European Journal of Medicinal Chemistry

Syntheses, pharmacological evaluation and molecular modelling of substituted 6-alkoxyimidazo[1,2-b]pyridazines as new ligands for the benzodiazepine receptor
pp. 651-662(12)
Authors: Harrison P.; Barlin G.; Davies L.; Ireland S.; Matyus P.; Wong M.

Synthesis and pharmacological study of new 3,4-dihydro-2H,6H-pyrimido-[2,1-b][1,3]thiazines
pp. 663-668(6)
Authors: Bozsing D.; Sohar P.; Gigler G.; Kovacs G.

Synthesis of 1-(4-acyloxybenzoyloxyacetyl)-4-alkylpiperazines and 1-(4-acyloxybenzoyl)-4-alkylpiperazines as inhibitors of chymotrypsin
pp. 669-674(6)
Authors: Zlatoidsky P.; Maliar T.

Synthesis and testosterone 5-reductase inhibitory activity of 11-substituted 4-aza-5-androstane compounds
pp. 675-681(7)
Authors: Ishibashi K.; Kurata H.; Hamada T.; Horikoshi H.; Kojima K.

Structural optimization of 4-(2-chlorophenyl)-9-methyl-6H-thieno[3,2-f]-[1,2,4]triazolo[4,3-a][1,4]diaz epines as antagonists for platelet activating factor: pharmacological contribution of substituents at the 2- and 6-positions of a condensed ring system
pp. 683-692(10)
Authors: Kawakami Y.; Kitani H.; Yuasa S.; Abe M.; Moriwaki M.; Kagoshima M.; Terasawa M.; Tahara T.

A rational approach to the design of flavones as xanthine oxidase inhibitors
pp. 693-699(7)
Authors: Costantino L.; Rastelli G.; Albasini A.

Molecular simulation of 5,6-substituted 1-[(2-hydroxyethoxy)methyl]uracils with anti-HIV-1 activity
pp. 701-712(12)
Authors: Mager P.; De Clercq E.; Takashima H.; Ubasawa M.; Sekiya K.; Baba M.; Walther H.

Synthesis and ₂-adrenergic activity of 2-[(methyleneamino)oxy]-N-(guanidino)ethaneimines. A biososteric replacement of the aryl of guanabenz-type benzylideneaminoguanidine ₂-agonists with the [(methyleneamino)oxy]methyl moiety (MAOMM)
pp. 713-716(4)
Authors: Balsamo A.; Gentili D.; Macchia M.; Martinotti E.; Rossello A.; Scatizzi R.

New 7-hydroxy-1,3-diazabicyclo[3.3.0]octane derivatives: evaluation of their in vitro immunomodulating effects
pp. 717-723(7)
Authors: Issartel V.; Spehner V.; Bahaji H.; Seilles E.; Couquelet J.

Synthesis and pharmacological properties of 4(5)-(2-ethyl-2,3-dihydro-2-silainden-2-yl)imidazole, a silicon analogue of atipamezole
pp. 725-729(5)
Authors: Heinonen P.; Sipila H.; Neuvonen K.; Lonnberg H.; Cockcroft V.; Wurster S.; Virtanen R.; Savola M.; Salonen J.; Savola J.

Synthesis and antibacterial and antifungal properties of thiazolinoethyl-2-(3H)-benzoxazolone derivatives. II
pp. 731-734(4)
Authors: Erol D.; Aytemir M.; Yulug N.

Synthesis of 1-(isoxazol-3-yl)triazene derivatives. Antimetastatic activity of 3,3-dimethyl-1-(5-methylisoxazol-3-yl)triazene
pp. 735-740(6)
Authors: Tontini A.; Diamantini G.; Balsamini C.; Tarzia G.; Perissin L.; Rapozzi V.

Synthesis of 6-methylimidazo[2,1-b]thiazole derivatives acting on neuromuscular transmission
pp. 741-744(4)
Authors: Andreani A.; Rambaldi M.; Leoni A.; Locatelli A.; Andreani F.; Bossa R.; Chiericozzi M.; Cozzi R.; Galatulas I.