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Publisher: Elsevier

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Volume 8, Number 18, 22 September 1998

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A photoactivated prodrug
pp. 2419-2422(4)
Authors: Yaoming, W.; Yinfa, Y.; dehua, P.; Bing, G.

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NMR and topochemical studies of peptidomimetic HIV-I protease inhibitors containing a cis-epoxide amide isostere
pp. 2423-2426(4)
Authors: Seonggu, R.; Baek, S.; Bogman, L.; Chihyo, P.; Nakyen, C.; Chang, S.L.; Young, C.S.; Hoil, C.; Jong, S.K.; Heungsik, Y.; Sung, C.K.; Jong, H.O.

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Design and synthesis of analogs of vitamin E: antiproliferative activity against human breast adenocarcinoma cells
pp. 2433-2438(6)
Authors: Arya, P.; Alibhai, N.; Qin, H.; Burton, G.W.; Batist, G.; You, S.X.; Alaoui-Jamali, M.A.

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Solid-phase synthesis of potential protein tyrosine phosphatase inhibitors via the UGI four-component condensation
pp. 2443-2446(4)
Authors: Zhengong, L.; Su, L.Y.; Pallen, C.J.; Ganesan, A.

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Synthesis and Biological Evaluation of Two Analogues of (S)-α-Methyl-3-carboxyphenylalanine
pp. 2447-2450(4)
Authors: Dawei, M.; Zhaochun, M.; Kozikowski, A.P.; Pshenichkin, S.; Wroblewski, J.T.

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N-carbamoyl analogs of Zafirlukast: potent receptor antagonists of leukotriene D4
pp. 2451-2456(6)
Authors: Brown, M.F.; Marfat, A.; Antognoli, G.; Chambers, R.J.; Cheng, J.B.; Damon, D.B.; Liston, T.E.; McGlynn, M.A.; O'Sullivan, S.P.; Owens, B.S.; Pillar, J.S.; Shirley, J.T.; Watson, J.W.

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Templates for design of inhibitors for serine proteases: application of the program dock to the discovery of novel inhibitors for thrombin
pp. 2463-2466(4)
Authors: Massova, I.; Martin, P.; Bulychev, A.; Kocz, R.; Doyle, M.; Edwards, B.F.P.; Mobashery, S.

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Design and synthesis of N-alkylated saccharins as selective α-1A adrenergic receptor antagonists
pp. 2467-2472(6)
Authors: Nerenberg, J.B.; Erb, J.M.; Thompson, W.J.; Lee, H.; Guare, J.P.; Munson, P.M.; Bergman, J.M.; Huff, J.R.; Broten, T.P.; Chang, R.S.L.; Chen, T.B.; O'Malley, S.; Schorn, T.W.; Scott, A.L.

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Synthesis and effects of novel thiazole derivatives against thrombocytopenia
pp. 2473-2478(6)
Authors: Tsuji, K.; Ogino, T.; Seki, N.; Sawada, M.; Sudo, Y.; Nishigaki, F.; Manda, T.; Matsuo, M.

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H-phosphonate derivatives as novel peptide deformylase inhibitors
pp. 2479-2482(4)
Authors: Hu, Y.; Rajagopalan, P.T.R.; Pei, D.

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The development of novel and selective p56lck tyrosine kinase inhibitors
pp. 2489-2494(6)
Authors: Bullington, J.L.; Cameron, J.C.; Davis, J.E.; Dodd, J.H.; Harris, C.A.; Henry, J.R.; Pellegrino-Gensey, J.L.; Rupert, K.C.; Siekierka, J.J.

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Selective α-1A adrenergic receptor antagonists. Effects of pharmacophore regio- and stereochemistry on potency and selectivity
pp. 2495-2500(6)
Authors: Patane, M.A.; DiPardo, R.M.; Price, R.P.; Chang, R.S.L.; Ransom, R.W.; O'Malley, S.S.; Di Salvo, J.; Bock, M.G.

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Naphthoquinone Analogs as Inactivators of cdc25 Phosphatase
pp. 2507-2510(4)
Authors: Seung, W.H.; Junguk, P.; Lee, S.; Wonho, K.; Kyunghwa, K.; Kyung, H.C.

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5'-peptidyl substituents allow a tuning of the affinity of oligodeoxyribonucleotides for RNA
pp. 2511-2516(6)
Authors: Sarracino, D.A.; Steinberg, J.A.; Vergo, M.T.; Woodworth, G.F.; Tetzlaff, C.N.; Richert, C.

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Design of Novel Tripeptides with Macrophage Migration-Enhancing Activity
pp. 2517-2520(4)
Authors: Nunami, K.; Yamada, M.; Shimizu, R.

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Inhibitors of farnesyl protein transferase. Synthesis and biological activity of amide and cyanoguanidine derivatives containing a 5,11-dihydro[1]benzthiepin, benzoxepin, and benzazepin [4,3-b]pyridine ring system
pp. 2521-2526(6)
Authors: Wolin, R.; Connolly, M.; Kelly, J.; Weinstein, J.; Rosenblum, S.; Afonso, A.; James, L.; Kirschmeier, P.; Bishop, W.R.

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Dibasic benzo[b]thiophene derivatives as a novel class of active site directed thrombin inhibitors. 2. Exploring interactions at the proximal (S2) binding site
pp. 2527-2532(6)
Authors: Sall, D.J.; Briggs, S.L.; Chirgadze, N.Y.; Clawson, D.K.; Gifford-Moore, D.S.; Klimkowski, V.J.; McCowan, J.R.; Smith, G.F.; Wikel, J.H.

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Modulation of apoptosis in human lymphocytes by adenosine analogues
pp. 2533-2538(6)
Authors: Barbieri, D.; Franceschi, C.; Camaioni, E.; Costanzi, S.; Vittori, S.; Volpini, R.; Cristalli, G.

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A new spacer group derived from arylmalonaldehydes for glucuronylated prodrugs
pp. 2545-2548(4)
Authors: Papot, S.; Combaud, D.; Gesson J.-P.

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Substrate specificity of thermostable farnesyl diphosphate synthase with alkyl group homologs of isopentenyl diphosphate
pp. 2549-2554(6)
Authors: Nagaki, M.; Kannari, H.; Ishibashi, J.; Maki, Y.; Nishino, T.; Ogura, K.; Koyama, T.

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Two Novel Oleanolic Acid Saponins Having a Sialyl Lewis X Mimetic Structure from Achyranthes fauriei Root
pp. 2555-2558(4)
Authors: Ida, Y.; Satoh, Y.; Katsumata, M.; Nagasao, M.; Hirai, Y.; Kajimoto, T.; Katada, N.; Yasuda, M.; Yamamoto, T.

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Benzylamine-based Selective and Orally Bioavailable Inhibitors of Thrombin
pp. 2563-2568(6)
Authors: Koo, L.; Jung, W.; Cheol, W.P.; Chang, Y.H.; In, C.K.; Sangsoo, K.; Yeong, S.O.; O, H.K.; Lee, S.; Hee, D.P.; Sang, W.K.; Yong, H.L.; Yung, J.Y.

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Synthesis of 13C labelled Daidzein and Formononetin
pp. 2569-2572(4)
Authors: Whalley, J.L.; Bond, T.J.; Botting, N.P.

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Synthesis of boronic acid analogs of L-arginine as alternate substrates or inhibitors of nitric oxide synthase
pp. 2573-2576(4)
Authors: Lebarbier, C.; Carreaux, F.; Carboni, B.; Boucher, J.L.

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New antifungals selected by molecular topology
pp. 2577-2582(6)
Authors: Pastor, L.; Garcia-Domenech, R.; Galvez, J.; Wolski, S.; Garcia, M.D.

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PD 176252 - The First High Affinity Non-peptide Gastrin-Releasing Peptide (BB2) Receptor Antagonist
pp. 2589-2594(6)
Authors: Ashwood, V.; Brownhill, V.; Higginbottom, M.; Horwell, D.C.; Hughes, J.; Lewthwaite, R.A.; McKnight, A.T.; Pinnock, R.D.; Pritchard, M.C.; Suman-Chauhan, N.; Webb, C.; Williams, S.C.

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In situ generated O-Glycan Core 1 Structure as Substrate for Gal(1-3)GalNAc -1,6-GlcNAc Transferase
pp. 2595-2598(4)
Authors: Dudziak, G.; Zeng, S.; Berger, E.G.; Gallego, R.G.; Kamerling, J.P.; Kragl, U.; Wandrey, C.

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General synthesis of 3-substituted alkenyl GABA as potential anticonvulsants
pp. 2599-2602(4)
Authors: Serfass, L.; Casara, P.J.

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Synthesis and binding of stable bisubstrate ligands for phosphoglycerate kinase
pp. 2603-2608(6)
Authors: Williams, D.M.; Jakeman, D.L.; Vyle, J.S.; Williamson, M.P.; Blackburn, G.M.

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Synthesis and properties of prodrugs activated in hypoxia to give bleomycin analogues
pp. 2609-2614(6)
Authors: Highfield, J.A.; Mehta, L.K.; Parrick, J.; Candeias, L.P.; Wardman, P.

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Mechanism based representation of the active site of 5α-reductase (5AR)
pp. 2615-2620(6)
Authors: Ahmed, S.; denison, S.

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In vitro evaluation and crystallographic analysis of a new class of selective, non-amide-based thrombin inhibitors
pp. 2621-2621(1)
Authors: Lu, T.; Tomczuk, B.; Illig, C.R.; Bone, R.; Murphy, L.; Spurlino, J.; Salemme, F.R.; Soll, R.M.

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