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Letters in Drug Design & Discovery publishes original letters on all areas of rational drug design and discovery including medicinal chemistry, in-silico drug design, combinatorial chemistry, high-throughput screening, drug targets, and structure-activity relationships. The emphasis will be on publishing quality papers very rapidly. Letters will be processed rapidly by taking full advantage of Internet technology for both the submission and review of manuscripts. The journal is essential reading to all pharmaceutical scientists involved in research in drug design and discovery.

Publisher: Bentham Science Publishers

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Volume 9, Number 3, March 2012

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Articles

Free Content Graphical Abstracts
pp. i-vi(6)
Author: Bentham Science Publishers,

Manipulating the Ability of Substituted Titanocene Derivatives to Induce Apoptosis in Castrate-Resistant Prostate Cancer Cells
pp. 226-233(8)
Authors: M. Dowling, Catherine; Cuffe, Sandra; Tacke, Matthias; Deally, Anthony; Hogan, Megan; M. Fitzpatrick, John; William G. Watson, R.

Synthesis, Anticancer Activity and Inhibition of Tubulin Polymerization of Bisindole Sulfonates
pp. 242-250(9)
Authors: Kamal, Ahmed; V.V. Srikanth, Y.; Naseer Ahmed Khan, M.; Ashraf, Md.; Basha Shaik, Thokhir; V. Kalivendi, Shasi

Cytotoxic Activity of Polysubstituted 7-chloro-4-quinolinylhydrazone Derivatives
pp. 251-256(6)
Authors: Carvalho Montenegro, Raquel; Veras Lotufo, Leticia; Odorico de Moraes, Manoel; do O Pessoa, Claudia; Augusto Rocha Rodrigues, Felipe; de Lima Ferreira Bispo, Marcelle; Abreu Freire, Bruna; Roland Kaiser, Carlos; Vinicius Nora de Souza, Marcus

Synthesis and Antitumoral Evaluation of Benzyl (1S)-2-[2-(monosubstituted-benzylidene)hydrazino]-1-(hydroxymethyl)-2-oxoethylcarbamate
pp. 257-262(6)
Authors: Carvalho Montenegro, Raquel; Veras Costa Lotufo, Leticia; Odorico de Moraes, Manoel; do O Pessoa, Claudia; Augusto Rocha Rodrigues, Felipe; Campbell Pinheiro, Alessandra; Cristina Mendonça Nogueira, Thais; Vinicius Nora de Souza, Marcus

Carbohydrate Based Blood Antigens in Cancer: Current Status and Future Perspectives
pp. 263-275(13)
Authors: Khalid Yousuf, Syed; Mukherjee, Debaraj; Chandra Taneja, Subhash

Synthesis of New S-alkylated-3-mercapto-1,2,4-triazole Derivatives Bearing Cyclic Amine Moiety as Potent Anticancer Agents
pp. 276-281(6)
Authors: S.R. Murty, M.; R. Ram, Kesur; Venkateswara Rao, Rayudu; S. Yadav, J.; Venkateswara Rao, Janapala; R. Velatooru, L.

Metal Complexes of Uracil Derivatives with Cytotoxicity and Superoxide Scavenging Activity
pp. 282-287(6)
Authors: Prachayasittikul, Supaluk; Worachartcheewan, Apilak; Pingaew, Ratchanok; Suksrichavalit, Thummaruk; Isarankura-Na-Ayudhya, Chartchalerm; Ruchirawat, Somsak; Prachayasittikul, Virapong

The Chemometric Evaluation of Antitumor Activity of Novel Benzensulfonamide Derivatives Based on their Physiochemical Properties
pp. 288-294(7)
Authors: Belka, Mariusz; Konieczna, Lucyna; Kawczak, Piotr; Ciesielski, Tomasz; Slawinski, Jaroslaw; Baczek, Tomasz

Design, Synthesis and Biochemical Evaluation of Estrogen Receptor Ligand Conjugates as Tumour Targeting Agents
pp. 295-304(10)
Authors: O. Keely, Niall; M. Zisterer, Daniela; J. Meegan, Mary

One Pot Synthesis and In Vitro Antitumor Activity of some Bipyrazolic Tripodal Derivatives
pp. 305-309(5)
Authors: Radi, Smaail; Toubi, Yahya; Draoui, Nihed; Feron, Olivier; Riant, Olivier

Synthesis and Biological Evaluation of Some Hydrazone Derivatives as Anti-inflammatory Agents
pp. 310-315(6)
Authors: Asim Kaplancikli, Zafer; Dilek Altintop, Mehlika; Ozdemir, Ahmet; Turan-Zitouni, Gulhan; I. Khan, Shabana; Tabanca, Nurhayat

Synthesis and In Vitro Antibacterial Screening of some New 2,4,6-Trisubstituted-1,3,5-Triazine Derivatives
pp. 316-321(6)
Authors: Bhushan Singh, Ravi; Das, Nirupam; Jana, Srabanti; Das, Aparoop

Calcium Level Controlling Activities of Novel Derivatives of Amlodipine,Riodipine and Cerebrocrast
pp. 322-328(7)
Authors: Vilskersts, R.; Vigante, B.; Neidere, Z.; Krauze, A.; Domracheva, I.; Bekere, L.; Shestakova, I.; Duburs, G.; Dambrova, M.

Design, Facile Synthesis, Antibacterial Activity and Structure-Activity Relationship of Novel Di- and Tri-Substituted 1,3,5-Triazines
pp. 329-335(7)
Authors: Kumar Ghosh, Surajit; Saha, Ashmita; Hazarika, Bornali; Pratap Singh, Udaya; Raj Bhat, Hans; Gahtori, Prashant

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