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Publisher: Elsevier

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Volume 5, Number 4, 16 February 1995

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Structural and stereochemical requirements of time-dependent inactivators of the interleukin-1 converting enzyme
pp. 315-318(4)
Authors: Prasad, C.V.C.; Prouty, C.P.; Hoyer, D.; Ross, T.M.; Salvino, J.M.; Awad, M.; Graybill, T.L.; Schmidt, S.J.; Osifo, I.K.; Dolle, R.E.; Helaszek, C.T.; Miller, R.E.; Ator, M.A.

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Inhibitors of human leukocyte elastase. 2.1 synthesis and SAR of benzisothiazolinylmethyl aryl ethers
pp. 319-324(6)
Authors: Subramanyam, C.; Bell, M.R.; Ferguson, E.; Gordon, R.G.; Dunlap, R.P.; Franke, C.; Mura, A.J.

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Inhibitors of human leukocyte elastase. 3.1 inhibition by tetrahydrobenzisothiazolinylmethyl aryl carboxylates.
pp. 325-330(6)
Authors: Subramanyam, C.; Bell, M.R.; Ghose, A.K.; Kumar, V.; Dunlap, R.P.; Franke, C.; Mura, A.J.

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The design of potent and stable benzisothiazolone inhibitors of human leukocyte elastase
pp. 331-336(6)
Authors: Hlasta, D.J.; Bell, M.R.; Court, J.J.; Cundy, K.C.; Desai, R.C.; Ferguson, E.W.; Gordon, R.J.; Kumar, V.; Maycock, A.L.; Subramanyan, C.; Dunlap, R.P.; Eiff, S.L.; Franke, C.A.; Mura, A.J.; Rowlands, A.G.

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Relationship between structure and bioavailability in a series of hydroxamate based metalloprotease inhibitors
pp. 337-342(6)
Authors: Singh, J.; Conzentino, P.; Cundy, K.; Gainor, J.A.; Gilliam, C.L.; Gordon, T.D.; Johnson, J.A.; Morgan, B.A.; Schneider, E.D.; Wahl, R.C.; Whipple, D.A.

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Hydroxamate inhibitors of the matrix metallo-proteinases (MMPs) containing novel P1' heteroatom based modifications
pp. 343-348(6)
Authors: Tomczuk, B.E.; Gowravaram, M.R.; Johnson, J.S.; Delecki, D.; Cook, E.R.; Ghose, A.K.; Mathiowetz, A.M.; Spurlino, J.C.; Rubin, B.; Smith, D.L.; Pulvino, T.; Wahl, R.C.

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Hydroxamate inhibitors of human gelatinase B (92 kDa).
pp. 349-352(4)
Authors: Wahl, R.C.; Pulvino, T.A.; Mathiowetz, A.M.; Ghose, A.K.; Johnson, J.S.; Delecki, D.; Cook, E.R.; Gainor, J.A.; Gowravaram, M.R.; Tomczuk, B.E.

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Structure activity relationships of non-peptide bradykinin B2 receptor antagonists
pp. 357-362(6)
Authors: Salvino, J.M.; Seoane, P.R.; Douty, B.D.; Awad, M.A.; Hoyer, D.; Ross, T.M.; Dolle, R.E.; Houck, W.T.; Faunce, D.M.; Sawutz, D.G.

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Synthesis of non-peptide bradykinin B2 receptor antagonists
pp. 363-366(4)
Authors: Douty, B.D.; Salvino, J.M.; Seoane, P.R.; Dolle, R.E.

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Ace inhibitors as a template for the design of bradykinin B2 receptor antagonists
pp. 367-370(4)
Authors: Hoyer, D.; Awad, M.M.A.; Salvino, J.M.; Seoane, P.R.; Dolle, R.E.; Houck, W.T.; Sawutz, D.G.

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Structure-activity studies of the natural product substance P antagonist win 64821
pp. 377-380(4)
Authors: Barrow, C.J.; Musza, L.L.; Cooper, R.

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Morpholinoalkylindenes as antinociceptive agents: novel cannabinoid receptor agonists
pp. 381-386(6)
Authors: Kumar, V.; Alexander, M.D.; Bell, M.R.; Eissenstat, M.A.; Casiano, F.M.; Chippari, S.M.; Haycock, D.A.; Luttinger, D.A.; Kuster, J.E.; Miller, M.S.; Stevenson, J.I.; Ward, S.J.

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Inhibition of human erythrocyte calpain I by novel quinolinecarboxamides
pp. 387-392(6)
Authors: Graybill, T.L.; Dolle, R.E.; Osifo, I.K.; Schmidt, S.J.; Gregory, J.S.; Harris, A.L.; Miller, M.S.

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Characterization of a continuous fluorogenic assay for calpain I. Kinetic evaluation of peptide aldehydes, halomethyl ketones and (acyloxy)methyl ketones as inhibitors of the enzyme
pp. 393-398(6)
Authors: Harris, A.L.; Gregory, J.S.; Maycock, A.L.; Graybill, T.L.; Osifo, I.K.; Schmidt, S.J.; Dolle, R.E.

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Potent mammalian topoisomerase II inhibitors: 1-cyclopropyl-6,8-difluoro-1,4-dihydro-7-(2,6-dimethyl-4-pyridinyl)-4-substi tuted-quinolines.
pp. 399-404(6)
Authors: Kuo, G.; Eissenstat, M.A.; Wentland, M.P.; Robinson, R.G.; Klingbeil, K.M.; Danz, D.W.; Coughlin, S.A.

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The antitumor activity of novel pyrazoloquinoline derivatives.
pp. 405-410(6)
Authors: Wentland, M.P.; Aldous, S.C.; Gruett, M.D.; Perni, R.B.; Powles, R.G.; Danz, D.W.; Klingbeil, K.M.; Peverly, A.D.; Robinson, R.G.; Corbett, T.H.; Rake, J.B.; Coughlin, S.A.

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Achiral Internucleoside Linkages 3: CH2-NH-CH2 Linkage
pp. 411-414(4)
Authors: Prasad, C.V.C.; Caulfield, T.J.; Prouty, C.P.; Saha, A.K.; Schairer, W.C.; Yawman, A.; Upson, D.A.; Kruse, L.I.

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