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Publisher: Elsevier

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Volume 10, Number 17, September 2000

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DNA Triple Helix Stabilization by Aminoglycoside Antibiotics
pp. 1897-1899(3)
Authors: Arya, D.P.; Coffee, R.L.

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Targeting the dimerization interface for irreversible inhibition of HIV-1 protease
pp. 1901-1903(3)
Authors: Zutshi, R.; Chmielewski, J.

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Potent inhibition of retinoic acid metabolism enzyme(s) by novel azolyl retinoids
pp. 1905-1908(4)
Authors: Njar, V.C.O.; Nnane, I.P.; Brodie, A.M.H.

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Simple Bi- and tricyclic inhibitors of human steroid 5α-reductase
pp. 1909-1911(3)
Authors: Abell, A.D.; Prince, M.J.; McNulty, A.M.; Neubauer, B.L.

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5-HETE congeners as modulators of cell proliferation
pp. 1913-1916(4)
Authors: Miller, T.A.; Ghosh, J.; Myers, C.E.; Macdonald, T.L.

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Preparation and evaluation of 1,3-diaminocyclopentane-linked dihydropyrimidinone derivatives as selective α1a-receptor antagonists
pp. 1917-1920(4)
Authors: Barrow, J.C.; Glass, K.L.; Selnick, H.G.; Freidinger, R.M.; Chang, R.S.L.; O'Malley, S.S.; Woyden, C.

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Synthesis and antiviral evaluation of nucleic acid-based (NABTM) libraries
pp. 1921-1925(5)
Authors: Jin, Y.; Roland, A.; Zhou, W.; Fauchon, M.; Lyaku, J.; Iyer, R.P.

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The Synthesis of 4-Arylsulfanyl-substituted Kainoid Analogues from trans-4-Hydroxy-l-proline
pp. 1927-1929(3)
Authors: Baldwin, J.E.; Pritchard?, G.J.; Williamson, D.S.

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The binding of cocaine to cyclodextrins
pp. 1931-1933(3)
Authors: Nesnas, N.; Lou, J.; Breslow, R.

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Solid-Phase synthesis of 4-substituted imidazoles using a scaffold approach
pp. 1935-1938(4)
Authors: Gelens, E.; Koot, W.J.; Menge, W.M.P.B.; Ottenheijm, H.C.J.; Timmerman, H.

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Quantitative structure-intestinal permeability relationship of benzamidine analogue thrombin inhibitor
pp. 1939-1942(4)
Authors: Sugano, K.; Yoshida, S.; Takaku, M.; Haramura, M.; Saitoh, R.; Nabuchi, Y.; Ushio, H.

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Nonpeptide GPIIB/IIIA receptor antagonists. Part 21: C-6 flexibility and amide bond orientation are important factors in determining the affinity of compounds for activated or resting platelet receptors
pp. 1943-1948(6)
Authors: Egbertson, M.S.; Bednar, B.; Askew, B.C.; Bednar, R.A.; Brashear, K.; Breslin, M.J.; Duggan, M.E.; Fisher, T.E.; Halczenko, W.; Hutchinson, J.H.; Ihle, N.; Prugh, J.D.; Wai, J.S.; Gould, R.J.; Hartman, G.D.

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The discovery of non-basic atrial natriuretic peptide clearance receptor antagonists. part 1
pp. 1949-1952(4)
Authors: Veale, C.A.; Alford, V.C.; Aharony, D.; Banville, D.L.; Bialecki, R.A.; Brown, F.J.; Damewood, J.R.; Dantzman, C.L.; Edwards, P.D.; Jacobs, R.T.; Mauger, R.C.; Murphy, M.M.; Palmer, W.E.; Pine, K.K.; Rumsey, W.L.; Garcia-Davenport, L.E.; Shaw, A.; Steelman, G.B.; Surian, J.M.; Vacek, E.P.

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Synthesis and biological effects of a new series of 2-amino-3-benzoylthiophenes as allosteric enhancers of A1-adenosine receptor
pp. 1953-1957(5)
Authors: Baraldi, P.G.; Zaid, A.Z.; Lampronti, I.; Fruttarolo, F.F.; Pavani, M.G.; Tabrizi, M.A.; Shryock, J.C.S.; Leung, E.; Romagnoli, R.

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Some Selective Reactions of Moenomycin A
pp. 1963-1965(3)
Authors: Vogel, S.; Buchynskyy, A.; Stembera, K.; Richter, K.; Hennig, L.; Muller, D.; Welzel, P.; Maquin, F.; Bonhomme, C.; Lampilas, M.

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Synthesis of a water-soluble prodrug of entacapone
pp. 1967-1969(3)
Authors: Leppanen, J.; Huuskonen, J.; Savolainen, J.; Nevalainen, T.; Taipale, H.; Vepsalainen, J.; Gynther, J.; Jarvinen, T.

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Potent, selective 3-pyridylethanolamine 3 adrenergic receptor agonists possessing a thiazole benzenesulfonamide pharmacophore
pp. 1971-1973(3)
Authors: Mathvink, R.J.; Tolman, J.S.; Chitty, D.; Candelore, M.R.; Cascieri, M.A.; Colwell, L.F.; Deng, L.; Feeney, W.P.; Forrest, M.J.; Hom, G.J.; MacIntyre, D.E.; Tota, L.; Wyvratt, M.J.; Fisher, M.H.; Weber, A.E.

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Substituted 2-aminopyridines as inhibitors of nitric oxide synthases
pp. 1975-1978(4)
Authors: Hagmann, W.K.; Caldwell, C.G.; Chen, P.; Durette, P.L.; Esser, C.K.; Lanza, T.J.; Kopka, I.E.; Guthikonda, R.; Shah, S.K.; MacCoss, M.; Chabin, R.M.; Fletcher, D.; Grant, S.K.; Green, B.G.; Humes, J.L.; Kelly, T.M.; Luell, S.; Meurer, R.; Moore, V.; Pacholok, S.G.; Pavia, T.; Williams, H.R.; Wong, K.K.

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Solid-phase synthesis of acridine-based threading intercalator peptides
pp. 1979-1982(4)
Authors: Carlson, C.B.; Beal, P.A.

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Towards enzyme activated antiprostatic agents
pp. 1987-1989(3)
Authors: Jones, G.B.; Mitchell, M.O.; Weinberg, J.S.; D'Amico, A.V.; Bubley, G.J.

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Synthesis and 5-Hydroxytryptamine (5-HT) activity of 2,3,4,4a-Tetrahydro-1H-pyrazino[1,2-a]quinoxalin-5-(6H)ones and 2,3,4,4a,5,6-Hexahydro-1H-pyrazino[1,2-a]quinoxalines
pp. 1991-1994(4)
Authors: Welmaker, G.S.; Nelson, J.A.; Sabalski, J.E.; Sabb, A.L.; Potoski, J.R.; Graziano, D.; Kagan, M.; Coupet, J.; Dunlop, J.; Mazandarani, H.; Rosenzweig-Lipson, S.; Sukoff, S.; Zhang, Y.

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Synthesis and erythropoietin receptor binding affinities of N,N-disubstituted amino acids
pp. 1995-1999(5)
Authors: Connolly, P.J.; Wetter, S.K.; Murray, W.V.; Johnson, D.L.; McMahon, F.J.; Farrell, F.X.; Tullai, J.; Jolliffe, L.K.

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N1-Arylsulfonyl-N2-(1-aryl)ethyl-3-phenylpropane-1,2-diami nes as novel calcimimetics acting on the calcium sensing receptor
pp. 2001-2004(4)
Authors: Dauban, P.; Ferry, S.; Faure, H.; Ruat, M.; Dodd, R.H.

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2'-deoxy-8-(propyn-1-yl)adenosine-containing oligonucleotides: effects on stability of duplex and quadruplex structures
pp. 2005-2009(5)
Authors: Catalanotti, B.; Galeone, A.; Gomez-Paloma, L.; Mayol, L.; Pepe, A.

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The Synthesis and preliminary pharmacological evaluation of 4-Methyl fentanyl
pp. 2011-2014(4)
Authors: Micovic, I.V.; Ivanovic, M.D.; Vuckovic, S.M.; Prostran, M.; Dosen-Micovic, L.; Kiricojevic, V.D.

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-Keto-ester chemistry and ketolides. synthesis and antibacterial activity of 2-halogeno, 2-methyl and 2,3 enol-ether ketolides
pp. 2019-2022(4)
Authors: Denis, A.; Bretin, F.; Fromentin, C.; Bonnet, A.; Piltan, G.; Bonnefoy, A.; Agouridas, C.

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Design and synthesis of triglyceride analogue biotinylated suicide inhibitors for directed molecular evolution of lipolytic enzymes
pp. 2027-2031(5)
Authors: Deussen H.-J.; Danielsen, S.; Breinholt, J.; Borchert, T.V.

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Molecular topology: a useful tool for the search of new antibacterials
pp. 2033-2036(4)
Authors: de Gregorio Alapont, C.; Garca-Domenech, R.; Galvez, J.; Ros, M.J.; Wolski, S.; Garcab, M.D.

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Design and synthesis of potent thiol-based inhibitors of endothelin converting enzyme-1
pp. 2037-2039(3)
Authors: Fink, C.A.; Moskal, M.; Firooznia, F.; Hoyer, D.; Symonsbergen, D.; Wei, D.; Qiao, Y.; Savage, P.; Beil, M.E.; Trapani, A.J.; Jeng, A.Y.

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Phenyloxazoles and phenylthiazoles as benzamide bioisosteres: synthesis and dopamine receptor binding profiles
pp. 2041-2044(4)
Authors: Einsiedel, J.; Thomas, C.; Hubner, H.; Gmeiner, P.

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Corrigendum to ''First pharmacophoric hypothesis for 5-HT7 antagonism'' - [Bioorg. Med. Chem. Lett. 10 (2000) 1097]?
pp. 2045-2045(1)
Authors: Lopez-Rodrguez, M.L.; Porras, E.; Benhamu, B.; Ramos, J.A.; Morcillo, M.J.; Lavandera, J.L.

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