Publisher: Elsevier

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Volume 8, Number 13, 7 July 1998

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Novel 1,3-disubstituted-5, 10-dihydro-5, 10-dioxo-1H-benzo[g] isochromene-3 carboxamides as potent antitumor agents
pp. 1579-1584(6)
Authors: Wuyi, W.; Tiechao, L.; Milburn, R.; Yates, J.; Hinnant, E.; Luzzio, M.J.; Noble, S.A.; Attardo, G.

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Asymmetric synthesis and anti-HIV activity of L-carbocyclic 2?,3?-didehydro-2?,3?-dideoxyadenosine
pp. 1585-1588(4)
Authors: Peiyuan, W.; Schinazi, R.F.; Chu, C.K.

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Synthesis and biological evaluation of a series of 2?-fluorinated-2?,3?-dideoxy-2?,3?-dideh ydro-(l)-nucleosides
pp. 1589-1594(6)
Authors: Chen, S.; Qin, W.; Mao, J.; King, I.; Dutschman, G.E.; Gullen, E.A.; Cheng, Y.; Doyle, T.W.

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In vitro evaluation and crystallographic analysis of a new class of selective, non-amide-based thrombin inhibitors
pp. 1595-1600(6)
Authors: Tianbao, L.; Tomczuk, B.; Illig, C.R.; Bone, R.; Murphy, L.; Spurlino, J.; Salemme, F.R.; Soll, R.M.

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Novel modified tripeptide inhibitors of α47 mediated lymphoid cell adhesion to MAdCAM-1
pp. 1601-1606(6)
Authors: Shroff, H.N.; Schwender, C.F.; Baxter, A.D.; Brookfield, F.; Payne, L.J.; Cochran, N.A.; Gallant, D.L.; Briskin, M.J.

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Synthesis and Biological Properties of New 1-Methylcarbapenems
pp. 1607-1612(6)
Authors: Kye, J.S.; Kyung, H.Y.; Dong, J.K.; Sang, W.P.; Bong, S.K.; Sang, J.L.; Jae, D.H.; Seung, Y.P.

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Diarylsulfonamides as selective, non-peptidic thrombin inhibitors
pp. 1613-1618(6)
Authors: Weber, I.R.; Neidlein, R.; von der Saal, W.; Grams, F.; Leinert, H.; Strein, K.; Engh, R.A.; Kucznierz, R.

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Practical Synthesis of Taxol Side Chain
pp. 1619-1622(4)
Authors: Ha H.-J.; Park, G.; Ahn, Y.; Gwan, S.L.

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Carbohydrate modifications in the spirostane cellobioside cholesterol absorption inhibitor series
pp. 1623-1628(6)
Authors: deninno, M.P.; Eller, C.; Etienne, J.B.

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A new series of cyclic amino acids as inhibitors of S-adenosyl L-methionine synthetase
pp. 1629-1634(6)
Authors: Lavrador, K.; Guillerm, D.; Guillerm, G.

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Synthesis and Biological Activity of Lactones en route to Altohyrtin A
pp. 1635-1638(4)
Authors: Hermitage, S.A.; Murphy, A.; Roberts, S.M.

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Adenosine deaminase inhibitors. Synthesis and biological evaluation of aralkyladenines (ARADS)
pp. 1639-1642(4)
Authors: Curtis, M.A.; Varkhedkar, V.; Pragnacharyulu, P.V.P.; Abushanab, E.

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Inhibitors of the bacterial cell wall biosynthesis enzyme Mur d
pp. 1643-1648(6)
Authors: Gegnas, L.D.; Waddell, S.T.; Chabin, R.M.; Reddy, S.; Wong, K.K.

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Thrombin receptor (PAR-1) antagonists. Heterocycle-based peptidomimetics of the SFLLR agonist motif
pp. 1649-1654(6)
Authors: Hoekstra, W.J.; Hulshizer, B.L.; McComsey, D.F.; Andrade-Gordon, P.; Kauffman, J.A.; Addo, M.F.; Oksenberg, D.; Scarborough, R.M.; Maryanoff, B.E.

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Synthesis and acetylcholinesterase inhibitory activity of (±)-14-fluorohuperzine A
pp. 1661-1664(4)
Authors: Zeng, F.; Jiang, H.; Tang, X.; Chen, K.; Ji, R.

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Identification of a potent analogue of nazumamide a through iteration of combinatorial tetrapeptide libraries
pp. 1669-1672(4)
Authors: Kundu, B.; Bauser, M.; Betschinger, J.; Kraas, W.; Jung, G.

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Potent and efficacious thienylamidine-incorporated thrombin inhibitors
pp. 1683-1686(4)
Authors: Koo, L.; Sang, Y.H.; Mikyung, Y.; Dong, S.K.

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Carbaxylosides of 4-Ethyl-2-oxo-2H-benzopyran-7-yl as Non-hydrolyzable, Orally Active Venous Antithrombotic Agents
pp. 1687-1688(2)
Authors: Jeanneret, V.; Vogel, P.; Renaut, P.; Millet, J.; Theveniaux, J.; Barberousse, V.

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Conodiparines A-D, new bisindoles from Tabernaemontana. Reversal of vincristine-resistance with cultured cells
pp. 1693-1696(4)
Authors: Kam, T.; Sim, K.; Koyano, T.; Toyoshima, M.; Hayashi, M.; Komiyama, K.

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Identification and SAR for a selective, nonpeptidyl thrombin inhibitor
pp. 1697-1702(6)
Authors: Naylor-Olsen, A.M.; Ponticello, G.S.; Lewis, S.D.; Mulichak, A.M.; Zhonguo, C.; Habecker, C.N.; Phillips, B.T.; Sanders, W.M.; Tucker, T.J.; Shafer, J.A.; Vacca, J.P.

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Ascorbic acid-based inhibitors of α-amylases
pp. 1703-1706(4)
Authors: Abell, A.D.; Ratcliffe, M.J.; Gerrard, J.

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Synthesis of betulinic acid derivatives with activity against human melanoma
pp. 1707-1712(6)
Authors: Kim, D.S.H.L.; Pezzuto, J.M.; Pisha, E.

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Peptide-based inhibitors of the hepatitis C virus serine protease
pp. 1713-1718(6)
Authors: Llinas-Brunet, M.; Bailey, M.; Fazal, G.; Goulet, S.; Halmos, T.; Laplante, S.; Maurice, R.; Poirier, M.; Poupart, M.; Thibeault, D.; Wernic, D.; Lamarre, D.

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C6 modification of the pyridinone core of thrombin inhibitor L-374,087 as a means of enhancing its oral absorption
pp. 1719-1724(6)
Authors: Isaacs, R.C.A.; Cutrona, K.J.; Newton, C.L.; Sanderson, P.E.J.; Solinsky, M.G.; Baskin, E.P.; Chen, I.; Cooper, C.M.; Cook, J.J.; Gardell, S.J.; Lewis, S.D.; Lucas, R.J.; Lyle, E.A.; Lynch, J.J.; Naylor-Olsen, A.M.; Stranieri, M.T.; Vastag, K.; Vacca, J.P.

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Korundamine A, a novel HIV-inhibitory and antimalarial ?hybrid? naphthylisoquinoline alkaloid heterodimer from Ancistrocladus korupensis
pp. 1729-1734(6)
Authors: Hallock, Y.F.; Cardellina, J.H.; Schaffer, M.; Bringmann, G.; Francois, G.; Boyd, M.R.

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Neuronorm is a potent and water soluble Neurokinin A receptor antagonist
pp. 1735-1740(6)
Authors: Lombardi, A.; D'Agostino, B.; Filippelli, A.; Pedone, C.; Matera, M.G.; Falciani, M.; de Rosa, M.; Rossi, F.; Pavone, V.

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Synthesis and hypoxia-selective cytotoxicity of a 2-nitroimidazole mustard
pp. 1741-1744(4)
Authors: Lee, H.H.; Palmer, B.D.; Wilson, W.R.; denny, W.A.

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Heteroatom- and carbon-linked biphenyl analogs of Brequinar as immunosuppressive agents
pp. 1745-1750(6)
Authors: Batt, D.G.; Petraitis, J.J.; Sherk, S.R.; Copeland, R.A.; Dowling, R.L.; Taylor, T.L.; Jones, E.A.; Magolda, R.L.; Jaffee, B.D.

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The synthesis of symmetrical spermine conjugates using solid-phase chemistry
pp. 1751-1756(6)
Authors: Page, P.; Burrage, S.; Baldock, L.; Bradley, M.

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Synthesis of a high-mannose-type glycopeptide analog containing a glucose-asparagine linkage
pp. 1763-1766(4)
Authors: deras, I.L.; Takegawa, K.; Kondo, A.; Kato, I.; Lee, Y.C.

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The synthesis of new adenosine A3 selective ligands containing bioisosteric isoxazoles
pp. 1767-1770(4)
Authors: Mogensen, J.P.; Roberts, S.M.; Bowler, A.N.; Thomsen, C.; Knutsen, L.J.S.

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3. Endothelin antagonists: discovery of EMD 122946, a highly potent and orally active ETA selective antagonist
pp. 1771-1776(6)
Authors: Mederski, W.W.K.R.; Dorsch, D.; Osswald, M.; Anzali, S.; Christadler, M.; Schmitges, C.; Schelling, P.; Wilm, C.; Fluck, M.

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Peptidyl human heart chymase inhibitors. Part 1: Synthesis and inhibitory activity of difluoromethylene ketone derivatives bearing P' binding subsites
pp. 1778-1778(1)
Authors: Eda, M.; Ashimori, A.; Akahoshi, F.; Yoshimura, T.; Inoue, Y.; Fukaya, C.; Nakajima, M.; Fukuyama, H.; Imada, T.; Nakamura, N.

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Peptidyl human heart chymase inhibitors. Part 2: Discovery of highly selective difluoromethylene ketone derivatives with Glu at P3 site
pp. 1779-1779(1)
Authors: Eda, M.; Ashimori, A.; Akahoshi, F.; Yoshimura, T.; Inoue, Y.; Fukaya, C.; Nakajima, M.; Fukuyama, H.; Imada, T.; Nakamura, N.

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