Publisher: Elsevier

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Volume 10, Number 11, 5 June 2000

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Hepatitis C viral IRES inhibition by phenazine and phenazine-like molecules
pp. 1151-1154(4)
Authors: Wang, W.; Preville, P.; Morin, N.; Mounir, S.; Cai, W.; Siddiqui, M.A.

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Prediction of drug solubility from Monte Carlo simulations
pp. 1155-1158(4)
Authors: Jorgensen, W.L.; Duffy, E.M.

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Novel inhibitors of HIV protease - design, synthesis and biological evaluation of picomolar inhibitors containing cyclic P1/P2 scaffolds
pp. 1159-1162(4)
Authors: Spaltenstein, A.; Almond, M.R.; Bock, W.J.; Cleary, D.G.; Furfine, E.S.; Hazen, R.J.; Kazmierski, W.M.; Salituro, F.G.; Tung, R.D.; Wright, L.L.

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Carbacyclic peptide mimetics as VCAM-VLA-4 antagonists
pp. 1163-1165(3)
Authors: Tilley, J.; Kaplan, G.; Fotouhi, N.; Wolitzky, B.; Rowan, K.

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Cyclic thioether peptide mimetics as VCAM-VLA-4 antagonists
pp. 1167-1169(3)
Authors: Fotouhi, N.; Joshi, P.; Tilley, J.W.; Rowan, K.; Schwinge, V.; Wolitzky, B.

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The design and synthesis of potent cyclic peptide VCAM-VLA-4 antagonists incorporating an achiral Asp-Pro mimetic
pp. 1171-1173(3)
Authors: Fotouhi, N.; Joshi, P.; Fry, D.; Cook, C.; Tilley, J.W.; Kaplan, G.; Hanglow, A.; Rowan, K.; Schwinge, V.; Wolitzky, B.

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Design, synthesis and SAR of a series of 2-substituted 4-amino-quinazoline neuropeptide Y Y5 receptor antagonists
pp. 1175-1179(5)
Authors: Rueeger, H.; Rigollier, P.; Yamaguchi, Y.; Schmidlin, T.; Schilling, W.; Criscione, L.; Whitebread, S.; Chiesi, M.; Walker, M.W.; Dhanoab?, D.; Islamb?, I.; Zhang, J.; Gluchowskib?, C.

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Immunomodulatory activity of hexapeptides related to proline rich peptide from colostrum
pp. 1181-1183(3)
Authors: Kundu, B.; Puri, A.; Singh, G.; Sahai, R.; Tripathi, L.M.; Srivastava, V.M.L.

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-Casomorphins: substitution of phenylalanine with -homo phenylalanine increases the -type opioid receptor affinity
pp. 1185-1188(4)
Authors: Longobardo, L.; Melck, D.; Siciliano, R.; Santini, A.; Marzo, V.D.; Cammarota, G.

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The basal SAR of a novel insulin receptor activator
pp. 1189-1192(4)
Authors: Wood, H.B.; Black, R.; Salituro, G.; Szalkowski, D.; Li, Z.; Zhang, Y.; Moller, D.E.; Zhang, B.; Jones, A.B.

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COBRA-1, A rationally-designed epoxy-THF containing compound with potent tubulin depolymerizing activity as a novel anticancer agent
pp. 1193-1197(5)
Authors: Jan, S.; Mao, C.; Vassilev, A.O.; Navara, C.S.; Uckun, F.M.

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Diamino benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors. Part 6: Further focus on the contracted C4'-side chain analogues
pp. 1199-1202(4)
Authors: Takeuchi, K.; Kohn, T.J.; Harper, R.W.; Lin, H.; Gifford-Moore, D.S.; Richett, M.E.; Sall, D.J.; Smith, G.F.; Zhang?, M.

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Methaqualone derivatives are potent noncompetitive AMPA receptor antagonists
pp. 1203-1205(3)
Authors: Chenard, B.L.; Menniti, F.S.; Pagnozzi, M.J.; Shenk, K.D.; Ewing, F.E.; Welch, W.M.

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9-Benzylpurines with inhibitory activity against Mycobacterium tuberculosis
pp. 1207-1210(4)
Authors: Bakkestuen, A.K.; Gundersen L.-L.; Langli, G.; Liu, F.; Nolsoe, J.M.J.

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Synthesis and structure-activity relationships of quaternary ammonium cephalosporins with 3-pyrazolylpyridinium derivatives
pp. 1211-1214(4)
Authors: Chang, K.Y.; Kim, S.H.; Nam, G.; Seo, J.H.; Kim, J.H.; Ha, D.

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Bicyclic nucleoside inhibitors of Varicella-Zoster Virus (VZV): the effect of a terminal halogen substitution in the side-chain
pp. 1215-1217(3)
Authors: Brancale, A.; McGuigan, C.; Andrei, G.; Snoeck, R.; de Clercq, E.; Balzarini, J.

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Mass spectrometry reveals elastase inhibitors from the reactive centre loop of α1-antitrypsin
pp. 1219-1221(3)
Authors: Wright, P.A.; Rostom, A.A.; Robinson, C.V.; Schofield, C.J.

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A focused compound library of novel N-(7-indolyl)benzenesulfonamides for the discovery of potent cell cycle inhibitors
pp. 1223-1226(4)
Authors: Owa, T.; Okauchi?, T.; Yoshimatsu, K.; Sugi, N.H.; Ozawa, Y.; Nagasu, T.; Koyanagi, N.; Okabe, T.; Kitoh, K.; Yoshino, H.

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'Double-drugs'- A new class of prodrug form of an HIV protease inhibitor conjugated with a reverse transcriptase inhibitor by a spontaneously cleavable linker
pp. 1227-1231(5)
Authors: Matsumoto, H.; Hamawaki, T.; Ota, H.; Kimura, T.; Goto, T.; Sano, K.; Hayashi, Y.; Kiso, Y.

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Synthesis of glycosylated polyethylenimine with reduced toxicity and high transfecting efficiency
pp. 1233-1235(3)
Authors: Leclercq, F.; Dubertret, C.; Pitard, B.; Scherman, D.; Herscovici, J.

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Squalamine analogues as potential anti-trypanosomal and anti-leishmanial compounds
pp. 1237-1239(3)
Authors: Khabnadideh, S.; Tan, C.L.; Croft, S.L.; Kendrick, H.; Yardley, V.; Gilbert, I.H.

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(+)-4-Phosphonophenylglycine (PPG) a new group III selective metabotropic glutamate receptor agonist
pp. 1241-1244(4)
Authors: Gasparini, F.; Inderbitzin, W.; Francotte, E.; Lecis, G.; Richert, P.; Dragic, Z.; Kuhn, R.; Flor, P.J.

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The design and synthesis of the high efficacy, non-peptide CCK1 receptor agonist PD 170292
pp. 1245-1248(4)
Authors: Bernad, N.; Burgaud, B.G.M.; Horwell, D.C.; Lewthwaite, R.A.; Martinez, J.; Pritchard, M.C.

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Nucleotide libraries as a source of biologically relevant chemical diversity: solution-phase synthesis
pp. 1249-1252(4)
Authors: Zhou, W.; Upendran, S.; Roland, A.; Jin, Y.; Iyer, R.P.

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Synthesis and activity studies of conformationally restricted α-ketoamide factor Xa inhibitors
pp. 1253-1256(4)
Authors: Cacciola, J.; Fevig, J.M.; Stouten?, P.F.W.; Alexander, R.S.; Knabb, R.M.; Wexler, R.R.

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Carbocyclic influenza neuraminidase inhibitors possessing a C3-cyclic amine side chain: synthesis and inhibitory activity
pp. 1257-1260(4)
Authors: Lew, W.; Wu, H.; Chen, X.; Graves, B.J.; Escarpe, P.A.; MacArthur, H.L.; Mendel, D.B.; Kim, C.U.

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SAR of 4-hydroxypiperidine and hydroxyalkyl substituted heterocycles as novel p38 map kinase inhibitors
pp. 1261-1264(4)
Authors: Revesz, L.; Di Padova, F.E.; Buhl, T.; Feifel, R.; Gram, H.; Hiestand, P.; Manning, U.; Zimmerlin, A.G.

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The synthesis and in vitro cytotoxic studies of novel oxa-spermidine derivatives and homologues
pp. 1265-1267(3)
Authors: Kuksa, V.A.; Pavlov, V.A.; Lin, P.K.T.

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Cytotoxic halogenoacrylic derivatives of distamycin A
pp. 1269-1272(4)
Authors: Cozzi, P.; Beria, I.; Caldarelli, M.; Capolongo, L.; Geroni, C.; Mongelli, N.

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Cytotoxic α-bromoacrylic derivatives of distamycin analogues modified at the amidino moiety
pp. 1273-1276(4)
Authors: Cozzi, P.; Beria, I.; Caldarelli, M.; Geroni, C.; Mongelli, N.; Pennella, G.

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Conformationally-restricted ligands for the histamine H1 receptor
pp. 1277-1279(3)
Authors: Upton, C.; Osborne, R.H.; Jaffar, M.

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4-[(8-Alkyl-8-azabicyclo[3.2.1]octyl-3-yl)-3-arylanilino]-N,N-diethylbenzami des: high affinity, selective ligands for the delta opioid receptor illustrate factors important to antagonist activity
pp. 1281-1284(4)
Authors: Thomas, J.B.; Atkinson, R.N.; Rothman, R.B.; Burgess, J.P.; Mascarella, S.W.; dersch, C.M.; Xu, H.; Carroll, F.I.

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Discovery of a potent, non-triketone type inhibitor of 4-hydroxyphenylpyruvate dioxygenase
pp. 1297-1298(2)
Authors: Lin, S.; Lin, Y.; Lin, T.; Yang D.-Y.

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Functionalized nucleoside 5'-triphosphates for in vitro selection of new catalytic ribonucleic acids
pp. 1299-1302(4)
Authors: Matulic-Adamic, J.; Daniher, A.T.; Karpeisky, A.; Haeberli, P.; Sweedler, D.; Beigelman, L.

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Synthesis and evaluation of geldanamycin-testosterone hybrids
pp. 1303-1306(4)
Authors: Kuduk, S.D.; Harris, C.R.; Zheng, F.F.; Sepp-Lorenzino, L.; Ouerfelli, Q.; Rosen, N.; Danishefsky, S.J.

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