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Publisher: Elsevier

Volume 10, Number 8, April 2000

Isoxazolines and isoxazoles as factor Xa inhibitors
pp. 685-689(5)
Authors: Pruitt, J.R.; Pinto, D.J.; Estrella, M.J.; Bostrom, L.L.; Knabb, R.M.; Wong, P.C.; Wright, M.R.; Wexler, R.R.

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The synthesis and vasopressin (AVP) antagonist activity of a novel series of n-aroyl-2,4,5,6-tetrahydropyrazolo [3,4-d]thieno[3,2-b]azepines
pp. 695-698(4)
Authors: Albright, J.D.; Santos, E.G.D.; Dusza, J.P.; Chan, P.S.; Coupet, J.; Ru, X.; Mazandarani, H.

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Antitumor agents. Part 202: Novel 2'-amino chalcones: design, synthesis and biological evaluation
pp. 699-701(3)
Authors: Xia, Y.; Yang, Z.; Xia, P.; Bastow, K.F.; Nakanishi, Y.; Lee K.-H.

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Suitably functionalised pyrimidines as potential antimycotic agents
pp. 703-706(4)
Authors: Agarwal, N.; Raghuwanshi, S.K.; Upadhyay, D.N.; Shukla, P.K.; Ram, V.J.

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α-Ketoamides, α-ketoesters and α-diketones as HCV NS3 protease inhibitors
pp. 711-713(3)
Authors: Han, W.; Hu, Z.; Jiang, X.; decicco, C.P.

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4-Thiazolidinones: novel inhibitors of the bacterial enzyme murB
pp. 715-717(3)
Authors: Andres, C.J.; Bronson, J.J.; D'Andrea, S.V.; deshpande, M.S.; Falk, P.J.; Grant-Young, K.A.; Harte, W.E.; Ho, H.; Misco, P.F.; Robertson, J.G.; Stock, D.; Sun, Y.; Walsh, A.W.

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Heterocyclic bibenzimidazole derivatives as topoisomerase I inhibitors
pp. 719-723(5)
Authors: Jin, S.; Kim, J.S.; Sim, S.; Liu, A.; Pilch, D.S.; Liu, L.F.; LaVoie, E.J.

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N-Acyl phenylalanine analogues as potent small molecule VLA-4 antagonists
pp. 725-727(3)
Authors: Chen, L.; Tilley, J.W.; Huang, T.; Miklowski, D.; Trilles, R.; Guthrie, R.W.; Luk, K.; Hanglow, A.; Rowan, K.; Schwinge, V.; Wolitzky, B.

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N-Benzylpyroglutamyl-l-phenylalanine derivatives as VCAM/VLA-4 antagonists
pp. 729-733(5)
Authors: Chen, L.; Tilley, J.W.; Guthrie, R.W.; Mennona, F.; Huang, T.; Kaplan, G.; Trilles, R.; Miklowski, D.; Huby, N.; Schwinge, V.; Wolitzky, B.; Rowan, K.

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High incorporation of l-amino acids to cereulide, an emetic toxin from Bacillus cereus
pp. 735-739(5)
Authors: Kuse, M.; Franz, T.; Koga, K.; Suwan, S.; Isobe, M.; Agata, N.; Ohta, M.

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Cyclodextrin-peptide hybrid as a hydrolytic catalyst having multiple functional groups
pp. 741-743(3)
Authors: Tsutsumi, H.; Hamasaki, K.; Mihara, H.; Ueno, A.

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Guanylpiperidine peptidomimetics: potent and selective bis-cation inhibitors of factor Xa
pp. 745-749(5)
Authors: Tamura, S.Y.; Levy, O.E.; Uong, T.H.; Reiner, J.E.; Goldman, E.A.; Ho, J.Z.; Cohen, C.R.; Bergum, P.W.; Nutt, R.F.; Brunck, T.K.; Semple, J.E.

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Conversion of a polysaccharide to nitric oxide-releasing form. dual-mechanism anticoagulant activity of diazeniumdiolated heparin
pp. 751-753(3)
Authors: Saavedra, J.E.; Mooradian, D.L.; Mowery, K.A.; Schoenfisch, M.H.; Citro, M.L.; Davies, K.M.; Meyerhoff, M.E.; Keefer, L.K.

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Structural comparison between type I and type II antagonists: possible implications in the drug design of AT1 antagonists
pp. 755-758(4)
Authors: Roumelioti, P.; Tselios, T.; Alexopoulos, K.; Mavromoustakos, T.; Kolocouris, A.; Moore, G.J.; Matsoukas, J.M.

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Macrocarpins A-D, new cytotoxic nor-triterpenes from Maytenus macrocarpa
pp. 759-762(4)
Authors: Chavez, H.; Rodrguez, G.; Estevez-Braun, A.; Ravelo, A.G.; Estevez-Reyes, R.; Gonzalez, A.G.; Fdez-Puente, J.L.; Garca-Gravalos, D.

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The abasic site as a target for generation of locally multiply damaged sites
pp. 763-766(4)
Authors: Martelli, A.; Berthet, N.; Constant, J.; demeunynck, M.; Lhomme, J.

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Synthesis and pharmacology of new enantiopure Δ3-4-arylkainoids
pp. 771-773(3)
Authors: Rondeau, D.; Gill, P.; Chan, M.; Curry, K.; Lubell, W.D.

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Serendipitous synthesis of novel dehydro- and dechloro-pseudomycin B (PSB) derivatives
pp. 775-778(4)
Authors: Zhang, Y.; Boyer, R.; Sun, X.; Paschal, J.; Chen S.-H.

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The design, synthesis and physical chemical properties of novel human vasopressin V2-receptor antagonists optimized for parenteral delivery
pp. 783-786(4)
Authors: Ashwell, M.A.; Bagli, J.F.; Caggiano, T.J.; Chan, P.S.; Molinari, A.J.; Palka, C.; Park, C.H.; Rogers, J.F.; Sherman, M.; Trybulski, E.J.; Williams, D.K.

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Incorporation of a 4-hydroxy-N-acetylprolinol nucleotide analogue improves the 3'-exonuclease stability of 2'-5'-oligoadenylate-antisense conjugates
pp. 801-804(4)
Authors: Verheijen, J.C.; van Roon, A.; Meeuwenoord, N.J.; Stuivenberg, H.R.; Bayly, S.F.; Chen, L.; van der Marel, G.A.; Torrence, P.F.; van Boom, J.H.

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Novel 3-(4-piperidinylthio)-1H-indoles as potent nonopioid orally active central analgesics
pp. 805-809(5)
Authors: Potin, D.; Parnet, V.; Teulon, J.; Camborde, F.; Caussade, F.; Meignen, J.; Provost, D.; Cloarec, A.

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Leukotriene B4 photoaffinity probes: design, synthesis and evaluation of new arylazide-1,3-disubstituted cyclohexanes
pp. 811-814(4)
Authors: Durand, D.; Hullot, P.; Vidal, J.; Girard, J.; Baneres, J.L.; Parello, J.; Muller, A.; Bonne, C.; Rossi, J.

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Synthesis and antibacterial activity of novel 6-O-substituted erythromycin A derivatives
pp. 815-819(5)
Authors: Clark, R.F.; Ma, Z.; Wang, S.; Griesgraber, G.; Tufano, M.; Yong, H.; Li, L.; Zhang, X.; Nilius, A.M.; Chu, D.T.W.; Or, Y.S.

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Design, synthesis, and structure-activity relationship studies of ATP analogues as DNA gyrase inhibitors
pp. 821-826(6)
Authors: Lubbers, T.; Angehrn, P.; Gmunder, H.; Herzig, S.; Kulhanek, J.

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Chemo- and enzymatic synthesis of partially and fully N-deacetylated 4-methylumbelliferyl chitobiosides: Fluorogenic substrates for chitinase
pp. 827-829(3)
Authors: Honda, Y.; Tanimori, S.; Kirihata, M.; Kaneko, S.; Tokuyasu, K.; Hashimoto, M.; Watanabe, T.

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ORL1 receptor ligands: Structure-activity relationships of 8-cycloalkyl-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-ones
pp. 831-834(4)
Authors: Rover, S.; Wichmann, J.; Jenck, F.; Adam, G.; Cesura, A.M.

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Synthesis and antifungal activity of a ferrocene-fluconazole analogue
pp. 839-841(3)
Authors: Biot, C.; Francois, N.; Maciejewski, L.; Brocard, J.; Poulain, D.

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