Medicinal Chemistry

Graphical Abstracts
pp. i-vi(6)

Novel Structurally Varied N-Alkyl 1,4-Dihydropyridines as ABCB1 Inhibitors: Structure-Activity Relationships, Biological Activity and First Bioanalytical Evaluation
pp. 487-493(7)
Authors: Hilgeroth, Andreas; Baumert, Christiane; Coburger, Claudius; Seifert, Marianne; Krawczyk, Soren; Hempel, Cornelius; Neubauer, Felix; Krug, Martin; Molnar, Josef; Lage, Hermann

Synthesis and ABCG2 Inhibitory Activity of Novel Fumitremorgin C Analogs – Specificity and Structure Activity Correlations
pp. 494-509(16)
Authors: Szolomajer-Csikos, Orsolya; Beery, Erzsebet; Kosa, Levente; Rajnai, Zsuzsanna; Jani, Marton; Hetenyi, Anasztazia; Tauber Jakab, Katalin; Krajcsi, Peter; K Toth, Gabor

Parallel Synthesis of “Click” Chalcones as Antitubulin Agents
pp. 510-516(7)
Authors: Utsintong, Maleeruk; Massarotti, Alberto; Caldarelli, Antonio; Theeramunkong, Sewan

Antitumor Activity of Novel Benzensulfonamide Derivatives in View of their Physiochemical Properties Searched by Principal Component Analysis
pp. 517-525(9)
Authors: Belka, Mariusz; Slawinski, Jaroslaw; Konieczna, Lucyna; Kawczak, Piotr; Ciesielski, Tomasz; Baczek, Tomasz

Nanosized Tamoxifen-Porphyrin-Glucose [TPG] Conjugate: Novel Selective Anti-breast-cancer Agent, Synthesis and In Vitro Evaluations
pp. 526-538(13)
Authors: Amanlou, Massoud; Heidari, Zahra; Davar Siadat, Seyed; Reza Aghasadeghi, Mohammad; Ghorbani, Masoud; Esmaeil Sadat Ebrahimi, Seyed; Mehdi Sadat, Seyed; Hajmohammadi, Mehdi; Jabbari Arabzadeh, Ali; Hekmat, Soheila; Alaei-Beirami, Mahmood; Azizi Saraji, Alireza; Fathi Moghaddam, Hadi; Shafiee Alavidjeh, Mohammad; Ali Delbaz, Seyed; Dashtbani-Roozbehani, Abolfazl; Shafiee Ardestani, Mehdi

Synthesis of Trans-(4-hydroxypyridine)(Ammine)Dichloroplatinum(II) and its Activity in the Human Ovarian Tumour Models
pp. 539-544(6)
Authors: Deqnah, Narjes; Qing Yu, Jun; Beale, Philip; Fisher, Keith; Huq, Fazlul

The Synthesis, Structural Study and Anticancer Activity Evaluation of Emodin Derivatives Containing Conjugative Groups
pp. 545-552(8)
Authors: Wen-Feng, Wang; Feng-Sen, Zhang; Wen-Na, Zhao; Ze-Dong, Bai; Hui-Jun, Yang; Jing-Wei, Shao; Yao-Feng, Yuan

Computer Aided Discovery of Potential Anti-inflammatory (S)-naproxen Analogs as COX-2 Inhibitors
pp. 553-559(7)
Authors: Manjunathaiah Raghavendra, Nulgumnalli; Ramakrishna, Kota; Sirisha, Vippula; Divya, Pingli; Venkateswara Rao, Alapati

3D-QSAR Modeling of Non-peptide Antagonists for the Human Luteinizing Hormone-releasing Hormone Receptor
pp. 560-570(11)
Authors: Tundidor-Camba, Alain; Caballero, Julio; Coll, Deysma

Imidazole Incorporated Semicarbazone Derivatives as a New Class of Anticonvulsants: Design, Synthesis and In-Vivo Screening
pp. 571-580(10)
Authors: Amir, Mohammad; Ali, Israr; Zaheen Hassan, Mohd.

Synthesis and Biological Evaluation of Novel Pyrimido[4,5-b]quinoline-2,4- dione Derivatives as MDM2 Ubiquitin Ligase Inhibitors
pp. 581-587(7)
Authors: Dou, Xiaoxue; Li, Xin; Tao, Liu; Hu, Chunqi; Zhang, Lei; He, Qiaojun; Yang, Bo; Hu, Yongzhou

Synthesis of Benzophenonehydrazone Schiff Bases and their In Vitro Antiglycating Activities
pp. 588-595(8)
Authors: Mohammed Khan, Khalid; Rahim, Fazal; Ambreen, Nida; Taha, Muhammad; Khan, Momin; Jahan, Humaira; Najeebullah; Shaikh, Azizuddin; Iqbal, Sarosh; Perveen, Shahnaz; Iqbal Choudhary, Muhammad

New Quinolinyl–1,3,4–Oxadiazoles: Synthesis, In Vitro Antibacterial, Antifungal and Antituberculosis Studies
pp. 596-607(12)
Authors: V. Patel, Rahul; Kumari, Premlata; H. Chikhalia, Kishor

In-Silico Analysis of Chromone Containing Sulfonamide Derivatives as Human Carbonic Anhydrase Inhibitors
pp. 608-616(9)
Authors: Ul-Haq, Zaheer; Usmani, Saman; Mahmood, Uzma; al-Rashida, Mariya; Abbas, Ghulam

6-Chloro-7-methyl-3', 4'-dimethoxyflavone - a Potent Selective COX-2 Inhibitor
pp. 617-623(7)
Authors: Bashir, Rafia; Javed, Kalim; Yaseen, Shafiya; Ovais, Syed; Rathore, Pooja; Hamid, Hinna; Alam, M. S.; Samim, Mohammed; Singh, Surender; Nair, Vinod

Investigations Towards New Antidiabetic Drugs from Fungal Endophytes Associated with Salvadora Oleoides Decne
pp. 624-632(9)
Authors: Dhankhar, Seema; Dhankhar, Sandeep; Parkash Yadav, Jaya