Skip to main content

Publisher: Elsevier

Volume 5, Number 2, 19 January 1995

Alkoxy substituted benzisothiazolone (BIT) derivatives: potent inhibitors of human leukocyte elastase.
pp. 105-109(5)
Authors: Desai, R.C.; Dunlap, R.P.; Farrell, R.P.; Ferguson, E.; Franke, C.A.; Gordon, R.; Hlasta, D.J.; Talomie, T.G.

Favourites:
ADD

Synthesis of conformationally restricted substance P antagonists
pp. 111-114(4)
Authors: Howard, H.R.; Shenk, K.D.; Coffman, K.C.; Bryce, D.K.; Crawford, R.T.; McLean, S.A.

Favourites:
ADD

Synthesis of 2-o-heteroaroyl taxanes: evaluation of microtubule assembly promotion and cytotoxicity
pp. 115-118(4)
Authors: Georg, G.I.; Harriman, G.C.B.; Ali, S.M.; Datta, A.; Hepperle, M.; Himes, R.H.

Favourites:
ADD

Non-peptide oxytocin antagonists: identification and synthesis of a potent camphor aminosuccinimide
pp. 119-122(4)
Authors: Hobbs, D.W.; Gould, N.P.; Hoffman, J.B.; Clineschmidt, B.V.; Pettibone, D.J.; Veber, D.F.; Freidinger, R.M.

Favourites:
ADD

Bivalent indoles exhibiting serotonergic binding affinity
pp. 123-126(4)
Authors: LeBoulluec, K.L.; Mattson, R.J.; Mahle, C.D.; McGovern, R.T.; Nowak, H.P.; Gentile, A.J.

Favourites:
ADD

SCH 51048, a novel broad-spectrum orally active antifungal agent: synthesis and preliminary structure-activity profile
pp. 127-132(6)
Authors: Saksena, A.K.; Girijavallabhan, V.M.; Lovey, R.G.; Desai, J.A.; Pike, R.E.; Jao, E.; Wang, H.; Ganguly, A.K.; Loebenberg, D.; Hare, R.S.; Cacciapuoti, A.; Parmegiani, R.M.

Favourites:
ADD

Synthesis and estrogen receptor binding of fluorinated diethylstilbestrol derivatives
pp. 133-138(6)
Authors: Rhee, C.K.; Chae, K.; Levy, L.A.; Korach, K.S.

Favourites:
ADD

Synthesis and Anticonvulsant Properties of BW A78U Structurally-Related Compounds
pp. 139-144(6)
Authors: Desaubry, L.; Wermuth, C.G.; Boehrer, A.; Marescaux, C.; Bourguignon, J.

Favourites:
ADD

Non-peptidic inhibitors of neutral endopeptidase 24.11 - 1. Discovery and optimization of potency
pp. 145-150(6)
Authors: de Lombaert, S.; Blanchard, L.; Tan, J.; Sakane, Y.; Berry, C.; Ghai, R.D.

Favourites:
ADD

Non-peptidic inhibitors of neutral endopeptidase 24.11 - 2. Design and pharmacology of orally active phosphonate prodrugs
pp. 151-154(4)
Authors: de Lombaert, S.; Blanchard, L.; Berry, C.; Ghai, R.D.; Trapani, A.J.

Favourites:
ADD

AT1 selective angiotensin II antagonists with phenoxyphenylacetic acid as a biphenyl replacement part I
pp. 155-158(4)
Authors: Fitch, K.J.; Walsh, T.F.; Patchett, A.A.; Chang, R.S.L.; Siegl, P.K.S.; Faust, K.A.; Chen, T.; Lotti, V.J.; Kivlighn, S.D.; Zingaro, G.J.; Greenlee, W.J.

Favourites:
ADD

Ruthenium tetroxide oxidation of grundmann's ketone derived from vitamin D3
pp. 159-162(4)
Authors: Sicinski, R.R.; DeLuca, H.F.

Favourites:
ADD

Acyl CoA:cholesterol acyltransferase (ACAT) inhibitors: ureas bearing heterocyclic groups bioisosteric for an imidazole
pp. 167-172(6)
Authors: Wilde, R.G.; Billheimer, J.T.; Germain, S.J.; Gillies, P.J.; Higley, C.A.; Kezar, H.S.; Maduskuie, T.P.; Shimshick, E.S.; Wexler, R.R.

Favourites:
ADD
Favourites:
ADD

Acyl CoA:cholesterol acyltransferase (ACAT) inhibitors: heterocyclic bioisosteres for the urea group in DuP 128
pp. 177-180(4)
Authors: Wilde, R.G.; Klaczkiewicz, J.D.; Billheimer, J.T.; Wexler, R.R.; Gillies, P.J.

Favourites:
ADD

A pair of new apotirucallane triterpenes, meliavolkensins A and B, from Melia volkensii (Meliaceae)
pp. 181-184(4)
Authors: Zeng, L.; Gu, Z.; Chang, C.; Smith, D.L.; McLaughlin, J.L.

Favourites:
ADD

Thiophene Derivatives as Extremely High Affinity P3' Ligands for the Hydroxyethylpiperazine Class of HIV-1 Protease Inhibitors
pp. 185-190(6)
Authors: Kim, B.M.; Guare, J.P.; Vacca, J.P.; Michelson, S.R.; Darke, P.L.; Zugay, J.A.; Emini, E.A.; Schleif, W.; Lin, J.H.; Chen, I.W.; Vastag, K.; Anderson, P.S.; Huff, J.R.

Favourites:
ADD

Murayaanthraquinone, a hybrid benz[a]anthraquinone from a UV mutant of streptomyces murayamaensis
pp. 191-194(4)
Authors: Hassan, A.M.; Cone, M.C.; Melville, C.R.; Gould, S.J.

Favourites:
ADD

Access Key

Free Content
Free content
New Content
New content
Open Access Content
Open access content
Subscribed Content
Subscribed content
Free Trial Content
Free trial content
Cookie Policy
X
Cookie Policy
ingentaconnect website makes use of cookies so as to keep track of data that you have filled in. I am Happy with this Find out more