Arylboronic Acid-Lead Tetraacetate-Copper Diacetate: A One-Pot System for Copper-Catalyzed N-Arylation Under Neutral Conditions
Abstract:The one-pot reaction of arylboronic acids with lead tetraacetate in chloroform followed by treatment with 3,4-dimethylaniline in the presence of catalytic copper diacetate gave the corresponding diarylamines under neutral conditions in good to high yields. The reaction proceeded with electron-rich as well as with electron-depleted arylboronic derivatives.
Document Type: Review Article
Affiliations: Laboratoire de Valorisation de la Chimie Fine, UMR CNRS 6178; Universite Paul Cezanne - Case 552; Faculte des Sciences St Jerome, 13397 Marseille Cedex 20, France;
Publication date: August 1, 2005
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