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Publisher: Elsevier

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Volume 11, Number 11, 4 June 2001

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Graphical Abstracts
pp. xi-xviii(8)

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Synthesis and antiviral activities of the major metabolites of the HIV protease inhibitor ABT-378 (Lopinavir)
pp. 1351-1353(3)
Authors: Sham, H.L.; Betebenner, D.A.; Herrin, T.; Kumar, G.; Saldivar, A.; Vasavanonda, S.; Molla, A.; Kempf, D.J.; Plattner, J.J.; Norbeck, D.W.

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Identification of novel potent hydroxamic acid inhibitors of peptidyl deformylase and the importance of the hydroxamic acid functionality on inhibition
pp. 1355-1358(4)
Authors: Thorarensen, A.; Douglas, J.; Rohrer, D.C.; Vosters, A.F.; Yem, A.W.; Marshall, V.D.; Lynn, J.C.; Bohanon, M.J.; Tomich, P.K.; Zurenko, G.E.; Sweeney, M.T.; Jensen, R.M.; Nielsen, J.W.; Seest, E.P.; Dolak, L.A.

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Synthesis and hydrolytic stability studies of albendazole carrier prodrugs
pp. 1359-1362(4)
Authors: Hernandez-Luis, F.; Hernandez-Campos, A.; Yepez-Mulia, L.; Cedillo, R.; Castillo, R.

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A new Antennapedia-derived vector for intracellular delivery of exogenous compounds
pp. 1363-1366(4)
Authors: Garca-Echeverra, C.; Jiang, L.; Ramsey, T.M.; Sharma, S.K.; Chenb, Y.

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6,6'-Bis(2-hydroxyphenyl)-2,2'-bipyridine manganese(III) complexes: A novel series of superoxide dismutase and catalase mimetics
pp. 1367-1370(4)
Authors: Giblin, G.M.P.; Box, P.C.; Campbell, I.B.; Hancock, A.P.; Roomans, S.; Mills, G.I.; Molloy, C.; Tranter, G.E.; Walker, A.L.; Doctrow, S.R.; Huffman, K.; Malfroy, B.

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5,5-Diaryl-2-amino-4-pentenoates as novel, potent, and selective glycine transporter type-2 reuptake inhibitors
pp. 1371-1373(3)
Authors: Isaac, M.; Slassi, A.; Silva, K.D.; Arora, J.; MacLean, N.; Hung, B.; McCallum, K.

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Synthesis of potent and selective dopamine D4 antagonists as candidate radioligands
pp. 1375-1377(3)
Authors: Huang, Y.; Kegeles, L.S.; Bae, S.; Hwang, D.; Roth, B.L.; Savage, J.E.; Laruelle, M.

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Structure-Based design, synthesis and sAR of a novel series of thiopheneamidine urokinase plasminogen activator inhibitors
pp. 1379-1382(4)
Authors: Subasinghe, N.L.; Illig, C.; Hoffman, J.; Rudolph, M.J.; Wilson, K.J.; Soll, R.; Randle, T.; Green, D.; Lewandowski, F.; Zhang, M.; Bone, R.; Spurlino, J.; desJarlais, R.; deckman, I.; Molloy, C.J.; Manthey, C.; Zhou, Z.; Sharp, C.; Maguire, D.; Crysler, C.; Grasberger, B.

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Interaction between morphine and lysine
pp. 1383-1387(5)
Authors: Nakai, S.; Yoneda, F.

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4,1-Benzoxazepinone analogues of efavirenz (Sustiva?) as HIV-1 reverse transcriptase inhibitors
pp. 1389-1392(4)
Authors: Cocuzza, A.J.; Chidester, D.R.; Cordova, B.C.; Klabe, R.M.; Jeffrey, S.; Diamond, S.; Weigelt, C.A.; Ko, S.S.; Bacheler, L.T.; Erickson-Viitanen, S.K.; Rodgers, J.D.

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Structure-activity relationships of phenylcyclohexene and biphenyl antitubulin compounds against plant and mammalian cells
pp. 1393-1396(4)
Authors: Young, D.H.; Tice, C.M.; Michelotti, E.L.; Roemmele, R.C.; Slawecki, R.A.; Rubio, F.M.; Rolling, J.A.

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Synthesis and pharmacological evaluation of 2,5-cycloamino-5H-[1]benzopyrano[4,3-d]pyrimidines endowed with in vitro antiplatelet activity
pp. 1397-1400(4)
Authors: Bruno, O.; Brullo, C.; Ranise, A.; Schenone, S.; Bondavalli, F.; Barocelli, E.; Ballabeni, V.; Chiavarini, M.; Tognolini, M.; Impicciatore, M.

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Indazolylamino quinazolines and pyridopyrimidines as inhibitors of the EGFr and c-erbB-2
pp. 1401-1405(5)
Authors: Cockerill, S.; Stubberfield, C.; Stables, J.; Carter, M.; Guntrip, S.; Smith, K.; McKeown, S.; Shaw, R.; Topley, P.; Thomsen, L.; Affleck, K.; Jowett, A.; Hayes, D.; Willson, M.; Woollard, P.; Spalding, D.

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MEK (MAPKK) inhibitors. Part 2: structure-activity relationships of 4-anilino-3-cyano-6,7-dialkoxyquinolines
pp. 1407-1410(4)
Authors: Zhang, N.; Wu, B.; Eudy, N.; Wang, Y.; Ye, F.; Powell, D.; Wissner, A.; Feldberg, L.R.; Kim, S.C.; Mallon, R.; Kovacs, E.D.; Toral-Barza, L.; Kohler, C.A.

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Aryloxy substituted N-arylpiperazinones as dual inhibitors of farnesyltransferase and geranylgeranyltransferase-I
pp. 1411-1415(5)
Authors: Bergman, J.M.; Abrams, M.T.; Davide, J.P.; Greenberg, I.B.; Robinson, R.G.; Buser, C.A.; Huber, H.E.; Koblan, K.S.; Kohl, N.E.; Lobell, R.B.; Graham, S.L.; Hartman, G.D.; Williams, T.M.; Dinsmore, C.J.

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Synthesis of a disulfide-linked octameric peptide construct carrying three different antigenic determinants
pp. 1417-1420(4)
Authors: Kragol, G.; Otvos, J.; Feng, J.; Gerhard, W.; Wade, J.D.

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Modification of constrained peptides by ring-closing metathesis reaction
pp. 1421-1423(3)
Authors: Kotha, S.; Sreenivasachary, N.; Mohanraja, K.; Durani, S.

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Amino acids and peptides. Part 39: A bivalent poly(ethylene glycol) hybrid containing an active site (RGD) and its synergistic site (PHSRN) of fibronectin
pp. 1429-1432(4)
Authors: Hojo, K.; Susuki, Y.; Maeda, M.; Okazaki, I.; Nomizu, M.; Kamada, H.; Yamamoto, Y.; Nakagawa, S.; Mayumi, T.; Kawasaki, K.

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Discovery of a nuclease-resistant, non-natural dinucleotide that inhibits HIV-1 integrase
pp. 1433-1435(3)
Authors: Taktakishvili, M.; Neamati, N.; Pommier, Y.; Nair, V.

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1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists. Part 1: discovery of the pyrrolidine scaffold and determination of its stereochemical requirements
pp. 1437-1440(4)
Authors: Hale, J.J.; Budhu, R.J.; Mills, S.G.; MacCoss, M.; Malkowitz, L.; Siciliano, S.; Gould, S.L.; deMartino, J.A.; Springer, M.S.

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Discovery of potent and selective phenylalanine derived CCR3 antagonists. Part 1
pp. 1441-1444(4)
Authors: Dhanak, D.; Christmann, L.T.; Darcy, M.G.; Jurewicz, A.J.; Keenan, R.M.; Lee, J.; Sarau, H.M.; Widdowson, K.L.; White, J.R.

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Discovery of potent and selective phenylalanine derived CCR3 receptor antagonists. Part 2
pp. 1445-1450(6)
Authors: Dhanak, D.; Christmann, L.T.; Darcy, M.G.; Keenan, R.M.; Knight, S.D.; Lee, J.; Ridgers, L.H.; Sarau, H.M.; Shah, D.H.; White, J.R.; Zhang, L.

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Inhibitors of the bacterial cell wall biosynthesis enzyme MurC
pp. 1451-1454(4)
Authors: Reck, F.; Marmor, S.; Fisher, S.; Wuonola, M.A.

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Hydrophobic forms of morphine-6-glucosides
pp. 1455-1459(5)
Authors: Schwarzinger, S.; Hartmann, M.; Kremminger, P.; Muller, N.

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Fine Tuning of physico-chemical parameters to optimise a new series of novobiocin analogues
pp. 1461-1464(4)
Authors: Schio, L.; Chatreaux, F.; Loyau, V.; Murer, M.; Ferreira, A.; Mauvais, P.; Bonnefoy, A.; Klich, M.

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Arylsulphonyl hydroxamic acids: potent and selective matrix metalloproteinase inhibitors
pp. 1465-1468(4)
Authors: Baxter, A.D.; Bhogal, R.; Bird, J.; Keily, J.F.; Manallack, D.T.; Montana, J.G.; Owen, D.A.; Pitt, W.R.; Watson, R.J.; Wills, R.E.

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