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Publisher: Elsevier

Volume 8, Number 19, 6 October 1998

Biaryl acids: novel non-nucleoside inhibitors of HIV reverse transcriptase types 1 and 2
pp. 2623-2628(6)
Authors: Milton, J.; Slater, M.J.; Bird, A.J.; Spinks, D.; Scott, G.; Price, C.E.; Downing, S.; Green, D.V.S.; Madar, S.; Bethell, R.; Stammers, D.K.

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Synthesis and evaluation of a novel series of phosphodiesterase IV inhibitors. A potential treatment for asthma
pp. 2629-2634(6)
Authors: Beasley, S.C.; Cooper, N.; Gowers, L.; Gregory, J.P.; Haughan, A.F.; Hellewell, P.G.; Macari, D.; Miotla, J.; Montana, J.G.; Morgan, T.; Naylor, R.; Runcie, K.A.; Tuladhar, B.; Warneck, J.B.H.

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Aryl sulfonamides as selective PDE4 inhibitors
pp. 2635-2640(6)
Authors: Montana, J.G.; Buckley, G.M.; Cooper, N.; Dyke, H.J.; Gowers, L.; Gregory, J.P.; Hellewell, P.G.; Kendall, H.J.; Lowe, C.; Maxey, R.; Miotla, J.; Naylor, R.J.; Runcie, K.A.; Tuladhar, B.; Warneck, J.B.H.

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Potassium peroxymonosulfate (oxone) - an efficient oxidizing agent for phosphothio compounds
pp. 2641-2646(6)
Authors: Wozniak, L.A.; Koziolkiewicz, M.; Kobylanska, A.; Stec, W.J.

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P2-proline-derived inhibitors of Calpain I
pp. 2647-2652(6)
Authors: Tripathy, R.; Gu, Z.; Dunn, D.; Senadhi, S.E.; Ator, M.A.; Chatterjee, S.

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Novel antineoplastic agents with efficacy against multidrug resistant tumor cells
pp. 2653-2656(4)
Authors: Medina, J.C.; Shan, B.; Beckmann, H.; Farrell, R.P.; Clark, D.L.; Learned, R.M.; Roche, D.; Li, A.; Baichwal, V.; Case, C.; Baeuerle, P.A.; Rosen, T.; Jaen, J.C.

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The synthesis and biological activity of a novel series of diazepine MMP inhibitors
pp. 2657-2662(6)
Authors: Levin, J.I.; DiJoseph, J.F.; Killar, L.M.; Sung, A.; Walter, T.; Sharr, M.A.; Roth, C.E.; Skotnicki, J.S.; Albright, J.D.

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Thalidomide analogs and PDE4 inhibition
pp. 2669-2674(6)
Authors: Muller, G.W.; Shire, M.G.; Wong, L.M.; Corral, L.G.; Patterson, R.T.; Chen, Y.; Stirling, D.I.

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New generation dopaminergic agents. 5. Heterocyclic bioisosteres that exploit the 3-OH-N1-phenylpiperazine dopaminergic template
pp. 2675-2680(6)
Authors: Mewshaw, R.E.; Verwijs, A.; Shi, X.; McGaughey, G.B.; Nelson, J.A.; Mazandarani, H.; Brennan, J.A.; Marquis, K.L.; Coupet, J.; Andree, T.H.

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A high affinity, mu-opioid receptor-selective enkephalin analogue lacking an N-terminal tyrosine
pp. 2681-2684(4)
Authors: Mosberg, H.I.; Ho, J.C.; Sobczyk-Kojiro, K.

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Design of a high affinity peptidomimetic opioid agonist from peptide pharmacophore models
pp. 2685-2688(4)
Authors: Wang, C.; McFadyen, I.J.; Traynor, J.R.; Mosberg, H.I.

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Pyrroles and other heterocycles as inhibitors of P38 kinase
pp. 2689-2694(6)
Authors: de Laszlo, S.E.; Visco, D.; Agarwal, L.; Chang, L.; Chin, J.; Croft, G.; Forsyth, A.; Fletcher, D.; Frantz, B.; Hacker, C.; Hanlon, W.; Harper, C.; Kostura, M.; Li, B.; Luell, S.; MacCoss, M.; Mantlo, N.; O'Neill, E.A.; Orevillo, C.; Pang, M.; Parsons, J.; Rolando, A.; Sahly, Y.; Sidler, K.; Widmer, W.R.; O'Keefe, S.J.

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Novel protein kinase C inhibitors: α-terthiophene derivatives
pp. 2695-2698(4)
Authors: Kim, D.S.H.L.; Ashendel, C.L.; Zhou, Q.; Chang, C.; Lee, E.; Chang, C.

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Tropane-based amino acids for peptide structure-function studies: inhibitors of platelet aggregation
pp. 2699-2704(6)
Authors: Thompson, P.E.; Steer, D.L.; Aguilar, M.; Hearn, M.T.W.

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The de novo design and synthesis of cyclic urea inhibitors of factor Xa: initial sar studies
pp. 2705-2710(6)
Authors: Galemmo, R.A.; Maduskuie, T.P.; Dominguez, C.; Rossi, K.A.; Knabb, R.M.; Wexler, R.R.; Stouten, P.F.W.

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NGB 2904 and NGB 2849: two highly selective dopamine D3 receptor antagonists
pp. 2715-2718(4)
Authors: Yuan, J.; Chen, X.; Brodbeck, R.; Primus, R.; Braun, J.; Wasley, J.W.F.; Thurkauf, A.

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Studies on the C-terminal of hexapeptide inhibitors of the hepatitis C virus serine protease
pp. 2719-2724(6)
Authors: Llinas-Brunet, M.; Bailey, M.; deziel, R.; Fazal, G.; Gorys, V.; Goulet, S.; Halmos, T.; Maurice, R.; Poirier, M.; Poupart, M.; Rancourt, J.; Thibeault, D.; Wernic, D.; Lamarre, D.

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Synthesis and Biological Activity of Novel Thiazolidinediones
pp. 2725-2730(6)
Authors: Prabhakar, C.; Madhusudhan, G.; Sahadev, K.; Reddy, C.M.; Sarma, M.R.; Reddy, G.O.; Chakrabarti, R.; Rao, C.S.; Kumar, T.D.; Rajagopalan, R.

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Nonsteroidal progesterone receptor antagonists based on a conformationally-restricted subseries of 6-aryl-1,2-dihydro-2,2,4-trimethylquinolines
pp. 2731-2736(6)
Authors: Hamann, L.G.; Winn, D.T.; Pooley, C.L.F.; Tegley, C.M.; West, S.J.; Farmer, L.J.; Zhi, L.; Edwards, J.P.; Marschke, K.B.; Mais, D.E.; Goldman, M.E.; Jones, T.K.

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2-substituted-4-methoxybenzimidazole-based PDE4 inhibitors
pp. 2737-2742(6)
Authors: Regan, J.; Bruno, J.; McGarry, D.; Poli, G.; Hanney, B.; Bower, S.; Travis, J.; Sweeney, D.; Miller, B.; Souness, J.; Djuric, S.

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Voltage-dependent ion channel formation by rigid rod-shaped polyols in planar lipid bilayers
pp. 2743-2746(4)
Authors: Sakai, N.; Ni, C.; Bezrukov, S.M.; Matile, S.

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Conformationally constrained inhibitors of caspase-1 (interleukin-1 converting enzyme) and of the human CED-3 homologue caspase-3 (CPP32, APOPAIN)
pp. 2757-2762(6)
Authors: Karanewsky, D.S.; Bai, X.; Linton, S.D.; Krebs, J.F.; Wu, J.; Pham, B.; Tomaselli, K.J.

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Synthesis and cytotoxicity of acetyl-4H, 9H-naphtho[2,3-b]thiophene-4,9-diones
pp. 2763-2768(6)
Authors: Huang, L.; Kuo, S.; Perng, C.; Chao, Y.; Wu, T.; McPhail, A.T.; Mauger, A.; Cheng, H.; Lee, K.

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Reversal of multidrug resistance (MDR) by aspidofractinine-type indole alkaloids
pp. 2769-2772(4)
Authors: Kam, T.; Subramaniam, G.; Sim, K.; Yoganathan, K.; Koyano, T.; Toyoshima, M.; Rho, M.; Hayashi, M.; Komiyama, K.

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Synthesis and anticancer evaluation of certain -aryloxymethyl-α-methylene--phenyl--butyrolactones
pp. 2773-2776(4)
Authors: Wang, T.; Lee, K.; Chen, Y.; Liou, S.; Tzeng, C.

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2-pyridinyl-3-(4-methylsulfonyl)phenylpyridines: selective and orally active cyclooxygenase-2 inhibitors
pp. 2777-2782(6)
Authors: Friesen, R.W.; Brideau, C.; Chan, C.C.; Charleson, S.; deschenes, D.; Dube, D.; Ethier, D.; Fortin, R.; Gauthier, J.Y.; Girard, Y.; Gordon, R.; Greig, G.M.; Riendeau, D.; Savoie, C.; Wang, Z.; Wong, E.; Visco, D.; Xu, L.J.; Young, R.N.

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Sialyl Lewis X-Polysaccharide Conjugates : Targeting Inflammatory Lesions
pp. 2783-2786(4)
Authors: Sakagami, M.; Horie, K.; Nakamoto, K.; Kawaguchi, T.; Hamana, H.

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Synthesis and immunosuppressant activity of pyrazole carboxamides
pp. 2787-2792(6)
Authors: Wang, A.X.; Xie, Q.; Lane, B.; Mollison, K.W.; Hsieh, G.C.; Marsh, K.; Sheets, M.P.; Luly, J.R.; Coghlan, M.J.

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Synthesis and antibacterial activity of 2-alkoxy penems
pp. 2793-2796(4)
Authors: Afonso, A.; Hon, F.; Fett, N.; Weinstein, J.; Ganguly, A.K.; Naples, L.; Hare, R.S.; Miller, G.H.

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Structure-activity studies related to ABT-594, a potent nonopioid analgesic agent: effect of pyridine and azetidine ring substitutions on nicotinic acetylcholine receptor binding affinity and analgesic activity in mice
pp. 2797-2802(6)
Authors: Holladay, M.W.; Bai, H.; Li, Y.; Lin, N.; Daanen, J.F.; Ryther, K.B.; Wasicak, J.T.; Kincaid, J.F.; He, Y.; Hettinger, A.; Huang, P.; Anderson, D.J.; Bannon, A.W.; Buckley, M.J.; Campbell, J.E.; Donnelly-Roberts, D.L.; Gunther, K.L.; Kim, D.J.B.; Kuntzweiler, T.A.; Sullivan, J.P.; decker, M.W.; Arneric, S.P.

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Exploration of -turn scaffolding motifs as components of sialyl Lex mimetics and their relevance to P-selectin
pp. 2803-2808(6)
Authors: Hanessian, S.; Huynh, H.K.; Reddy, G.V.; McNaughton-Smith, G.; Ernst, B.; Kolb, H.C.; Magnani, J.; Sweeley, C.

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Design and synthesis of dipeptidyl α','-epoxy ketones, potent irreversible inhibitors of the cysteine protease cruzain
pp. 2809-2812(4)
Authors: Roush, W.R.; Gonzalez, F.V.; McKerrow, J.H.; Hansell, E.

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Design and synthesis of a pyridone-based phosphotyrosine mimetic
pp. 2813-2816(4)
Authors: Fu, J.; Castelhano, A.L.

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