyl)-N-(phenylsulfonyl)amino]-2-(phenyl)-4-[4-(substituted)piperidi n-1-yl]butanes
pp. 2469-2473(5)
Authors: Finke, P.E.; Meurer, L.C.; Oates, B.; Shah, S.K.; Loebach, J.L.; Mills, S.G.; MacCoss, M.; Castonguay, L.; Malkowitz, L.; Springer, M.S.; Gould, S.L.; deMartino, J.A.

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Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 4: synthesis and structure-Activity relationships for 1-[N-(Methyl)-N-(phenylsulfonyl)amino]-2-(phenyl)-4-(4-(N-(alkyl)-N-(benzylo xycarbonyl)amino)piperidin-1-yl)butanes
pp. 2475-2479(5)
Authors: Finke, P.E.; Oates, B.; Mills, S.G.; MacCoss, M.; Malkowitz, L.; Springer, M.S.; Gould, S.L.; deMartino, J.A.; Carella, A.; Carver, G.; Holmes, K.; Danzeisen, R.; Hazuda, D.; Kessler, J.; Lineberger, J.; Miller, M.; Schleif, W.A.; Emini, E.A.

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Selective, orally active MMP inhibitors with an aryl backbone
pp. 2481-2483(3)
Authors: Barta, T.E.; Becker, D.P.; Bedell, L.J.; de Crescenzo, G.A.; McDonald, J.J.; Mehta, P.; Munie, G.E.; Villamil, C.I.

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A selective inhibitor of Escherichia coli prephenate dehydratase
pp. 2485-2488(4)
Authors: Husain, A.; Chen, S.; Wilson, D.B.; Ganem, B.

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Derivatives of (2R,3R,4S)-2-Aminomethylpyrrolidine-3,4-diol are selective α-Mannosidase inhibitors
pp. 2489-2493(5)
Authors: Popowycz, F.; Gerber-Lemaire, S.; demange, R.; Rodriguez-Garca, E.; Asenjo, A.T.C.; Robina, I.; Vogel, P.

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Syntheses and preliminary pharmacological evaluation of the two epimers of the 5-F2t-isoprostane
pp. 2495-2498(4)
Authors: Durand, T.; Cracowski, J.; Guy, A.; Rossi, J.

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Inhibitors of Bacterial Tyrosyl tRNA Synthetase: Synthesis of Carbocyclic Analogues of the Natural Product SB-219383
pp. 2499-2502(4)
Authors: Jarvest, R.L.; Berge, J.M.; Houge-Frydrych, C.S.V.; Mensah, L.M.; O'Hanlon, P.J.; Pope, A.J.

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Chemo-Enzymatic synthesis of the galili epitope Galα(1->3)Gal(1->4)GlcNAc on a homogeneously soluble PEG polymer by a multi-Enzyme system
pp. 2503-2506(4)
Authors: Brinkmann, N.; Malissard, M.; Ramuz, M.; Romer, U.; Schumacher, T.; Berger, E.G.; Elling, L.; Wandrey, C.; Liese, A.

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Bicyclic anti-VZV nucleosides: Thieno analogues retain full antiviral activity
pp. 2507-2510(4)
Authors: Brancale, A.; McGuigan, C.; Algain, B.; Savy, P.; Benhida, R.; Fourrey, J.; Andrei, G.; Snoeck, R.; de Clercq, E.; Balzarini, J.

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Synthesis and evaluation of the sunflower derived trypsin inhibitor as a potent inhibitor of the type II transmembrane serine protease, matriptase
pp. 2515-2519(5)
Authors: Long, Y.; Lee, S.; Lin, C.; Enyedy, I.J.; Wang, S.; Li, P.; Dickson, R.B.; Roller, P.P.

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Furans with basic side chains: synthesis and biological evaluation of a novel series of antagonists with selectivity for the estrogen receptor alpha
pp. 2521-2524(4)
Authors: Mortensen, D.S.; Rodriguez, A.L.; Sun, J.; Katzenellenbogen, B.S.; Katzenellenbogen, J.A.

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Hydrophobicity, a physicochemical factor in the inhibition of the enzyme estrone sulfatase (ES)
pp. 2525-2528(4)
Authors: Ahmed, S.; James, K.; Owen, C.P.; Patel, C.K.; Patel, M.

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Synthesis and biological data of 4-amino-1-(2-chloro-2-phenylethyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid ethyl esters, a new series of A1-adenosine receptor (A1AR) ligands
pp. 2529-2531(3)
Authors: Schenone, S.; Bruno, O.; Fossa, P.; Ranise, A.; Menozzi, G.; Mosti, L.; Bondavalli, F.; Martini, C.; Trincavelli, L.

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Solid- and solution-Phase synthesis of highly-Substituted-Pyrrolidine libraries
pp. 2537-2540(4)
Authors: Steger, M.; Hubschwerlen?, C.; Schmid?, G.

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Studies on phytanoyl-CoA 2-hydroxylase and synthesis of phytanoyl-Coenzyme A
pp. 2545-2548(4)
Authors: Kershawa?, N.J.; Mukherji, M.; MacKinnon, C.H.; Claridge, T.D.W.; Odell, B.; Wierzbicki, A.S.; Lloyd, M.D.; Schofield, C.J.

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Substituted Imidazoles as Glucagon Receptor Antagonists
pp. 2549-2553(5)
Authors: Chang, L.L.; Sidler, K.L.; Cascieri, M.A.; de Laszlo, S.; Koch, G.; Li, B.; MacCoss, M.; Mantlo, N.; O'Keefe, S.; Pang, M.; Rolando, A.; Hagmann, W.K.

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New leads for selective inhibitors of α-l-fucosidases. Synthesis and glycosidase inhibitory activities of [(2R,3S,4R)-3,4-Dihydroxypyrrolidin-2-yl]furan derivatives
pp. 2555-2559(5)
Authors: Robina, I.; Moreno-Vargas, A.J.; Fernandez-Bolanos, J.G.; Fuentes, J.; demange, R.; Vogel, P.

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Glutamyl--boronate Inhibitors of Bacterial Glu-tRNAGln Amidotransferase
pp. 2561-2564(4)
Authors: decicco, C.P.; Nelson, D.J.; Luo, Y.; Shen, L.; Horiuchi, K.Y.; Amsler, K.M.; Foster, L.A.; Spitz, S.M.; Merrill, J.J.; Sizemore, C.F.; Rogers, K.C.; Copeland, R.A.; Harpel, M.R.

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