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Publisher: Elsevier

Volume 11, Number 16, 20 August 2001

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Graphical Abstracts
pp. xi-xx(10)

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Parallel solid-phase synthesis of nucleoside phosphoramidate libraries
pp. 2057-2060(4)
Authors: Jin, Y.; Chen, X.; Cote, M.; Roland, A.; Korba, B.; Mounir, S.; Iyer, R.P.

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1,4-Disubstituted imidazoles are potential antibacterial agents functioning as inhibitors of enoyl acyl carrier protein reductase (FabI)
pp. 2061-2065(5)
Authors: Heerding, D.A.; Chan, G.; deWolf, W.E.; Fosberry, A.P.; Janson, C.A.; Jaworski, D.D.; McManus, E.; Miller, W.H.; Moore, T.D.; Payne, D.J.; Qiu, X.; Rittenhouse, S.F.; Slater-Radosti, C.; Smith, W.; Takata, D.T.; Vaidya, K.S.; Yuan, C.C.K.; Huffman, W.F.

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Structure-Activity Study and Analgesic Efficacy of Amino Acid Derivatives as N-Type Calcium Channel Blockers
pp. 2067-2070(4)
Authors: Seko, T.; Kato, M.; Kohno, H.; Ono, S.; Hashimura, K.; Takimizu, H.; Nakai, K.; Maegawa, H.; Katsube, N.; Toda, M.

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Pyridopyrimidine analogues as novel adenosine kinase inhibitors
pp. 2071-2074(4)
Authors: Zheng, G.Z.; Lee, C.; Pratt, J.K.; Perner, R.J.; Jiang, M.Q.; Gomtsyan, A.; Matulenko, M.A.; Mao, Y.; Koenig, J.R.; Kim, K.H.; Muchmore, S.; Yu, H.; Kohlhaas, K.; Alexander, K.M.; McGaraughty, S.; Chu, K.L.; Wismer, C.T.; Mikusa, J.; Jarvis, M.F.; Marsh, K.; Kowaluk, E.A.; Bhagwat, S.S.; Stewart, A.O.

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Synthesis, antimalarial activity and inhibition of haem detoxification of novel bisquinolines
pp. 2075-2077(3)
Authors: Ayad, F.; Tilley, L.; deady, L.W.

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SAR Studies of Piperidine-Based Analogues of Cocaine. Part 3: Oxadiazoles
pp. 2079-2083(5)
Authors: Petukhov, P.A.; Zhang, M.; Johnson, K.J.; Tella, S.R.; Kozikowski, A.P.

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Amino acid derived sulfonamide hydroxamates as inhibitors of procollagen C-Proteinase: solid-Phase synthesis of ornithine analogues
pp. 2085-2088(4)
Authors: Dankwardt, S.M.; Martin, R.L.; Chan, C.S.; van Wart, H.E.; Walker, K.A.M.; delaet, N.G.; Robinson, L.A.

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Synthesis and potassium channel opening activity of substituted 10H-Benzo[4,5]furo[3,2-b]indole- and 5,10-Dihydro-indeno[1,2-b]indole-1-carboxylic acids
pp. 2093-2097(5)
Authors: Butera, J.A.; Antane, S.A.; Hirth, B.; Lennox, J.R.; Sheldon, J.H.; Norton, N.W.; Warga, D.; Argentieri, T.M.

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Enzymatic synthesis of aza-l-tyrosines
pp. 2099-2100(2)
Authors: Watkins, E.B.; Phillips, R.S.

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Biflavonoids as novel antituberculosis agents
pp. 2101-2104(4)
Authors: Lin Y.-M.; Flavin, M.T.; Cassidy, C.S.; Mar, A.; Chen, F.

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Thrombin receptor (PAR-1) antagonists. Solid-Phase synthesis of indole-Based peptide mimetics by anchoring to a secondary amide
pp. 2105-2109(5)
Authors: Zhang H.-C.; McComsey, D.F.; White, K.B.; Addo, M.F.; Andrade-Gordon, P.; derian, C.K.; Oksenberg, D.; Maryanoff, B.E.

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Stereoselective synthesis and antibacterial evaluation of 4-amido-isothiazolidinone oxides
pp. 2111-2115(5)
Authors: Chen, Z.; demuth, T.P.; Wireko, F.C.

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Novel Lipase-Catalysed Enantioselective Deacetylation of (+/-)-5-Acetoxy-3-(4-fluorophenyl)-2-phenylisoxazolidine
pp. 2117-2121(5)
Authors: Mukherjee, S.; Prasad, A.K.; Parmar, V.S.; Howarth, O.W.

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Leishmanicidal activity of some stilbenoids and related heterocyclic compounds
pp. 2123-2126(4)
Authors: del Olmo, E.; Armas, M.G.; Lopez-Perez, J.L.; Munoz, V.; deharo, E.; San Feliciano, A.

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Discovery of Thioazepinone Ligands for Src SH2: From Non-specific to Specific Binding
pp. 2127-2131(5)
Authors: Lesuisse, D.; deprez, P.; Albert, E.; Duc, T.T.; Sortais, B.; Gofflo, D.; Jean-Baptiste, V.; Marquette, J.; Schoot, B.; Sarubbi, E.; Lange, G.; Broto, P.; Mandine, E.

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5-HT3R Binding of lerisetron: an interdisciplinary approach to drug-Receptor interactions
pp. 2133-2136(4)
Authors: Parihar, H.S.; Suryanarayanan, A.; Ma, C.; Joshi, P.; Venkataraman, P.; Schulte, M.K.; Kirschbaum, K.S.

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Novel 3-(2-Adamantyl)pyrrolidines with potent activity against influenza A virus-identification of aminoadamantane derivatives bearing two pharmacophoric amine groups
pp. 2137-2142(6)
Authors: Stamatiou, G.; Kolocouris, A.; Kolocouris, N.; Fytas, G.; Foscolos, G.B.; Neyts, J.; de Clercq, E.

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Piperazine-Based CCR5 antagonists as HIV-1 inhibitors. I: 2(S)-methyl piperazine as a key pharmacophore element
pp. 2143-2146(4)
Authors: Tagat, J.R.; McCombie, S.W.; Steensma, R.W.; Lin, S.; Nazareno, D.V.; Baroudy, B.; vantuno, N.; Xu, S.; Liu, J.

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N-Hydroxyformamide peptidomimetics as TACE/Matrix metalloprotease inhibitors: oral activity via P1' isobutyl substitution
pp. 2147-2151(5)
Authors: Musso, D.L.; Andersen, M.W.; Andrews, R.C.; Austin, R.; Beaudet, E.J.; Becherer, J.D.; Bubacz, D.G.; Bickett, D.M.; Chan, J.H.; Conway, J.G.; Cowan, D.J.; Gaul, M.D.; Glennon, K.C.; Hedeen, K.M.; Lambert, M.H.; Leesnitzer, M.A.; McDougald, D.L.; Mitchell, J.L.; Moss, M.L.; Rabinowitz, M.H.; Rizzolio, M.C.; Schaller, L.T.; Stanford, J.B.; Tippin, T.; Warner, J.R.; Whitesell, L.G.; Wiethe, R.W.

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Synthesis of OSW-1 analogues and a dimer and their antitumor activities
pp. 2153-2156(4)
Authors: Ma, X.; Yu, B.; Hui, Y.; Miao, Z.; Ding, J.

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Artificial substrates of medium-chain elongating enzymes, hexaprenyl- and heptaprenyl diphosphate synthases
pp. 2157-2159(3)
Authors: Nagaki, M.; Kimura, K.; Kimura, H.; Maki, Y.; Goto, E.; Nishino, T.; Koyama, T.

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Combinatorial synthesis of libraries of indole derivatives
pp. 2169-2171(3)
Author: Nettekoven, M.

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Discovery of (R)-1-[2-Hydroxy-3-(4-hydroxy-phenyl)-propyl]-4-(4-methyl-benzyl)-piperidin- 4-ol: A Novel NR1/2B Subtype Selective NMDA Receptor Antagonist
pp. 2173-2176(4)
Authors: Pinard, E.; Alanine, A.; Bourson, A.; Buttelmann, B.; Gill, R.; Heitz, M.; Jaeschke, G.; Mutel, V.; Trube, G.; Wyler, R.

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Conformationally Restricted Indolopiperidine Derivatives as Potent CCR2B Receptor Antagonists
pp. 2177-2180(4)
Authors: Witherington, J.; Bordas, V.; Cooper, D.G.; Forbes, I.T.; Gribble, A.D.; Ife, R.J.; Berkhout, T.; Gohil, J.; Groot, P.H.E.

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Caged Q-rhodamine dextran: a new photoactivated fluorescent tracer
pp. 2181-2183(3)
Authors: Gee, K.R.; Weinberg, E.S.; Kozlowski, D.J.

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Design and synthesis of novel antibacterial agents with inhibitory activity against DNA polymerase III
pp. 2185-2188(4)
Authors: Ali, A.; Aster, S.D.; Graham, D.W.; Patel, G.F.; Taylor, G.E.; Tolman, R.L.; Painter, R.E.; Silver, L.L.; Young, K.; Ellsworth, K.; Geissler, W.; Harris, G.S.

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The discovery of anthranilic acid-Based MMP inhibitors. Part 2: SAR of the 5-position and P11 groups
pp. 2189-2192(4)
Authors: Levin, J.I.; Chen, J.; Du, M.; Hogan, M.; Kincaid, S.; Nelson, F.C.; Venkatesan, A.M.; Wehr, T.; Zask, A.; DiJoseph, J.; Killar, L.M.; Skala, S.; Sung, A.; Sharr, M.; Roth, C.; Jin, G.; Cowling, R.; Mohler, K.M.; Black, R.A.; March, C.J.; Skotnicki, J.S.

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Anticancer Properties for 4,4'-Dihydroxybenzophenone-2,4-dinitrophenylhydrazone (A-007)/3,7-Diaminophenothiazin-5-ium Double Salts
pp. 2193-2195(3)
Authors: Morgan, L.R.; Rodgers, A.H.; LeBlanc, B.W.; Boue, S.M.; Yang, Y.; Jursic, B.S.; Cole, R.B.

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Synthesis and antiproliferative activity of epoxy and bromo compounds derived from estrone
pp. 2197-2200(4)
Authors: Milic, D.R.; Kop, T.; Juranic, Z.; Gasic, M.J.; Solaja, B.A.

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Synthesis and pharmacology of modified amidine isoxazoline glycoprotein IIb/IIIa receptor antagonists
pp. 2201-2204(4)
Authors: Sielecki, T.M.; Liu, J.; Mousa, S.A.; Racanelli, A.L.; Hausner, E.A.; Wexler, R.R.; Olson, R.E.

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Design, synthesis and antiproliferative activity of tripentones: A new series of antitubulin agents
pp. 2205-2208(4)
Authors: Lisowski, V.; Enguehard, C.; Lancelot, J.; Caignard, D.; Lambel, S.; Leonce, S.; Pierre, A.; Atassi, G.; Renard, P.; Rault, S.

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Identification of selective inhibitors of cyclin dependent kinase 4
pp. 2209-2211(3)
Authors: Carini, D.J.; Kaltenbach, R.F.; Liu, J.; Benfield, P.A.; Boylan, J.; Boisclair, M.; Brizuela, L.; Burton, C.R.; Cox, S.; Grafstrom, R.; Harrison, B.A.; Harrison, K.; Akamike, E.; Markwalder, J.A.; Nakano, Y.; Seitz, S.P.; Sharp, D.M.; Trainor, G.L.; Sielecki, T.M.

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Novel 4-piperidinopyridine inhibitors of oxidosqualene cyclase-lanosterol synthase derived by consideration of inhibitor pKa
pp. 2213-2216(4)
Authors: Brown, G.R.; Foubister, A.J.; Johnson, M.C.; Newcombe, N.J.; Waterson, D.; Wells, S.L.

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Absolute stereostructures of novel norcadinane- and trinoreudesmane-type sesquiterpenes with nitric oxide production inhibitory activity from Alpinia oxyphylla
pp. 2217-2220(4)
Authors: Muraoka, O.; Fujimoto, M.; Tanabe, G.; Kubo, M.; Minematsu, T.; Matsuda, H.; Morikawa, T.; Toguchida, I.; Yoshikawa, M.

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Synthesis of 6-(2-thienyl)purine nucleoside derivatives that form unnatural base pairs with pyridin-2-one nucleosides
pp. 2221-2223(3)
Authors: Fujiwara, T.; Kimoto, M.; Sugiyama, H.; Hirao, I.; Yokoyama, S.

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