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Publisher: Elsevier

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Volume 5, Number 22, 16 November 1995

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Isosteric replacement of the indole nucleus by benzothiophene in a series of pyrido[2,3-b]indoles with potential anxiolytic activity
pp. 2589-2592(4)
Authors: Blackburn, T.P.; Davies, D.T.; Forbes, I.T.; Hayward, C.J.; Johnson, C.N.; Martin, R.T.; Piper, D.C.; Thomas, D.R.; Thompson, M.; Upton, N.; Ward, R.W.

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Inhibitors of human collagenase: dipeptide mimetics with lactam and azalactam moieties at the P2'P3' position
pp. 2593-2598(6)
Authors: Bird, J.; Harper, G.P.; Hughes, I.; Hunter, D.J.; Karran, E.H.; Markwell, R.E.; Miles-Williams, A.J.; Rahman, S.S.; Ward, R.W.

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Synthesis and Antiviral Evaluation of Enantiomeric 2',3'-Dideoxy-and 2',3'-Didehydro-2',3'-dideoxy-4'-Thionucleosides.
pp. 2599-2604(6)
Authors: Young, R.J.; Shaw-Ponter, S.; Thomson, J.B.; Miller, J.A.; Cumming, J.G.; Pugh, A.W.; Rider, P.

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Balanced AT1 and AT2 angiotensin II antagonists. I. new orally active 5-carboxyl imidazolyl biphenyl sulfonylureas.
pp. 2605-2610(6)
Authors: Deprez, P.; Heckmann, B.; Corbier, A.; Vevert, J.; Fortin, M.; Guillaume, J.

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Balanced AT1 and AT2 angiotensin II antagonists. II. Potent 5 α-hydroxyacid imidazolyl biphenyl sulfonylureas
pp. 2611-2616(6)
Authors: Deprez, P.; Guillaume, J.; Corbier, A.; Fortin, M.; Vevert, J.; Heckmann, B.

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Balanced AT1 and AT2 angiotensin II antagonists. III. Potent and orally active 5--ketosulfoxide imidazolyl biphenyl sulfonylureas.
pp. 2617-2622(6)
Authors: Deprez, P.; Guillaume, J.; Corbier, A.; Vevert, J.; Fortin, M.; Heckmann, B.

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Rational design, synthesis, and X-ray structure of renin inhibitors with extended P1 sidechains
pp. 2623-2626(4)
Authors: Lefker, B.A.; Hada, W.A.; Wright, A.S.; Martin, W.H.; Stock, I.A.; Schulte, G.K.; Pandit, J.; Danley, D.E.; Ammirati, M.J.; Sneddon, S.F.

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Synthesis of conformationally-constrained stereospecific analogs of glutamic acid as antagonists of metabotropic receptors
pp. 2627-2632(6)
Authors: Tellier, F.; Acher, F.; Brabet, I.; Pin, J.; Bockaert, J.; Azerad, R.

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The synthesis and biological evaluation of hypericin analogs
pp. 2633-2636(4)
Authors: Kraus, G.A.; Zhang, W.

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Spiroketal Glycomimetics: The Synthesis of a Conformationally Restrained Sialyl Lewis X Mimic.
pp. 2637-2642(6)
Authors: Birkbeck, A.A.; Ley, S.V.; Prodger, J.C.

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Tetramic acids as novel glycine site antagonists
pp. 2643-2648(6)
Authors: Mawer, I.M.; Kulagowski, J.J.; Leeson, P.D.; Grimwood, S.; Marshall, G.R.

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The discovery of a series of new non-indole 5HT1D agonists
pp. 2649-2654(6)
Authors: van Lommen, G.; de Bruyn, M.; Schroven, M.; Verschueren, W.; Janssens, W.; Verrelst, J.; Leysen, J.

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Inhibition of glycosidases by substituted amidines
pp. 2655-2660(6)
Authors: Bleriot, Y.; Dintinger, T.; Genre-Grandpierre, A.; Padrines, M.; Tellier, C.

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4,5-Dihydro-4-oxo-3H-imidazo[4,5-c]pyridines: potent arylacetic acid-derived AT1 antagonists with improved affinity for the AT2 receptor
pp. 2665-2670(6)
Authors: Mederski, W.W.K.R.; Dorsch, D.; Osswald, M.; Beier, N.; Lues, I.; Minck, K.; Schelling, P.; Ladstetter, B.J.

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Spiro-piperidine non-peptide neurokinin-1 receptor antagonists
pp. 2671-2676(6)
Authors: Armour, D.R.; Watson, S.P.; Pegg, N.A.; Heron, N.M.; Middlemiss, D.; C., C.; Cholerton, T.J.; Hubbard, T.; Vinader, M.V.; Davies, H.G.; Cocker, J.D.; Bays, D.E.; Ward, P.

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Local constrained shifty pseudopeptides inhibitors of ras-farnesyl transferase
pp. 2677-2682(6)
Authors: Byk, G.; Duchesne, M.; Parker, F.; Lelievre, Y.; Guitton, J.D.; Clerc, F.F.; Becquart, J.; Tocque, B.; Scherman, D.

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Development of Fluorescence-Emitting Antibody Labeling Substance by Near-Infrared Ray Excitation
pp. 2689-2694(6)
Authors: Ito, S.; Muguruma, N.; Kakehashi, Y.; Hayashi, S.; Okamura, S.; Shibata, H.; Okahisa, T.; Kanamori, M.; Shibamura, S.; Takesako, K.; Nozawa, M.; Ishida, K.; Shiga, M.

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Synthesis of novel 20-oxo-pregnacalciferol analogs with binding affinity to the progesterone receptor
pp. 2695-2700(6)
Authors: Perlman, K.L.; Darwish, H.M.; DeLuca, H.F.; Sicinski, R.R.

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Cycloalkylpiperazines as HIV-1 Protease Inhibitors: Enhanced Oral Absorption
pp. 2707-2712(6)
Authors: Kim, B.M.; Evans, B.E.; Gilbert, K.F.; Hanifin, C.M.; Vacca, J.P.; Michelson, S.R.; Darke, P.L.; Zugay, J.A.; Emini, E.A.; Schleif, W.; Lin, J.H.; Chen, I.; Vastag, K.; Anderson, P.S.; Huff, J.R.

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Synthesis and biological evaluation of an alkenyldiarylmethane (ADAM) which acts as a novel non-nucleoside HIV-1 reverse transcriptase inhibitor
pp. 2713-2716(4)
Authors: Cushman, M.; Golebiewski, M.; Buckheit, R.W.; Graham, L.; Rice, W.G.

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6,3'-dinitroflavone, a novel high affinity ligand for the benzodiazepine receptor with potent anxiolytic properties.
pp. 2717-2720(4)
Authors: Marder, M.; Viola, H.; Wasowski, C.; Wolfman, C.; Waterman, P.G.; Medina, J.H.; Paladini, A.C.

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Synthesis and incorporation of 2'-amino acid conjugated nucleotides into ribozymes
pp. 2721-2724(4)
Authors: Matulic-Adamic, J.; Beigelman, L.; Dudycz, L.W.; Gonzalez, C.; Usman, N.

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Evaluation of substituted benzamides as P2 ligands for symmetry-based inhibitors of HIV protease
pp. 2725-2728(4)
Authors: Kempf, D.J.; Flentge, C.A.; Wideburg, N.E.; Saldivar, A.; Vasavanonda, S.; Norbeck, D.W.

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Differential RXR & RAR activity of stilbene retinoid analogs bearing thiazole and imidazole carboxylic acids
pp. 2729-2734(6)
Authors: Beard, R.L.; Colon, D.F.; Klein, E.S.; Vorse, K.A.; Chandraratna, R.A.S.

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Novel C-4 Paclitaxel (Taxol(R)) Analogs: Potent Antitumor Agents
pp. 2741-2746(6)
Authors: Shu-Hui, C.; Jian-Mei, W.; Long, B.H.; Fairchild, C.A.; Carboni, J.; Mamber, S.W.; Rose, W.C.; Johnston, K.; Casazza, A.M.; Kadow, J.F.; Farina, V.; Vyas, D.M.; Doyle, T.W.

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Synthesis of dibenzo[a,d]cycloheptanes as cytokine biosynthesis inhibitors
pp. 2749-2754(6)
Authors: Ting, P.C.; Lee, J.F.; Solomon, D.M.; Smith, S.R.; Terminelli, C.A.; Jakway, J.P.; Zambas, D.N.

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Inhibition of an HIV-1 tat-derived peptide binding to TAR RNA by aminoglycoside antibiotics
pp. 2755-2760(6)
Authors: Houng-Yau, M.; Galan, A.A.; Halim, N.S.; Mack, D.P.; Moreland, D.W.; Sanders, K.B.; Truong, H.N.; Czarnik, A.W.

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Phenyl-Glycinol Based NK1 Receptor Antagonists - Towards the Minimum Pharmacophore
pp. 2761-2766(6)
Authors: Owens, A.P.; Williams, B.J.; Harrison, T.; Swain, C.J.; Baker, R.; Sadowski, S.; Cascieri, M.A.

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