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Volume 6, Number 15, 6 August 1996

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Tc-99m-labeled fibrinogen receptor antagonists: design and synthesis of cyclic RGD peptides for the detection of thrombi
pp. 1741-1746(6)
Authors: Harris, T.D.; Rajopadhye, M.; Damphousse, P.R.; Glowacka, D.; Yu, K.; Bourque, J.P.; Barrett, J.A.; Damphousse, D.J.; Heminway, S.J.; Lazewatsky, J.; Mazaika, T.; Carroll, T.R.

Determination of the absolute configuration of the nonsteroidal contraceptive agent centchroman by X-ray crystallography on its N-methyl iodide salt
pp. 1747-1752(6)
Authors: Srivastava, N.; Ray, S.; Dwivedy, I.; Wilson, S.R.; Hom, R.K.; Katzenellenbogen, J.A.

Tetrazole-substituted ureas as inhibitors of acyl-CoA:cholesterol O-acyltransferase (ACAT). A novel preparation of ureas from weakly nucleophilic amines
pp. 1753-1758(6)
Authors: Purchase, C.F.; White, A.D.; Anderson, M.K.; Bocan, T.M.A.; Bousley, R.F.; Hamelehle, K.L.; Homan, R.; Krause, B.R.; Lee, P.; Mueller, S.B.; Speyer, C.; Stanfield, R.L.; Reindel, J.F.

Potent and selective PKC inhibitory 5-membered ring analogs of balanol with replacement of the carboxamide moiety
pp. 1759-1764(6)
Authors: Jagdmann, G.E.; defauw, J.M.; Lampe, J.W.; Darges, J.W.; Kalter, K.

Modelisation, synthesis and antiviral evaluation of new 2,3-disubstituted thiazolidinone nucleoside analogues
pp. 1775-1780(6)
Authors: Graciet, J.C.; Niddam, V.; Gamberoni, M.; Trabaud, C.; dessolin, J.; Medou, M.; Mourier, N.; Zoulim, F.; Borel, C.; Hantz, O.; Camplo, M.; Chermann, J.C.; Kraus, J.L.

Preparation, antimicrobial evaluation and mutagenicity of differently substituted [2-hydroxyaryl]-[1-methyl-5-nitro-1H-2-imidazolyl]methanols.
pp. 1781-1784(4)
Authors: Arredondo, Y.; Moreno-Manas, M.; Pleixats, R.; Palacin, C.; Raga, M.M.; Castello, J.M.; Ortiz, J.A.

Synthesis and properties of 2'-5' and 3'-5' linked α-oligoriboadenylates
pp. 1785-1790(6)
Authors: Sawai, H.; Ito, T.; Kokaji, K.; Shimazu, M.; Shinozuka, K.; Taira, H.

Identification and structure-activity relationship studies of osthol, a cytotoxic principle from Cnidium monnieri
pp. 1791-1794(4)
Authors: Hitotsuyanagi, Y.; Kojima, H.; Ikuta, H.; Takeya, K.; Itokawa, H.

Synthesis of a piperidinomethylthiophene derivative as H2-antagonist with inhibitory activity against helicobacter pylori
pp. 1795-1798(4)
Authors: Kojima, K.; Nakajima, K.; Kurata, H.; Tabata, K.; Utsui, Y.

8-Amino-6-(arylsulphonyl)-5-nitroquinolines: novel nonpeptide neuropeptide Y1 receptor antagonists
pp. 1809-1814(6)
Authors: Wright, J.; Bolton, G.; Creswell, M.; Downing, D.; Georgic, L.; Heffner, T.; Hodges, J.; MacKenzie, R.; Wise, L.

Synthesis of furo[2,3-c]pyran--D-thymidine
pp. 1815-1818(4)
Authors: Bousquie, I.; Madiot, V.; Florent, J.; Monneret, C.

The chemical evolution of N,N-dimethyl-2-[5-(1,2,4-triazol-4-yl)-1H-indol-3-yl]ethylamine (L-741,604) and analogues: potent and selective agonists for 5-HT1D receptors
pp. 1825-1830(6)
Authors: Sternfeld, F.; Baker, R.; Broughton, H.B.; Guiblin, A.R.; Jelley, R.A.; Matassa, V.G.; Reeve, A.J.; Beer, M.S.; Stanton, J.A.; Hargreaves, R.J.; Shepheard, S.L.; Longmore, J.; Razzaque, Z.; Graham, M.I.; Sohal, B.; Street, L.J.

DNA threading agents: effect of sidechain bulk on DNA binding and cytotoxicity of 9-anilinoacridine-4-carboxamides
pp. 1831-1836(6)
Authors: Searcey, M.; Martin, P.N.; Howarth, N.M.; Madden, B.; Wakelin, L.P.G.

Synthesis and antitumor evaluation of paclitaxel phosphonooxymethyl ethers: a novel class of water soluble paclitaxel pro-drugs
pp. 1837-1842(6)
Authors: Golik, J.; Wong, H.S.L.; Shu, H.C.; Doyle, T.W.; Wright, J.J.K.; Knipe, J.; Rose, W.C.; Casazza, A.M.; Vyas, D.M.

Synthesis and evaluation of amino acid ester prodrugs of penciclovir
pp. 1849-1854(6)
Authors: Dae-Kee, K.; Namkyu, L.; Guang, J.I.; Young-Woo, K.; Kieyoung, C.; Hun-Taek, K.; Yong-Baik, C.; Won-Son, C.; Inho, J.; Key, H.K.

Synthesis and in vitro evaluation of sugar-modified carboranyluridines
pp. 1855-1858(4)
Authors: Imamura, K.; Yamamoto, Y.

Synthesis and bioactivity of new antineoplastic terpenylquinones
pp. 1859-1864(6)
Authors: Gordaliza, M.; del Corral, J.M.M.; Castro, M.A.; Mahiques, M.M.; Garcia-Gravalos, M.D.; Feliciano, A.S.

A Novel Class of Vitamin D Analogs Synthesis and Preliminary Biological Evaluation
pp. 1865-1868(4)
Authors: Kanzler, S.; Halkes, S.; van de Velde, J.P.; Reischl, W.

Identification and characterisation of an inhibitor of interleukin-8: a receptor based approach.
pp. 1869-1874(6)
Authors: Attwood, M.R.; Borkakoti, N.; Bottomley, G.A.; Conway, E.A.; Cowan, I.; Fallowfield, A.G.; Handa, B.K.; Jones, P.S.; Keech, E.; Kirtland, S.J.; Williams, G.; Wilson, F.X.

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